Synthesis of oxytocin antagonists containing conformationally constrained amino acids in position 2

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(99)00041-4 ◽

1999 ◽

Vol 9 (5) ◽

pp. 667-672 ◽

Author(s):

Gábor K. Tóth ◽

Krisztina Bakos ◽

Botond Penke ◽

Imre Pávó ◽

Csaba Varga ◽

...

Keyword(s):

Amino Acids ◽

Conformationally Constrained ◽

Oxytocin Antagonists ◽

Conformationally Constrained Amino Acids ◽

Constrained Amino Acids

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ChemInform Abstract: Synthesis and Pharmacological Properties of Oxytocin Antagonists Containing Conformationally Constrained Amino Acids

10.1002/chin.200017275 ◽

2010 ◽

Vol 31 (17) ◽

pp. no-no

Author(s):

G. K. Toth ◽

K. Bakos ◽

I. Zupko ◽

F. Fulop ◽

I. Pavo ◽

...

Keyword(s):

Amino Acids ◽

Pharmacological Properties ◽

Conformationally Constrained ◽

Oxytocin Antagonists ◽

Conformationally Constrained Amino Acids ◽

Constrained Amino Acids

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Synthesis and pharmacological properties of oxytocin antagonists containing conformationally constrained amino acids

Peptide Science — Present and Future ◽

10.1007/0-306-46864-6_247 ◽

2006 ◽

pp. 724-725

Author(s):

G. K. Tóth ◽

K. Bakos ◽

I. Zupkóo ◽

F. FüLöP ◽

I. Pávó ◽

...

Keyword(s):

Amino Acids ◽

Pharmacological Properties ◽

Conformationally Constrained ◽

Oxytocin Antagonists ◽

Conformationally Constrained Amino Acids ◽

Constrained Amino Acids

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Entry to New Conformationally Constrained Amino Acids. First Synthesis of 3-Unsubstituted 4-Alkyl-4-carboxy-2-azetidinone Derivatives via an IntramolecularNα-Cα-Cyclization Strategy

The Journal of Organic Chemistry ◽

10.1021/jo015559b ◽

2001 ◽

Vol 66 (10) ◽

pp. 3538-3547 ◽

Author(s):

Guillermo Gerona-Navarro ◽

Maria Angeles Bonache ◽

Rosario Herranz ◽

Maria Teresa García-López ◽

Rosario González-Muñiz

Keyword(s):

Amino Acids ◽

Conformationally Constrained ◽

Conformationally Constrained Amino Acids ◽

Constrained Amino Acids

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Conformationally Constrained Amino Acids in Peptide Design

SSRN Electronic Journal ◽

10.2139/ssrn.2767061 ◽

2016 ◽

Author(s):

V.S. Saravana Mani ◽

R. Narayanasamy

Keyword(s):

Amino Acids ◽

Peptide Design ◽

Conformationally Constrained ◽

Conformationally Constrained Amino Acids ◽

Constrained Amino Acids

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Incorporation of Conformationally Constrained ?-Amino Acids into Peptides

Journal of Peptide Science ◽

10.1002/1099-1387(200007)6:7<301::aid-psc260>3.0.co;2-1 ◽

2000 ◽

Vol 6 (7) ◽

pp. 301-313 ◽

Author(s):

Michael North

Keyword(s):

Amino Acids ◽

Conformationally Constrained ◽

Conformationally Constrained Amino Acids ◽

Constrained Amino Acids

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ChemInform Abstract: Application of 7-endo, 8-endo and 9-endo Radical Cyclizations to the Synthesis of Conformationally Constrained Amino Acids and Comparison with the Corresponding Heck Reactions.

10.1002/chin.199733208 ◽

2010 ◽

Vol 28 (33) ◽

pp. no-no

Author(s):

S. E. GIBSON ◽

N. GUILLO ◽

M. J. TOZER

Keyword(s):

Amino Acids ◽

Radical Cyclizations ◽

Heck Reactions ◽

Conformationally Constrained ◽

Conformationally Constrained Amino Acids ◽

Constrained Amino Acids

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ChemInform Abstract: Conformationally Constrained Amino Acids: A Convenient Approach to cis-2,3-Methano-GABAs.

10.1002/chin.199929193 ◽

2010 ◽

Vol 30 (29) ◽

pp. no-no

Author(s):

Luca Forti ◽

Franco Ghelfi ◽

Stefano Levizzani ◽

Ugo M. Pagnoni

Keyword(s):

Amino Acids ◽

Conformationally Constrained ◽

Convenient Approach ◽

Conformationally Constrained Amino Acids ◽

Constrained Amino Acids

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Synthesis of Stereodefined Piperidines from Aziridines and Their Transformation into Conformationally Constrained Amino Acids, Amino Alcohols and 2,7-Diazabicyclo[3.3.1]nonanes

The Journal of Organic Chemistry ◽

10.1021/jo101646u ◽

2010 ◽

Vol 75 (22) ◽

pp. 7734-7744 ◽

Author(s):

Karel Vervisch ◽

Matthias D’hooghe ◽

Karl W. Törnroos ◽

Norbert De Kimpe

Keyword(s):

Amino Acids ◽

Amino Alcohols ◽

Conformationally Constrained ◽

Conformationally Constrained Amino Acids ◽

Constrained Amino Acids

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Monitoring of optical isomers of some conformationally constrained amino acids with tetrahydroisoquinoline or tetraline ring structures. Part II

Journal of Chromatography A ◽

10.1016/0021-9673(95)00316-f ◽

1995 ◽

Vol 705 (2) ◽

pp. 257-265 ◽

Author(s):

Antal Péter ◽

Géza Tóth ◽

Edit Olajos ◽

Ferenc Fülöp ◽

Dirk Tourwé

Keyword(s):

Amino Acids ◽

Optical Isomers ◽

Conformationally Constrained ◽

Ring Structures ◽

Conformationally Constrained Amino Acids ◽

Constrained Amino Acids

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Conformationally Constrained Amino Acids.1on the Synthesis of 4-Substituted 8-Membered Cyclic Tryptophan Derivatives

Synthetic Communications ◽

10.1080/00397919208019295 ◽

1992 ◽

Vol 22 (7) ◽

pp. 1039-1048 ◽

Author(s):

John Y. L. Chung ◽

James T. Wasicak ◽

Alex M. Nadzan

Keyword(s):

Amino Acids ◽

Conformationally Constrained ◽

Tryptophan Derivatives ◽

Conformationally Constrained Amino Acids ◽

Constrained Amino Acids

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