Synthesis of Conformationally Constrained Glutamic Acid Homologues and Investigation of Their Pharmacological Profiles

Pharmacological Profiles

ChemInform Abstract: Synthesis of Conformationally Constrained Glutamic Acid Homologues and Investigation of Their Pharmacological Profiles.

ChemInform ◽

10.1002/chin.200810204 ◽

2008 ◽

Vol 39 (10) ◽

Author(s):

Paola Conti ◽

Andrea Pinto ◽

Lucia Tamborini ◽

Giovanni Grazioso ◽

Giovambattista De Sarro ◽

...

Keyword(s):

Glutamic Acid ◽

Pharmacological Profiles

ChemInform Abstract: Synthesis and Pharmacological Evaluation of Novel Conformationally Constrained Homologues of Glutamic Acid.

ChemInform ◽

10.1002/chin.200801185 ◽

2008 ◽

Vol 39 (1) ◽

Author(s):

Paola Conti ◽

Antonio Caligiuri ◽

Andrea Pinto ◽

Gabriella Roda ◽

Lucia Tamborini ◽

...

Keyword(s):

Glutamic Acid ◽

Pharmacological Evaluation

ChemInform Abstract: Synthesis of Some Conformationally-Constrained Glutamate Mimics of N-( 5-(2-(2-Amino-3,4-dihydro-4-oxo-5,6,7,8-tetrahydropyrido(2,3-d) pyrimidin-6-yl)ethyl)thien-2-ylcarbonyl)-L-glutamic Acid (LY254155).

ChemInform ◽

10.1002/chin.199734181 ◽

2010 ◽

Vol 28 (34) ◽

pp. no-no

Author(s):

E. C. TAYLOR ◽

B. HU

Keyword(s):

Glutamic Acid ◽

Synthesis and pharmacological evaluation of novel conformationally constrained homologues of glutamic acid

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2007.01.013 ◽

2007 ◽

Vol 42 (8) ◽

pp. 1059-1068 ◽

Cited By ~ 21

Author(s):

Paola Conti ◽

Antonio Caligiuri ◽

Andrea Pinto ◽

Gabriella Roda ◽

Lucia Tamborini ◽

...

Keyword(s):

Glutamic Acid ◽

Pharmacological Evaluation

Synthesis and pharmacological evaluation of conformationally constrained glutamic acid higher homologues

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2016.09.029 ◽

2016 ◽

Vol 24 (22) ◽

pp. 5741-5747 ◽

Cited By ~ 2

Author(s):

Lucia Tamborini ◽

Gregorio Cullia ◽

Birgitte Nielsen ◽

Carlo De Micheli ◽

Paola Conti ◽

...

Keyword(s):

Glutamic Acid ◽

Pharmacological Evaluation

Kainic acid as conformationally constrained glutamic acid analog in peptide synthesis

Tetrahedron Letters ◽

10.1016/0040-4039(95)02000-f ◽

1995 ◽

Vol 36 (51) ◽

pp. 9309-9312 ◽

Cited By ~ 5

Author(s):

Florinda Artuso ◽

Giovanni Sindona ◽

Constantinos Athanassopoulos ◽

George Stavropoulos ◽

Dionissios Papaioannou

Keyword(s):

Glutamic Acid ◽

Kainic Acid ◽

Peptide Synthesis ◽

Acid Analog

Synthesis of Some Conformationally-constrained Glutamate Mimics of N-{5-[2-amino-3,4-dihydro-4-oxo-5,6,7,8-tetrahydropyrido[2,3-d]pyrimidine-6-yl)ethyl]thien-2-ylcarbonyl-L-glutamic Acid (LY254155)

Heterocycles ◽

10.3987/com-96-7608 ◽

1997 ◽

Vol 45 (2) ◽

pp. 241 ◽

Cited By ~ 7

Author(s):

Edward C. Taylor ◽

Baihua Hu

Keyword(s):

Glutamic Acid ◽

Spiro[2.2]pentane as a Dissymmetric Scaffold for Conformationally Constrained Analogues of Glutamic Acid: Focus on Racemic 1-Aminospiro[2.2]pentyl-1,4-dicarboxylic Acids

The Journal of Organic Chemistry ◽

10.1021/jo020138v ◽

2002 ◽

Vol 67 (16) ◽

pp. 5497-5507 ◽

Cited By ~ 24

Author(s):

Roberto Pellicciari ◽

Maura Marinozzi ◽

Emidio Camaioni ◽

Maria del Carmen Nùnez ◽

Gabriele Costantino ◽

...

Keyword(s):

Glutamic Acid ◽

Dicarboxylic Acids ◽

Synthesis of conformationally-constrained stereospecific analogs of glutamic acid as antagonists of metabotropic receptors

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/0960-894x(95)00457-5 ◽

1995 ◽

Vol 5 (22) ◽

pp. 2627-2632 ◽

Cited By ~ 10

Author(s):

Frédérique Tellier ◽

Francine Acher ◽

Isabelle Brabet ◽

Jean-Philippe Pin ◽

Joël Bockaert ◽

...

Keyword(s):

Glutamic Acid ◽

Metabotropic Receptors ◽

Novel stereocontrolled approach to conformationally constrained analogues of l-glutamic acid and l-proline via stereoselective cyclopropanation of 3,4-didehydro-l-pyroglutamic ABO ester

Tetrahedron ◽

10.1016/j.tet.2005.06.051 ◽

2005 ◽

Vol 61 (35) ◽

pp. 8456-8464 ◽

Cited By ~ 21

Author(s):

Makoto Oba ◽

Naohiro Nishiyama ◽

Kozaburo Nishiyama

Keyword(s):

Glutamic Acid ◽