Design and synthesis of ring-constrained boropeptide thrombin inhibitors

1996 ◽  
Vol 6 (3) ◽  
pp. 295-300 ◽  
Author(s):  
John M. Fevig ◽  
Matthew M. Abelman ◽  
David R. Brittelli ◽  
Charles A. Kettner ◽  
Robert M. Knabb ◽  
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ChemInform Abstract: Design and Synthesis of Conformationally Constrained Arginal Thrombin Inhibitors.

ChemInform ◽  
2010 ◽  
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pp. no-no
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A. SALIMBENI ◽  
F. PALEARI ◽  
R. CANEVOTTI ◽  
M. CRISCUOLI ◽  
A. LIPPI ◽  
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Conformationally Constrained ◽  
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Structure based design and synthesis of novel orally active thrombin inhibitors

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pp. 639-641
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M. Haramura ◽  
T. Shiraishi ◽  
T. Haneishi ◽  
K. Kuromaru ◽  
M. Oota ◽  
...  
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Thrombin Inhibitors ◽  
Design And Synthesis ◽  
Orally Active

Design and synthesis of conformationally constrained arginal thrombin inhibitors

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Vol 7 (17) ◽  
pp. 2205-2210 ◽  
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Aldo Salimbeni ◽  
Fabio Paleari ◽  
Renato Canevotti ◽  
Marco Criscuoli ◽  
Marco Criscuoli ◽  
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Thrombin Inhibitors ◽  
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Heterocyclic thrombin inhibitors. Part 1: design and synthesis of amidino-phenoxy quinoline derivatives

2003 ◽  
Vol 13 (14) ◽  
pp. 2291-2295 ◽  
Author(s):  
Uwe J. Ries ◽  
Henning W.M. Priepke ◽  
Norbert H. Hauel ◽  
Eric E.J. Haaksma ◽  
Jean M. Stassen ◽  
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Design and synthesis of potent and selective macrocyclic thrombin inhibitors

2003 ◽  
Vol 13 (16) ◽  
pp. 2781-2784 ◽  
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Philippe G. Nantermet ◽  
James C. Barrow ◽  
Christina L. Newton ◽  
Janetta M. Pellicore ◽  
MaryBeth Young ◽  
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The design and synthesis of thrombin inhibitors: analogues of MD805 containing non-polar surrogates for arginine at the P1 position

2000 ◽  
Vol 10 (14) ◽  
pp. 1563-1566 ◽  
Author(s):  
Urs Baettig ◽  
Lyndon Brown ◽  
Derek Brundish ◽  
Colin Dell ◽  
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Rational design and synthesis of a novel, selective class of thrombin inhibitors: P1-argininal derivatives incorporating P3P4 quaternary lactam dipeptide surrogates

1997 ◽  
Vol 7 (18) ◽  
pp. 2421-2426 ◽  
Author(s):  
J.Edward Semple ◽  
Nathaniel K. Minami ◽  
Susan Y. Tamura ◽  
Terence K. Brunck ◽  
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Thrombin Inhibitors ◽  
Design And Synthesis
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