Synthesis and Structure—Activity Relationships of 1-Arylmethyl-3-(2-aminopropyl)-5-aryl-6-methyluracils as Potent GnRH Receptor Antagonists.

Synthesis and structure–activity relationships of ( R )-1-alkyl-3-[2-(2-amino)phenethyl]-5-(2-fluorophenyl)-6-methyluracils as human GnRH receptor antagonists

10.1016/j.bmcl.2004.02.004 ◽

2004 ◽

Vol 14 (9) ◽

pp. 2269-2274 ◽

Cited By ~ 14

Author(s):

Martin W Rowbottom ◽

Fabio C Tucci ◽

Yun-Fei Zhu ◽

Zhiqiang Guo ◽

Timothy D Gross ◽

...

Keyword(s):

Gnrh Receptor ◽

Receptor Antagonists ◽

Design, synthesis and structure–Activity relationships of novel imidazolo[1,2-a]pyrimid-5-ones as potent GnRH receptor antagonists

10.1016/s0960-894x(02)00371-2 ◽

2002 ◽

Vol 12 (16) ◽

pp. 2185-2187 ◽

Cited By ~ 16

Author(s):

Timothy D. Gross ◽

Yun-Fei Zhu ◽

John Saunders ◽

Keith M. Wilcoxen ◽

Yinghong Gao ◽

...

Keyword(s):

Gnrh Receptor ◽

Receptor Antagonists ◽

Design Synthesis ◽

A Novel Synthesis of 2-Arylpyrrolo[1,2-a]pyrimid-7-ones and Their Structure–Activity Relationships as Potent GnRH Receptor Antagonists

10.1016/s0960-894x(01)00780-6 ◽

2002 ◽

Vol 12 (3) ◽

pp. 403-406 ◽

Cited By ~ 20

Author(s):

Yun-Fei Zhu ◽

Keith Wilcoxen ◽

John Saunders ◽

Zhiqiang Guo ◽

Yinghong Gao ◽

...

Keyword(s):

Gnrh Receptor ◽

Receptor Antagonists ◽

Novel Synthesis ◽

Design and Structure−Activity Relationships of 2-Alkyl-3-aminomethyl-6-(3-methoxyphenyl)-7-methyl-8-(2-fluorobenzyl)imidazolo[1,2-a]pyrimid-5-ones as Potent GnRH Receptor Antagonists

Journal of Medicinal Chemistry ◽

10.1021/jm0205402 ◽

2003 ◽

Vol 46 (9) ◽

pp. 1769-1772 ◽

Cited By ~ 26

Author(s):

Yun-Fei Zhu ◽

Zhiqiang Guo ◽

Timothy D. Gross ◽

Yinghong Gao ◽

Patrick J. Connors, ◽

...

Keyword(s):

Gnrh Receptor ◽

Receptor Antagonists ◽

ChemInform Abstract: A Novel Synthesis of 2-Arylpyrrolo[1,2-a]pyrimid-7-ones and Their Structure-Activity Relationships as Potent GnRH Receptor Antagonists.

ChemInform ◽

10.1002/chin.200224167 ◽

2010 ◽

Vol 33 (24) ◽

pp. no-no

Author(s):

Yun-Fei Zhu ◽

Chen Chen ◽

et al. et al.

Keyword(s):

Gnrh Receptor ◽

Receptor Antagonists ◽

Novel Synthesis ◽

ChemInform Abstract: Synthesis and Initial Structure-Activity Relationships of a Novel Series of Imidazolo[1,2-a]pyrimid-5-ones as Potent GnRH Receptor Antagonists

ChemInform ◽

10.1002/chin.200249142 ◽

2010 ◽

Vol 33 (49) ◽

pp. no-no

Author(s):

Keith M. Wilcoxen ◽

Yun-Fei Zhu ◽

Patrick J. Connors Jr. ◽

John Saunders ◽

Timothy D. Gross ◽

...

Keyword(s):

Gnrh Receptor ◽

Initial Structure ◽

Receptor Antagonists ◽

Synthesis and Structure?Activity Relationships of Uracil Derived Human GnRH Receptor Antagonists: (R)-3-[2-(2-Amino)phenethyl]-1-(2,6-difluorobenzyl)-6-methyluracils Containing a Substituted Thiophene or Thiazole at C-5.

ChemInform ◽

10.1002/chin.200502158 ◽

2005 ◽

Vol 36 (2) ◽

Author(s):

Martin W. Rowbottom ◽

et al. et al.

Keyword(s):

Gnrh Receptor ◽

Receptor Antagonists ◽

Synthesis and structure–Activity relationships of thieno[2,3- d ]pyrimidine-2,4-dione derivatives as potent GnRH receptor antagonists

10.1016/s0960-894x(03)00746-7 ◽

2003 ◽

Vol 13 (20) ◽

pp. 3617-3622 ◽

Cited By ~ 20

Author(s):

Zhiqiang Guo ◽

Yongsheng Chen ◽

Dongpei Wu ◽

Yun-Fei Zhu ◽

R.Scott Struthers ◽

...

Keyword(s):

Gnrh Receptor ◽

Receptor Antagonists ◽

Synthesis and Structure—Activity Relationships of Thieno[2,3-d]pyrimidine-2,4-dione Derivatives as Potent GnRH Receptor Antagonists.

ChemInform ◽

10.1002/chin.200404228 ◽

2004 ◽

Vol 35 (4) ◽

Author(s):

Zhiqiang Guo ◽

Yongsheng Chen ◽

Dongpei Wu ◽

Yun-Fei Zhu ◽

R. Scott Struthers ◽

...

Keyword(s):

Gnrh Receptor ◽

Receptor Antagonists ◽