Identification of 6-Hydroxypyrimidin-4(1H)-one-3-carboxamides as Potent and Orally Active APJ Receptor Agonists

2021 ◽  
Author(s):  
Zulan Pi ◽  
James A. Johnson ◽  
Wei Meng ◽  
Monique Phillips ◽  
William A. Schumacher ◽  
...  
Keyword(s):  
Receptor Agonists ◽  
Orally Active

(S)- and (R)-8-(di-n-propylamino)-6,7,8,9-tetrahydro-3H-benz[e]indole-1-carbaldehyde: a new class of orally active 5-HT1A-receptor agonists

1993 ◽  
Vol 36 (15) ◽  
pp. 2059-2065 ◽  
Author(s):  
Peter Stjernloef ◽  
Maria Gullme ◽  
Thomas Elebring ◽  
Bengt Andersson ◽  
Haakan Wikstroem ◽  
...  
Keyword(s):  
Receptor Agonists ◽  
New Class ◽  
Orally Active

Preparation, Resolution, and Biological Evaluation of 5-Aryl-1,2-dihydro-5H-chromeno[3,4-f]quinolines:  Potent, Orally Active, Nonsteroidal Progesterone Receptor Agonists

1998 ◽  
Vol 41 (15) ◽  
pp. 2779-2785 ◽  
Author(s):  
James P. Edwards ◽  
Lin Zhi ◽  
Charlotte L. F. Pooley ◽  
Christopher M. Tegley ◽  
Sarah J. West ◽  
...  
Keyword(s):  
Progesterone Receptor ◽  
Biological Evaluation ◽  
Receptor Agonists ◽  
Orally Active

scholarly journals Benzofuran Derivatives as Potent, Orally Active S1P1 Receptor Agonists: A Preclinical Lead Molecule for MS

2010 ◽  
Vol 2 (2) ◽  
pp. 97-101 ◽  
Author(s):  
Ashis K. Saha ◽  
Xiang Yu ◽  
Jian Lin ◽  
Mercedes Lobera ◽  
Anurag Sharadendu ◽  
...  
Keyword(s):  
Receptor Agonists ◽  
S1p1 Receptor ◽  
Orally Active

Enhanced Gastrointestinal Motility with Orally Active Ghrelin Receptor Agonists

2009 ◽  
Vol 329 (3) ◽  
pp. 1178-1186 ◽  
Author(s):  
Soratree Charoenthongtrakul ◽  
Derek Giuliana ◽  
Kenneth A. Longo ◽  
Elizabeth K. Govek ◽  
Anna Nolan ◽  
...  
Keyword(s):  
Gastrointestinal Motility ◽  
Ghrelin Receptor ◽  
Receptor Agonists ◽  
Orally Active

5-Aryl-1,2-dihydro-5H-chromeno[3,4-f]quinolines as Potent, Orally Active, Nonsteroidal Progesterone Receptor Agonists:  The Effect of D-Ring Substituents

1998 ◽  
Vol 41 (3) ◽  
pp. 303-310 ◽  
Author(s):  
James P. Edwards ◽  
Sarah J. West ◽  
Keith B. Marschke ◽  
Dale E. Mais ◽  
Marco M. Gottardis ◽  
...  
Keyword(s):  
Progesterone Receptor ◽  
Receptor Agonists ◽  
Orally Active

Discovery of Diphenylcarbamate Derivatives as Highly Potent and Selective IP Receptor Agonists: Orally Active Prostacyclin Mimetics. Part 3.

ChemInform ◽  
2005 ◽  
Vol 36 (44) ◽  
Author(s):  
Kouji Hattori ◽  
Akira Tanaka ◽  
Osamu Okitsu ◽  
Seiichiro Tabuchi ◽  
Kiyoshi Taniguchi ◽  
...  
Keyword(s):  
Receptor Agonists ◽  
Ip Receptor ◽  
Orally Active

Discovery of diphenylcarbamate derivatives as highly potent and selective IP receptor agonists: Orally active prostacyclin mimetics. Part 3

2005 ◽  
Vol 15 (12) ◽  
pp. 3091-3095 ◽  
Author(s):  
Kouji Hattori ◽  
Akira Tanaka ◽  
Osamu Okitsu ◽  
Seiichiro Tabuchi ◽  
Kiyoshi Taniguchi ◽  
...  
Keyword(s):  
Receptor Agonists ◽  
Ip Receptor ◽  
Orally Active
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