Convergent, parallel synthesis of a series of β-substituted 1,2,4-oxadiazole butanoic acids as potent and selective αvβ3 receptor antagonists

2006 ◽  
Vol 16 (4) ◽  
pp. 839-844 ◽  
Author(s):  
Mark L. Boys ◽  
Lori A. Schretzman ◽  
Nizal S. Chandrakumar ◽  
Michael B. Tollefson ◽  
Scott B. Mohler ◽  
...  
Keyword(s):  
Parallel Synthesis ◽  
Receptor Antagonists ◽  
Αvβ3 Receptor

ChemInform Abstract: Parallel Synthesis of a Series of Subtype-Selective NMDA Receptor Antagonists.

ChemInform ◽  
2010 ◽  
Vol 31 (26) ◽  
pp. no-no
Author(s):  
Tracy F. Gregory ◽  
Jon L. Wright ◽  
Lawrence D. Wise ◽  
Leonard T. Meltzer ◽  
Kevin A. Serpa ◽  
...  
Keyword(s):  
Nmda Receptor ◽  
Parallel Synthesis ◽  
Nmda Receptor Antagonists ◽  
Receptor Antagonists ◽  
Subtype Selective

Synthesis of pyrazoles and isoxazoles as potent αvβ3 receptor antagonists

2006 ◽  
Vol 16 (12) ◽  
pp. 3156-3161 ◽  
Author(s):  
Thomas D. Penning ◽  
Albert Khilevich ◽  
Barbara B. Chen ◽  
Mark A. Russell ◽  
Mark L. Boys ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Αvβ3 Receptor

Rapid parallel synthesis applied to the optimization of a series of potent nonpeptide neuropeptide Y-1 receptor antagonists

Tetrahedron ◽  
1999 ◽  
Vol 55 (39) ◽  
pp. 11619-11639 ◽  
Author(s):  
Miles G. Siegel ◽  
Michael O. Chaney ◽  
Robert F. Bruns ◽  
Michael P. Clay ◽  
Douglas A. Schober ◽  
...  
Keyword(s):  
Neuropeptide Y ◽  
Parallel Synthesis ◽  
Receptor Antagonists

Parallel synthesis and SAR study of novel oxa-steroids as potent and selective progesterone receptor antagonists

2007 ◽  
Vol 17 (9) ◽  
pp. 2531-2534 ◽  
Author(s):  
Fu-An Kang ◽  
Jihua Guan ◽  
Nareshkumar Jain ◽  
George Allan ◽  
Olivia Linton ◽  
...  
Keyword(s):  
Progesterone Receptor ◽  
Parallel Synthesis ◽  
Receptor Antagonists ◽  
Sar Study

Highly potent and selective αVβ3-receptor antagonists: solid-phase synthesis and SAR of 1-substituted 4-amino-1H-pyrimidin-2-ones

2003 ◽  
Vol 13 (2) ◽  
pp. 165-169 ◽  
Author(s):  
Christian Zechel ◽  
Gisela Backfisch ◽  
Jürgen Delzer ◽  
Hervé Geneste ◽  
Claudia Graef ◽  
...  
Keyword(s):  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Receptor Antagonists ◽  
Phase Synthesis ◽  
Αvβ3 Receptor

Discovery and SAR of 4-amino-2-biarylbutylurea MCH 1 receptor antagonists through solid-phase parallel synthesis

2005 ◽  
Vol 15 (16) ◽  
pp. 3691-3695 ◽  
Author(s):  
Tao Guo ◽  
Rachael C. Hunter ◽  
Huizhong Gu ◽  
Laura L. Rokosz ◽  
Tara M. Stauffer ◽  
...  
Keyword(s):  
Solid Phase ◽  
Parallel Synthesis ◽  
Receptor Antagonists

Parallel synthesis of a series of subtype-selective NMDA receptor antagonists

2000 ◽  
Vol 10 (6) ◽  
pp. 527-529 ◽  
Author(s):  
Tracy F. Gregory ◽  
Jon L. Wright ◽  
Lawrence D. Wise ◽  
Leonard T. Meltzer ◽  
Kevin A. Serpa ◽  
...  
Keyword(s):  
Nmda Receptor ◽  
Parallel Synthesis ◽  
Nmda Receptor Antagonists ◽  
Receptor Antagonists ◽  
Subtype Selective

Synthesis of Pyrazoles and Isoxazoles as Potent αvβ3 Receptor Antagonists.

ChemInform ◽  
2006 ◽  
Vol 37 (37) ◽  
Author(s):  
Thomas D. Penning ◽  
et al. et al.
Keyword(s):  
Receptor Antagonists ◽  
Αvβ3 Receptor
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