Design, synthesis and biological evaluation of triaryl compounds as novel 20S proteasome inhibitors

2020 ◽  
Vol 30 (21) ◽  
pp. 127508
Author(s):  
Yajun Yang ◽  
Ke Wang ◽  
Bo Wu ◽  
Ying Yang ◽  
Fangfang Lai ◽  
...  
Keyword(s):  
Proteasome Inhibitors ◽  
Biological Evaluation ◽  
20S Proteasome ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation

Convergent Synthesis and Biological Evaluation of Syringolin A and Derivatives as Eukaryotic 20S Proteasome Inhibitors

2010 ◽  
Vol 2010 (21) ◽  
pp. 3991-4003 ◽  
Author(s):  
Jérôme Clerc ◽  
Barbara Schellenberg ◽  
Michael Groll ◽  
André S. Bachmann ◽  
Robert Huber ◽  
...  
Keyword(s):  
Proteasome Inhibitors ◽  
Biological Evaluation ◽  
20S Proteasome ◽  
Convergent Synthesis ◽  
Synthesis And Biological Evaluation

Design, synthesis and biological evaluation of tripeptide boronic acid proteasome inhibitors

2009 ◽  
Vol 17 (19) ◽  
pp. 6851-6861 ◽  
Author(s):  
Yongqiang Zhu ◽  
Shuyang Yao ◽  
Bo Xu ◽  
Zemei Ge ◽  
Jingrong Cui ◽  
...  
Keyword(s):  
Boronic Acid ◽  
Proteasome Inhibitors ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation

Psoralenquinones as a Novel Class of Proteasome Inhibitors: Design, Synthesis and Biological Evaluation

ChemMedChem ◽  
2011 ◽  
Vol 6 (6) ◽  
pp. 996-1000 ◽  
Author(s):  
Giovanni Marzaro ◽  
Valentina Gandin ◽  
Christine Marzano ◽  
Adriano Guiotto ◽  
Adriana Chilin
Keyword(s):  
Proteasome Inhibitors ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation

Design, Synthesis and Biological Evaluation of Peptidyl Epoxyketone Proteasome Inhibitors Composed ofβ-amino Acids

2014 ◽  
Vol 84 (5) ◽  
pp. 497-504 ◽  
Author(s):  
Jiankang Zhang ◽  
Mengmeng Han ◽  
Xiaodong Ma ◽  
Lei Xu ◽  
Jiayi Cao ◽  
...  
Keyword(s):  
Amino Acids ◽  
Proteasome Inhibitors ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation
Sign in / Sign up

Export Citation Format

Share Document