Comparison of the structure-activity relationships of melatonin receptor agonists and antagonists: lengthening the N-acyl side-chain has differing effects on potency on Xenopus melanophores

1998 ◽  
Vol 358 (5) ◽  
pp. 522-528 ◽  
Author(s):  
M.-T. Teh ◽  
D. Sugden
Keyword(s):  
Side Chain ◽  
Melatonin Receptor ◽  
Structure Activity Relationships ◽  
Receptor Agonists ◽  
Structure Activity ◽  
Acyl Side Chain ◽  
Melatonin Receptor Agonists ◽  
Receptor Agonists And Antagonists

scholarly journals Fluorine substituted methoxyphenylalkyl amides as potent melatonin receptor agonists

MedChemComm ◽  
2019 ◽  
Vol 10 (3) ◽  
pp. 460-464 ◽  
Author(s):  
Andrew Tsotinis ◽  
Rodanthi Kompogennitaki ◽  
Ioannis Papanastasiou ◽  
Peter J. Garratt ◽  
Alina Bocianowska ◽  
...  
Keyword(s):  
Side Chain ◽  
Melatonin Receptor ◽  
Receptor Agonists ◽  
Methoxy Groups ◽  
Melatonin Receptor Agonists

A series of fluorine substituted methoxyphenylalkyl amides were prepared with different orientations of the fluorine and methoxy groups with respect to the alkylamide side chain and with alkyl sides of differing lengths (n= 1–3).

Structure Activity Relationships of P2 Receptor Agonists and Antagonists

1998 ◽  
pp. 81-107 ◽  
Author(s):  
Kenneth A. Jacobson ◽  
Yong-Chul Kim ◽  
Emidio Camaioni ◽  
A. Michiel van Rhee
Keyword(s):  
P2 Receptor ◽  
Structure Activity Relationships ◽  
Receptor Agonists ◽  
Structure Activity ◽  
Receptor Agonists And Antagonists

Synthesis and structure–activity relationship of novel benzoxazole derivatives as melatonin receptor agonists

2004 ◽  
Vol 14 (14) ◽  
pp. 3799-3802 ◽  
Author(s):  
Li-Qiang Sun ◽  
Jie Chen ◽  
Marc Bruce ◽  
Jeffrey A Deskus ◽  
James R Epperson ◽  
...  
Keyword(s):  
Structure Activity Relationship ◽  
Activity Relationship ◽  
Melatonin Receptor ◽  
Receptor Agonists ◽  
Structure Activity ◽  
Melatonin Receptor Agonists ◽  
Relationship Of
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