Solid phase synthesis of sec-amides and removal from the polymeric support under mild conditions

1997 ◽  
Vol 38 (42) ◽  
pp. 7325-7328 ◽  
Author(s):  
D. Sarantakis ◽  
J.J. Bicksler
ChemInform ◽  
1990 ◽  
Vol 21 (20) ◽  
Author(s):  
E. BARDAJI ◽  
J. L. TORRES ◽  
P. CLAPES ◽  
F. ALBERICIO ◽  
G. BARANY ◽  
...  

Peptides ◽  
1988 ◽  
pp. 159-161 ◽  
Author(s):  
Fernando Albericio ◽  
Nancy Kneib-Cordonier ◽  
Lajos Gera ◽  
Robert P. Hammer ◽  
Derek Hudson ◽  
...  

1990 ◽  
Vol 29 (3) ◽  
pp. 291-292 ◽  
Author(s):  
Eduard Bardají ◽  
Josep L. Torres ◽  
Pere Clapés ◽  
Fernando Albericio ◽  
George Barany ◽  
...  

2003 ◽  
Vol 2003 (9) ◽  
pp. 599-600
Author(s):  
Jing Tang ◽  
Xian Huang

The resin-bound 5-monosubstituted cyclic malonic ester 3 was generated and reacted with an α–bromoketone to give the corresponding 5,5-disubstituted cyclic malonic ester resin (4). Subsequent reaction with hydrazine resulted in cyclisation with concomitant cleavage from the polymeric support to release the final products, 4,6-disubstituted 4,5-dihydro-3(2 H)-pyridazinones, in good yield and high purity.


1996 ◽  
Vol 37 (47) ◽  
pp. 8589-8592 ◽  
Author(s):  
Markus Gude ◽  
Umberto Piarulli ◽  
Donatella Potenza ◽  
Barbara Salom ◽  
Cesare Gennari

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