ChemInform Abstract: Design, Synthesis, and Structure-Activity Relationships of Phthalimide-Phenylpiperazines: A Novel Series of Potent and Selective α1a-Adrenergic Receptor Antagonists.

Design, Synthesis, and Structure−Activity Relationships of Phthalimide-Phenylpiperazines: A Novel Series of Potent and Selective α1a-Adrenergic Receptor Antagonists

Journal of Medicinal Chemistry ◽

10.1021/jm9905918 ◽

2000 ◽

Vol 43 (11) ◽

pp. 2183-2195 ◽

Cited By ~ 25

Author(s):

Gee-Hong Kuo ◽

Catherine Prouty ◽

William V. Murray ◽

Virginia Pulito ◽

Linda Jolliffe ◽

...

Keyword(s):

Adrenergic Receptor ◽

Receptor Antagonists ◽

Design Synthesis ◽

Nonpeptide angiotensin II receptor antagonists. 2. Design, synthesis, and structure-activity relationships of 2-alkyl-4-(1H-pyrrol-l-yl)-1H-imidazole derivatives: profile of 2-propyl-1-[[2'-(1H-tetrazol-5-yl)-[1,1'-biphenyl]-4-yl]-methyl]-4-[2-(trifluoroacetyl)-1H-pyrrol-1-yl]-1H-imidazole-5-carboxylic acid (CI-996)

Journal of Medicinal Chemistry ◽

10.1021/jm00068a002 ◽

1993 ◽

Vol 36 (16) ◽

pp. 2253-2265 ◽

Cited By ~ 9

Author(s):

Ila Sircar ◽

John C. Hodges ◽

John Quin ◽

Amy M. Bunker ◽

R. Thomas Winters ◽

...

Keyword(s):

Angiotensin Ii ◽

Carboxylic Acid ◽

Angiotensin Ii Receptor ◽

Angiotensin Ii Receptor Antagonists ◽

Receptor Antagonists ◽

Design Synthesis ◽

Imidazole Derivatives ◽

Corrigendum to “Design, synthesis, and structure–activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin receptor antagonists” [Bioorg. Med. Chem. 22 (2014) 6071–6088]

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2015.04.042 ◽

2015 ◽

Vol 23 (13) ◽

pp. 3870

Author(s):

Yu Yoshida ◽

Taro Terauchi ◽

Yoshimitsu Naoe ◽

Yuji Kazuta ◽

Fumihiro Ozaki ◽

...

Keyword(s):

Receptor Antagonists ◽

Design Synthesis ◽

Structure Activity ◽

Orally Active

Design, synthesis and structure–Activity relationships of novel imidazolo[1,2-a]pyrimid-5-ones as potent GnRH receptor antagonists

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(02)00371-2 ◽

2002 ◽

Vol 12 (16) ◽

pp. 2185-2187 ◽

Cited By ~ 16

Author(s):

Timothy D. Gross ◽

Yun-Fei Zhu ◽

John Saunders ◽

Keith M. Wilcoxen ◽

Yinghong Gao ◽

...

Keyword(s):

Gnrh Receptor ◽

Receptor Antagonists ◽

Design Synthesis ◽

Rational Design, Synthesis, and Structure−Activity Relationships of Aryltriazoles as Novel Corticotropin-Releasing Factor-1 Receptor Antagonists

Journal of Medicinal Chemistry ◽

10.1021/jm049339c ◽

2005 ◽

Vol 48 (5) ◽

pp. 1540-1549 ◽

Cited By ~ 16

Author(s):

Richard F. Lowe ◽

Jodene Nelson ◽

Trunghau N. Dang ◽

Paul D. Crowe ◽

Anil Pahuja ◽

...

Keyword(s):

Rational Design ◽

Corticotropin Releasing Factor ◽

Receptor Antagonists ◽

Design Synthesis ◽

Design, synthesis, and structure–activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin receptor antagonists

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2014.08.034 ◽

2014 ◽

Vol 22 (21) ◽

pp. 6071-6088 ◽

Cited By ~ 12

Author(s):

Yu Yoshida ◽

Taro Terauchi ◽

Yoshimitsu Naoe ◽

Yuji Kazuta ◽

Fumihiro Ozaki ◽

...

Keyword(s):

Receptor Antagonists ◽

Design Synthesis ◽

Structure Activity ◽

Orally Active

Design, synthesis and structure–activity relationships of 5-alkylaminolquinolines as a novel series of CRF1 receptor antagonists

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2012.05.066 ◽

2012 ◽

Vol 22 (14) ◽

pp. 4756-4761 ◽

Cited By ~ 6

Author(s):

Kunitoshi Takeda ◽

Taro Terauchi ◽

Kogyoku Shin ◽

Mitsuhiro Ino ◽

Hisashi Shibata ◽

...

Keyword(s):

Receptor Antagonists ◽

Design Synthesis ◽

Crf1 Receptor ◽

ChemInform Abstract: Nonpeptide Angiotensin II Receptor Antagonists. Part 2. Design, Synthesis, and Structure-Activity Relationships of 2-Alkyl-4-(1H-pyrrol-1-yl)-1H-imidazole Derivatives: Profile of 2-Propyl-1-((2′-(1H-tetrazol-5-yl)-(1,1′-biphenyl)-4-yl

ChemInform ◽

10.1002/chin.199352180 ◽

2010 ◽

Vol 24 (52) ◽

pp. no-no

Author(s):

I. SIRCAR ◽

J. C. HODGES ◽

J. III QUIN ◽

A. M. BUNKER ◽

R. T. WINTERS ◽

...

Keyword(s):

Angiotensin Ii ◽

Angiotensin Ii Receptor ◽

Angiotensin Ii Receptor Antagonists ◽

Receptor Antagonists ◽

Design Synthesis ◽

Imidazole Derivatives ◽

ChemInform Abstract: Design, Synthesis, and Structure-Activity Relationships of Novel Non-Imidazole Histamine H3 Receptor Antagonists.

ChemInform ◽

10.1002/chin.200040113 ◽

2000 ◽

Vol 31 (40) ◽

pp. no-no

Author(s):

Ian D. Linney ◽

Ildiko M. Buck ◽

Elaine A. Harper ◽

S. Barret-Kalindjian ◽

Michael J. Pether ◽

...

Keyword(s):

Receptor Antagonists ◽

Design Synthesis ◽

Histamine H3 Receptor ◽

Structure Activity ◽

H3 Receptor ◽

Histamine H3

Design, synthesis, structure–activity relationships, and docking studies of pyrazole-containing derivatives as a novel series of potent glucagon receptor antagonists

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2016.04.053 ◽

2016 ◽

Vol 24 (12) ◽

pp. 2852-2863 ◽

Cited By ~ 9

Author(s):

Shuangjie Shu ◽

Xiaoqing Cai ◽

Jia Li ◽

Yang Feng ◽

Antao Dai ◽

...

Keyword(s):

Docking Studies ◽

Receptor Antagonists ◽

Glucagon Receptor ◽

Design Synthesis ◽