One-Pot Synthesis, Characterization And Invitro Antimicrobial Activity Of Novel Pyrimidine Derivatives

2021 ◽  
Vol 13 (03) ◽  
Keyword(s):  
Antimicrobial Activity ◽  
Pyrimidine Derivatives ◽  
One Pot ◽  
One Pot Synthesis

Polyoxometalate based ionic crystal: dual applications in selective colorimetric sensor for hydrated ZnCl2 and antimicrobial activity

2021 ◽  
Vol 45 (12) ◽  
pp. 5576-5588
Author(s):  
C. Sabarinathan ◽  
M. Karthikeyan ◽  
R. M. Murugappan ◽  
Savarimuthu Philip Anthony ◽  
Bhaskaran Shankar ◽  
...  
Keyword(s):  
Antimicrobial Activity ◽  
Ionic Crystal ◽  
Colorimetric Sensor ◽  
Icp Oes ◽  
One Pot ◽  
One Pot Synthesis ◽  
Acidic Conditions

One-pot synthesis of POM-salt ([Himi]4[SiMo12O40] (1)) was achieved by mixing silicomolybdic acid and imidazole in acidic conditions and characterized by FTIR, TGA, SEM, EDX, ICP-OES and XPS.

Three-Component, One-Pot Synthesis of Pyrido[2,3-d]pyrimidine Derivatives Catalyzed by KF-Alumina.

ChemInform ◽  
2005 ◽  
Vol 36 (49) ◽  
Author(s):  
Xiang-Shan Wang ◽  
Zhao-Sen Zeng ◽  
Da-Qing Shi ◽  
Shu-Jiang Tu ◽  
Xian-Yong Wei ◽  
...  
Keyword(s):  
Pyrimidine Derivatives ◽  
One Pot ◽  
One Pot Synthesis

scholarly journals Regioselective Green Synthesis and Antimicrobial properties of full fused non mixed Heterocyclic Systems

2017 ◽  
Vol 13 (2) ◽  
pp. 6006-6020
Author(s):  
Amira A. El-Sayed ◽  
Maher El-HAshash ◽  
Sameh Rizk
Keyword(s):  
Antimicrobial Activity ◽  
Green Synthesis ◽  
Elemental Analysis ◽  
Spectroscopic Data ◽  
Heterocyclic Compounds ◽  
Antimicrobial Properties ◽  
One Pot ◽  
One Pot Synthesis ◽  
Electrophilic Reagents

One pot synthesis and reaction of triazinthione and triazinohydrazide derivatives with different electrophilic reagents in ordered to synthesis of some interesting non-mixed heterocyclic compounds. Structures of thiazolotriazine, triazolotriazine, pyrimidinyltriazine, and triazinotriazine derivatives were established via spectroscopic data and elemental analysis. The synthesized compounds were screened for their antimicrobial activity.

scholarly journals A Synthesis of 4-Chloro-2-(trichloromethyl)pyrimidines and Their Study in Nucleophilic Substitution

Synthesis ◽  
2018 ◽  
Vol 51 (02) ◽  
pp. 530-537 ◽  
Author(s):  
Moisés Romero-Ortega ◽  
Michelle Trujillo-Lagunas ◽  
Ignacio Medina-Mercado ◽  
Ivann Zaragoza-Galicia ◽  
Horacio Olivo
Keyword(s):  
Nucleophilic Substitution ◽  
Intramolecular Cyclization ◽  
Nitrogen Heterocycles ◽  
Cyclization Reaction ◽  
Substitution Reactions ◽  
Pyrimidine Derivatives ◽  
One Pot ◽  
Acyl Chlorides ◽  
Nucleophilic Substitution Reactions ◽  
One Pot Synthesis

A convenient two-step, one-pot synthesis of 4-chloro-2-(trichloromethyl)pyrimidines starting from 2-(trichloromethyl)-1,3-diazabutadienes is described. These nitrogen heterocycles were prepared by a sequential acylation/intramolecular cyclization reaction between 2-(trichloromethyl)-1,3-diazabutadienes and acyl chlorides in the presence of triethylamine followed by treatment with POCl3. This is the first report for the synthesis of this type of 4-chloro-2-(trichloromethyl)pyrimidine derivatives and serves as a source for a wide variety of other substituted pyrimidines by nucleophilic substitution reactions.

PTSA-Catalyzed One Pot Domino Synthesis of Dihydropyrido[2,3-d]pyrimidine Derivatives and their Antimicrobial Activity

2021 ◽  
Vol 6 (3) ◽  
pp. 222-227
Author(s):  
Krishna A. Bhensdadia ◽  
Prakash L. Kalavadiya ◽  
Nilam H. Lalavani ◽  
Shipra H. Baluja
Keyword(s):  
Antimicrobial Activity ◽  
Spectral Analysis ◽  
Pyrimidine Derivatives ◽  
One Pot ◽  
In Vitro Antimicrobial Activity ◽  
Aryl Aldehydes ◽  
Three Component Reaction ◽  
The One

A novel series of dihydropyrido[2,3-d]pyrimidine derivatives were synthesized by multicomponent domino cyclization via the one-pot three component reaction of 6-amino uracil, substituted aryl aldehydes and N-methyl-1-(methylthio)-2-nitroethenamine in the presence of PTSA 10 mol% as a catalyst. The structures of these synthesized compounds were characterized by spectral analysis. Further the synthesized compounds screened for in vitro antimicrobial activity. Among all the compounds, compound 4b containing flouro substitution exhibited good inhibition against the tested species.

One-Pot Synthesis of Imidazo[1,5-c]pyrimidine Derivatives from a 4,6-Dichloropyrimidine Derivative and Benzyl Isocyanides

Heterocycles ◽  
2017 ◽  
Vol 94 (1) ◽  
pp. 140 ◽  
Author(s):  
Kazuhiro Kobayashi ◽  
Daiki Fujiwara ◽  
Yuuho Shigemura ◽  
Hidetaka Hiyoshi ◽  
Kazuto Umezu
Keyword(s):  
Pyrimidine Derivatives ◽  
One Pot ◽  
One Pot Synthesis

An efficient one-pot synthesis of pyrazolyl-thiazolidinedione hybrid analogues and evaluation of their antimicrobial activity

2020 ◽  
Vol 29 ◽  
pp. 100507
Author(s):  
Sivaganesh Tummalacharla ◽  
Pannala Padmaja ◽  
Pedavenkatagari Narayana Reddy
Keyword(s):  
Antimicrobial Activity ◽  
One Pot ◽  
One Pot Synthesis
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