Potential Irreversible Ligands for Opioid Receptors. Cinnamoyl Derivatives of β-Naltrexamine

1996 ◽  
Vol 48 (2) ◽  
pp. 192-196 ◽  
Author(s):  
IAN DERRICK ◽  
JOHN W. LEWIS ◽  
HUMPHREY A. MOYNIHAN ◽  
JILLIAN BROADBEAR ◽  
JAMES H. WOODS
Keyword(s):  
Opioid Receptors ◽  
Derivatives Of

Synthesis and evaluation of derivatives of leucine enkephalin as potential affinity labels for δ opioid receptors

Biopolymers ◽  
2003 ◽  
Vol 71 (5) ◽  
pp. 552-557 ◽  
Author(s):  
Heekyung Choi ◽  
Thomas F. Murray ◽  
Jane V. Aldrich
Keyword(s):  
Opioid Receptors ◽  
Affinity Labels ◽  
Leucine Enkephalin ◽  
Derivatives Of

scholarly journals New psychoactive substances: psychiatrist's view

2019 ◽  
pp. 57-67
Author(s):  
Andrey Viktorovich Antsyborov ◽  
Irina Vladimirovna Dubatova
Keyword(s):  
Opioid Receptors ◽  
Psychotic Disorders ◽  
Synthetic Cannabinoids ◽  
Designer Drugs ◽  
New Psychoactive Substances ◽  
Psychoactive Substances ◽  
Gaba A ◽  
Psychoactive Effects ◽  
Legal High ◽  
Derivatives Of

Appearing not long ago, new psychoactive substances (designer drugs), including synthetic cannabinoids, derivatives of cathinone, phenethylamines, new stimulants, synthetic opioids, tryptamine derivatives, phencyclidine, piperazine, the GABA (A/B) receptors agonists, have become a serious problem for consumers and for physicians. Consumers of these substances are attracted primarily by the intensity of psychoactive effects, and the «legal high» declared by the black manufacturers, which indicates that significant difficulties in a laboratory identification of new surfactants. Designer drugs, when ingested, can be influenced on many neurotransmitter pathways/receptors: dopamine, cannabinoid (CB1), GABA (A/B), 5-HT2A, glutamate, and k-opioid receptors (KOR), the imbalance of which leads to the development of polymorphic psychotic disorders.

Persistent binding of fatty acyl derivatives of naltrexamine to opioid receptors

1991 ◽  
Vol 34 (7) ◽  
pp. 1966-1969 ◽  
Author(s):  
P. S. Portoghese ◽  
A. Garzon-Aburbeh ◽  
D. L. Larson
Keyword(s):  
Opioid Receptors ◽  
Fatty Acyl ◽  
Derivatives Of ◽  
Acyl Derivatives

Interaction of newly synthesized N-cyclopropylmethyl derivatives of (−)-6β-acetylthionormorphine with opioid receptors

1990 ◽  
Vol 21 (4) ◽  
pp. 541-546 ◽  
Author(s):  
I. Takayanagi ◽  
N. Goromaru ◽  
K. Koike ◽  
F. Konno ◽  
T. Mori ◽  
...  
Keyword(s):  
Opioid Receptors ◽  
Derivatives Of

N-Terminal alkylated derivatives of [D-Pro10]dynorphin A-(1-11) are highly selective for .kappa.-opioid receptors

1992 ◽  
Vol 35 (24) ◽  
pp. 4638-4639 ◽  
Author(s):  
Heekyung Choi ◽  
Thomas F. Murray ◽  
Gary E. DeLander ◽  
Valerie Caldwell ◽  
Jane V. Aldrich
Keyword(s):  
Opioid Receptors ◽  
Kappa Opioid Receptors ◽  
Dynorphin A ◽  
Kappa Opioid ◽  
Derivatives Of

7-Spiroindanyl Derivatives of Naltrexone and Oxymorphone as Selective Ligands for δ Opioid Receptors

1997 ◽  
Vol 40 (11) ◽  
pp. 1720-1725 ◽  
Author(s):  
S. Ohkawa ◽  
B. DiGiacomo ◽  
D. L. Larson ◽  
A. E. Takemori ◽  
P. S. Portoghese
Keyword(s):  
Opioid Receptors ◽  
Selective Ligands ◽  
Derivatives Of

Analgesic activity and selectivity of isothiocyanate derivatives of fentanyl analogs for opioid receptors

Life Sciences ◽  
1999 ◽  
Vol 65 (15) ◽  
pp. 1589-1595 ◽  
Author(s):  
Chen Bi-Yi ◽  
Jin Wen-Qiao ◽  
Chen Jie ◽  
Chen Xin-Jian ◽  
Zhu You-Cheng ◽  
...  
Keyword(s):  
Opioid Receptors ◽  
Analgesic Activity ◽  
Fentanyl Analogs ◽  
Derivatives Of
Sign in / Sign up

Export Citation Format

Share Document