Synthesis and Biological Evaluation of Pyridazinone Analogues as Potential Cardiac Positron Emission Tomography Tracers

Ajay Purohit; Heike Radeke; Michael Azure; Kelley Hanson; Richard Benetti; Fran Su; Padmaja Yalamanchili; Ming Yu; Megan Hayes; Mary Guaraldi; Mikhail Kagan; Simon Robinson; David Casebier

doi:10.1021/jm701443n

Synthesis and Biological Evaluation of Pyridazinone Analogues as Potential Cardiac Positron Emission Tomography Tracers

Journal of Medicinal Chemistry ◽

10.1021/jm701443n ◽

2008 ◽

Vol 51 (10) ◽

pp. 2954-2970 ◽

Cited By ~ 21

Author(s):

Ajay Purohit ◽

Heike Radeke ◽

Michael Azure ◽

Kelley Hanson ◽

Richard Benetti ◽

...

Keyword(s):

Positron Emission Tomography ◽

Biological Evaluation ◽

Emission Tomography ◽

Cardiac Positron Emission Tomography ◽

Positron Emission ◽

Synthesis And Biological Evaluation

Synthesis and Biological Evaluation of the Mitochondrial Complex 1 Inhibitor 2-[4-(4-Fluorobutyl)benzylsulfanyl]-3-methylchromene-4-one as a Potential Cardiac Positron Emission Tomography Tracer

Journal of Medicinal Chemistry ◽

10.1021/jm0701831 ◽

2007 ◽

Vol 50 (18) ◽

pp. 4304-4315 ◽

Cited By ~ 8

Author(s):

Heike Radeke ◽

Kelley Hanson ◽

Padmaja Yalamanchili ◽

Megan Hayes ◽

Zhi-Qin Zhang ◽

...

Keyword(s):

Positron Emission Tomography ◽

Biological Evaluation ◽

Emission Tomography ◽

Positron Emission Tomography Tracer ◽

Mitochondrial Complex ◽

Cardiac Positron Emission Tomography ◽

Positron Emission ◽

Synthesis And Biological Evaluation

Synthesis and Biological Evaluation of Substituted [18F]Imidazo[1,2-a]pyridines and [18F]Pyrazolo[1,5-a]pyrimidines for the Study of the Peripheral Benzodiazepine Receptor Using Positron Emission Tomography

Journal of Medicinal Chemistry ◽

10.1021/jm7014556 ◽

2008 ◽

Vol 51 (13) ◽

pp. 3700-3712 ◽

Cited By ~ 90

Author(s):

Christopher J. R. Fookes ◽

Tien Q. Pham ◽

Filomena Mattner ◽

Ivan Greguric ◽

Christian Loc’h ◽

...

Keyword(s):

Positron Emission Tomography ◽

Benzodiazepine Receptor ◽

Biological Evaluation ◽

Emission Tomography ◽

Peripheral Benzodiazepine Receptor ◽

Positron Emission ◽

Synthesis And Biological Evaluation

Synthesis and biological evaluation of potential positron emission tomography (PET) ligands for brain visualization of dopamine D3 receptors

ARKIVOC ◽

10.3998/ark.5550190.0007.811 ◽

2006 ◽

Vol 2006 (8) ◽

pp. 102-110 ◽

Cited By ~ 1

Author(s):

Enza Lacivita ◽

Francesco Berardi ◽

Nicola A. Colabufo ◽

Marcello Leopoldo ◽

Roberto Perrone ◽

...

Keyword(s):

Positron Emission Tomography ◽

Biological Evaluation ◽

Emission Tomography ◽

Dopamine D3 Receptors ◽

D3 Receptors ◽

Positron Emission ◽

Dopamine D3 ◽

Synthesis And Biological Evaluation

Synthesis and biological evaluation of 68Ga-bis-DOTA-PA as a potential agent for positron emission tomography imaging of necrosis

Nuclear Medicine and Biology ◽

10.1016/j.nucmedbio.2013.04.011 ◽

2013 ◽

Vol 40 (6) ◽

pp. 816-822 ◽

Cited By ~ 7

Author(s):

Kristof Prinsen ◽

Marlein M. Cona ◽

Bernard J. Cleynhens ◽

Junjie Li ◽

Hubert Vanbilloen ◽

...

Keyword(s):

Positron Emission Tomography ◽

Positron Emission Tomography Imaging ◽

Biological Evaluation ◽

Emission Tomography ◽

Tomography Imaging ◽

Positron Emission ◽

Synthesis And Biological Evaluation

Synthesis and biological evaluation of a series of novel N- or O-fluoroalkyl derivatives of tropane: potential positron emission tomography (PET) imaging agents for the dopamine transporter

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(01)00626-6 ◽

2001 ◽

Vol 11 (23) ◽

pp. 3049-3053 ◽

Cited By ~ 22

Author(s):

Xiao-Hui Gu ◽

Rushi Zong ◽

Nora S Kula ◽

Ross J Baldessarini ◽

John L Neumeyer

Keyword(s):

Positron Emission Tomography ◽

Dopamine Transporter ◽

Pet Imaging ◽

Biological Evaluation ◽

Emission Tomography ◽

Imaging Agents ◽

Positron Emission ◽

Synthesis And Biological Evaluation ◽

Derivatives Of

Stereoselective synthesis and biological evaluation of syn-1-amino-3-[18F]fluorocyclobutyl-1-carboxylic acid as a potential positron emission tomography brain tumor imaging agent

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2009.01.032 ◽

2009 ◽

Vol 17 (5) ◽

pp. 1982-1990 ◽

Cited By ~ 23

Author(s):

Weiping Yu ◽

Larry Williams ◽

Vernon M. Camp ◽

Eugene Malveaux ◽

Jeffrey J. Olson ◽

...

Keyword(s):

Positron Emission Tomography ◽

Brain Tumor ◽

Carboxylic Acid ◽

Stereoselective Synthesis ◽

Tumor Imaging ◽

Biological Evaluation ◽

Emission Tomography ◽

Imaging Agent ◽

Positron Emission ◽

Synthesis And Biological Evaluation

Development of a new epidermal growth factor receptor positron emission tomography imaging agent based on the 3-cyanoquinoline core: Synthesis and biological evaluation

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2010.08.004 ◽

2010 ◽

Vol 18 (18) ◽

pp. 6634-6645 ◽

Cited By ~ 36

Author(s):

Federica Pisaneschi ◽

Quang-De Nguyen ◽

Elham Shamsaei ◽

Matthias Glaser ◽

Edward Robins ◽

...

Keyword(s):

Positron Emission Tomography ◽

Growth Factor Receptor ◽

Positron Emission Tomography Imaging ◽

Biological Evaluation ◽

Emission Tomography ◽

Agent Based ◽

Tomography Imaging ◽

Positron Emission ◽

Epidermal Growth ◽

Synthesis And Biological Evaluation

Synthesis and biological evaluation ofS-[11C]methylated mercaptoimidazole piperazinyl derivatives as potential radioligands for imaging 5-HT1Areceptors by positron emission tomography (PET)

Journal of Labelled Compounds and Radiopharmaceuticals ◽

10.1002/jlcr.924 ◽

2005 ◽

Vol 48 (4) ◽

pp. 301-315 ◽

Cited By ~ 10

Author(s):

Raquel Garcia ◽

Catarina Xavier ◽

António Paulo ◽

Isabel Santos ◽

Torsten Kniess ◽

...

Keyword(s):

Positron Emission Tomography ◽

Biological Evaluation ◽

Emission Tomography ◽

Positron Emission ◽

Synthesis And Biological Evaluation

Synthesis and biological evaluation of two agents for imaging estrogen receptor β by positron emission tomography: challenges in PET imaging of a low abundance target

Nuclear Medicine and Biology ◽

10.1016/j.nucmedbio.2012.05.011 ◽

2012 ◽

Vol 39 (8) ◽

pp. 1105-1116 ◽

Cited By ~ 8

Author(s):

Jae Hak Lee ◽

Olaf Peters ◽

Lutz Lehmann ◽

Carmen S. Dence ◽

Terry L. Sharp ◽

...

Keyword(s):

Positron Emission Tomography ◽

Estrogen Receptor ◽

Pet Imaging ◽

Biological Evaluation ◽

Estrogen Receptor Β ◽

Emission Tomography ◽

Two Agents ◽

Positron Emission ◽

Synthesis And Biological Evaluation

Synthesis and biological evaluation of positron emission tomography radiotracers targeting serotonin 4 receptors in brain: [18F]MNI-698 and [18F]MNI-699

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2013.09.097 ◽

2013 ◽

Vol 23 (23) ◽

pp. 6243-6247 ◽

Cited By ~ 14

Author(s):

Fabien Caillé ◽

Thomas J. Morley ◽

Adriana Alexandre S. Tavares ◽

Caroline Papin ◽

Nicole M. Twardy ◽

...

Keyword(s):

Positron Emission Tomography ◽

Biological Evaluation ◽

Emission Tomography ◽

Positron Emission ◽

Synthesis And Biological Evaluation