[11C]MK-4232: The First Positron Emission Tomography Tracer for the Calcitonin Gene-Related Peptide Receptor

Emission Tomography ◽

Peptide Receptor ◽

Related Peptide ◽

Positron Emission ◽

Faculty Opinions recommendation of [(11)C]MK-4232: The First Positron Emission Tomography Tracer for the Calcitonin Gene-Related Peptide Receptor.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.718109510.793483822 ◽

2013 ◽

Author(s):

Roger Freidinger

Keyword(s):

Emission Tomography ◽

Peptide Receptor ◽

Related Peptide ◽

Positron Emission ◽

In Vivo Quantification of Calcitonin Gene-Related Peptide Receptor Occupancy by Telcagepant in Rhesus Monkey and Human Brain Using the Positron Emission Tomography Tracer [11C]MK-4232

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.113.206458 ◽

2013 ◽

Vol 347 (2) ◽

pp. 478-486 ◽

Cited By ~ 82

Author(s):

Eric D. Hostetler ◽

Aniket D. Joshi ◽

Sandra Sanabria-Bohórquez ◽

Hong Fan ◽

Zhizhen Zeng ◽

...

Keyword(s):

Rhesus Monkey ◽

Human Brain ◽

Receptor Occupancy ◽

Emission Tomography ◽

Peptide Receptor ◽

Positron Emission ◽

Faculty Opinions recommendation of Modulation of nocioceptive transmission with calcitonin gene-related peptide receptor antagonists in the thalamus.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.7743956.8985062 ◽

2011 ◽

Author(s):

Luis Villanueva ◽

Rodrigo Noseda

Keyword(s):

Receptor Antagonists ◽

Peptide Receptor ◽

Related Peptide ◽

Development of a highly-specific 18F-labeled irreversible positron emission tomography tracer for monoacylglycerol lipase mapping

Acta Pharmaceutica Sinica B ◽

10.1016/j.apsb.2021.01.021 ◽

2021 ◽

Author(s):

Zhen Chen ◽

Wakana Mori ◽

Jian Rong ◽

Michael A. Schafroth ◽

Tuo Shao ◽

...

Keyword(s):

Emission Tomography ◽

Monoacylglycerol Lipase ◽

Receptor activity modifying proteins regulate the activity of a calcitonin gene-related peptide receptor in rabbit aortic endothelial cells

FEBS Letters ◽

10.1016/s0014-5793(98)01587-7 ◽

1998 ◽

Vol 441 (3) ◽

pp. 366-368 ◽

Cited By ~ 56

Author(s):

Roman Muff ◽

Kerstin Leuthäuser ◽

Nicole Bühlmann ◽

Steven M. Foord ◽

Jan A. Fischer ◽

...

Keyword(s):

Endothelial Cells ◽

Receptor Activity ◽

Aortic Endothelial Cells ◽

Peptide Receptor ◽

Related Peptide ◽

Calcitonin Gene ◽

Receptor Activity Modifying Proteins ◽

Aortic Endothelial

Synthesis and evaluation of [18F]-fluoromethyl triphenylphosphonium cation as a novel mitochondria-specific positron emission tomography tracer

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2016.04.036 ◽

2016 ◽

Vol 118 ◽

pp. 90-97 ◽

Cited By ~ 4

Author(s):

Huahui Zeng ◽

Xiangxiang Wu ◽

Fahuan Song ◽

Caiyun Xu ◽

Hao Liu ◽

...

Keyword(s):

Emission Tomography ◽

Scavenging strategy for specific activity improvement: application to a new CXCR4-specific cyclopentapeptide positron emission tomography tracer

Journal of Labelled Compounds and Radiopharmaceuticals ◽

10.1002/jlcr.3095 ◽

2013 ◽

Vol 56 (13) ◽

pp. 679-685 ◽

Cited By ~ 6

Author(s):

Guillaume P. C. George ◽

Federica Pisaneschi ◽

Elizabeth Stevens ◽

Quang-Dé Nguyen ◽

Ola Åberg ◽

...

Keyword(s):

Specific Activity ◽

Emission Tomography ◽

Compelling case for fostering Titanium-45 for positron emission tomography tracer applications

Indian Journal of Nuclear Medicine ◽

10.4103/ijnm.ijnm_52_20 ◽

2020 ◽

Vol 35 (3) ◽

pp. 200

Author(s):

Natesan Ramamoorthy

Keyword(s):

Emission Tomography ◽

Pharmacological Properties of MK-3207, a Potent and Orally Active Calcitonin Gene-Related Peptide Receptor Antagonist

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.109.163816 ◽

2010 ◽

Vol 333 (1) ◽

pp. 152-160 ◽

Cited By ~ 52

Author(s):

Christopher A. Salvatore ◽

Eric L. Moore ◽

Amy Calamari ◽

Jacquelynn J. Cook ◽

Maria S. Michener ◽

...

Keyword(s):

Receptor Antagonist ◽

Pharmacological Properties ◽

Peptide Receptor ◽

Related Peptide ◽

Calcitonin Gene ◽

Orally Active

1 Calcitonin Gene-Related Peptide Receptor Antagonists for the Treatment of Migraine

Progress in Medicinal Chemistry - Progress in Medicinal Chemistry Volume 47 ◽

10.1016/s0079-6468(08)00201-4 ◽

2009 ◽

pp. 1-35 ◽

Cited By ~ 3

Author(s):

Theresa M. Williams ◽

Christopher S. Burgey ◽

Christopher A. Salvatore

Keyword(s):

Receptor Antagonists ◽

Peptide Receptor ◽

Related Peptide ◽