Synthesis and biological evaluation of some thiazolyl and thiadiazolyl derivatives of 1H-pyrazole as anti-inflammatory antimicrobial agents

Adnan A. Bekhit; Hayam M.A. Ashour; Yasser S. Abdel Ghany; Alaa El-Din A. Bekhit; Azza Baraka

doi:10.1016/j.ejmech.2007.03.030

Synthesis and biological evaluation of some thiazolyl and thiadiazolyl derivatives of 1H-pyrazole as anti-inflammatory antimicrobial agents

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2007.03.030 ◽

2008 ◽

Vol 43 (3) ◽

pp. 456-463 ◽

Cited By ~ 183

Author(s):

Adnan A. Bekhit ◽

Hayam M.A. Ashour ◽

Yasser S. Abdel Ghany ◽

Alaa El-Din A. Bekhit ◽

Azza Baraka

Keyword(s):

Antimicrobial Agents ◽

Biological Evaluation ◽

Anti Inflammatory ◽

Synthesis And Biological Evaluation ◽

Derivatives Of

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Synthesis and biological evaluation of diamide derivatives of (S)-BINOL and biphenyl as potential anti-inflammatory/anti-arthritic agents

Medicinal Chemistry Research ◽

10.1007/s00044-012-0410-6 ◽

2012 ◽

Vol 22 (9) ◽

pp. 4164-4172 ◽

Cited By ~ 2

Author(s):

Raj Rajadurai ◽

Ramar Padmanabhan ◽

Sarkkarai Ananthan

Keyword(s):

Biological Evaluation ◽

Anti Inflammatory ◽

Synthesis And Biological Evaluation ◽

Derivatives Of

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Synthesis and biological evaluation of pyrazolylthiazole carboxylic acids as potent anti-inflammatory–antimicrobial agents

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2015.02.004 ◽

2015 ◽

Vol 25 (6) ◽

pp. 1177-1181 ◽

Cited By ~ 24

Author(s):

Poonam Khloya ◽

Satish Kumar ◽

Pawan Kaushik ◽

Parveen Surain ◽

Dhirender Kaushik ◽

...

Keyword(s):

Carboxylic Acids ◽

Antimicrobial Agents ◽

Biological Evaluation ◽

Anti Inflammatory ◽

Synthesis And Biological Evaluation

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ChemInform Abstract: Synthesis and Biological Evaluation of Some Thiazolyl and Thiadiazolyl Derivatives of 1H-Pyrazole and Antiinflammatory Antimicrobial Agents.

ChemInform ◽

10.1002/chin.200830120 ◽

2008 ◽

Vol 39 (30) ◽

Author(s):

Adnan A. Bekhit ◽

Hayam M. A. Ashour ◽

Yasser S. Abdel Ghany ◽

Alaa El-Din A. Bekhit ◽

Azza Baraka

Keyword(s):

Antimicrobial Agents ◽

Biological Evaluation ◽

Synthesis And Biological Evaluation ◽

Derivatives Of

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Pyrazolylbenzyltriazoles as cyclooxygenase inhibitors: synthesis and biological evaluation as dual anti-inflammatory and antimicrobial agents

New Journal of Chemistry ◽

10.1039/c4nj00226a ◽

2014 ◽

Vol 38 (8) ◽

pp. 3662 ◽

Cited By ~ 14

Author(s):

Nisha Chandna ◽

Jitander K. Kapoor ◽

Jagdeep Grover ◽

Khemraj Bairwa ◽

Varsha Goyal ◽

...

Keyword(s):

Antimicrobial Agents ◽

Biological Evaluation ◽

Cyclooxygenase Inhibitors ◽

Anti Inflammatory ◽

Synthesis And Biological Evaluation

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Synthesis and Biological Evaluation of Amide Derivatives of (6-Chloro-2,3-dihydro-1H-inden-1-yl)acetic Acid as Potential Anti-inflammatory Agents with Lower Gastrointestinal Toxicity

Chemical and Pharmaceutical Bulletin ◽

10.1248/cpb.56.626 ◽

2008 ◽

Vol 56 (5) ◽

pp. 626-634 ◽

Cited By ~ 8

Author(s):

Meenakshi Sharma ◽

Saumendra Mohan Ray

Keyword(s):

Acetic Acid ◽

Biological Evaluation ◽

Gastrointestinal Toxicity ◽

Amide Derivatives ◽

Anti Inflammatory ◽

Synthesis And Biological Evaluation ◽

Derivatives Of

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Synthesis and biological evaluation of some thiazolylpyrazole derivatives as dual anti-inflammatory antimicrobial agents

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2010.10.001 ◽

2010 ◽

Vol 45 (12) ◽

pp. 6027-6038 ◽

Cited By ~ 52

Author(s):

Adnan A. Bekhit ◽

Hesham T.Y. Fahmy ◽

Sherif A.F. Rostom ◽

Alaa El-Din A. Bekhit

Keyword(s):

Antimicrobial Agents ◽

Biological Evaluation ◽

Anti Inflammatory ◽

Synthesis And Biological Evaluation

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Synthesis and biological evaluation of amide derivatives of (5,6-dimethoxy-2,3-dihydro-1H-inden-1-yl)acetic acid as anti-inflammatory agents with reduced gastrointestinal ulcerogenecity

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2007.08.008 ◽

2008 ◽

Vol 43 (10) ◽

pp. 2092-2102 ◽

Cited By ~ 16

Author(s):

Meenakshi Sharma ◽

S.M. Ray

Keyword(s):

Acetic Acid ◽

Biological Evaluation ◽

Amide Derivatives ◽

Anti Inflammatory ◽

Synthesis And Biological Evaluation ◽

Derivatives Of

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Synthesis and Biological Evaluation of Derivatives of 2-{2-Fluoro-4-[(2-oxocyclopentyl)methyl]phenyl}propanoic Acid: Nonsteroidal Anti-Inflammatory Drugs with Low Gastric Ulcerogenic Activity

Journal of Medicinal Chemistry ◽

10.1021/jm300049g ◽

2012 ◽

Vol 55 (11) ◽

pp. 5143-5150 ◽

Cited By ~ 17

Author(s):

Naoki Yamakawa ◽

Shintaro Suemasu ◽

Yoshinari Okamoto ◽

Ken-ichiro Tanaka ◽

Tomoaki Ishihara ◽

...

Keyword(s):

Biological Evaluation ◽

Propanoic Acid ◽

Ulcerogenic Activity ◽

Inflammatory Drugs ◽

Anti Inflammatory ◽

Synthesis And Biological Evaluation ◽

Derivatives Of ◽

Methyl Phenyl

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Synthesis and biological evaluation of some novel urea and thiourea derivatives of isoxazolo[4,5-d]pyridazine and structurally related thiazolo[4,5-d]pyridazine as antimicrobial agents

Archives of Pharmacal Research ◽

10.1007/s12272-013-0144-0 ◽

2013 ◽

Vol 36 (11) ◽

pp. 1354-1368 ◽

Cited By ~ 16

Author(s):

Hassan M. Faidallah ◽

Sherif A. F. Rostom ◽

Salem A. Basaif ◽

Mohammed S. T. Makki ◽

Khalid A. Khan

Keyword(s):

Antimicrobial Agents ◽

Biological Evaluation ◽

Thiourea Derivatives ◽

Synthesis And Biological Evaluation ◽

Derivatives Of

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Synthesis and biological evaluation of a novel series of 2,2-bisaminomethylated aurone analogues as anti-inflammatory and antimicrobial agents

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2010.03.045 ◽

2010 ◽

Vol 45 (7) ◽

pp. 3223-3227 ◽

Cited By ~ 52

Author(s):

Babasaheb P. Bandgar ◽

Sachin A. Patil ◽

Balaji L. Korbad ◽

Satish C. Biradar ◽

Shivraj N. Nile ◽

...

Keyword(s):

Antimicrobial Agents ◽

Biological Evaluation ◽

Anti Inflammatory ◽

Synthesis And Biological Evaluation

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