Transposition of Three Amino Acids Transforms the Human Metabotropic Glutamate Receptor (mGluR)-3-Positive Allosteric Modulation Site to mGluR2, and Additional Characterization of the mGluR2-Positive Allosteric Modulation Site

Allosteric Modulation ◽

Molecular characterization of a novel metabotropic glutamate receptor mGluR5 coupled to inositol phosphate/Ca2+ signal transduction.

Journal of Biological Chemistry ◽

10.1016/s0021-9258(18)42219-3 ◽

1992 ◽

Vol 267 (19) ◽

pp. 13361-13368 ◽

Cited By ~ 2

Author(s):

T Abe ◽

H Sugihara ◽

H Nawa ◽

R Shigemoto ◽

N Mizuno ◽

...

Keyword(s):

Signal Transduction ◽

Molecular Characterization ◽

Glutamate Receptor ◽

Inositol Phosphate ◽

Cloning and Characterization of a Metabotropic Glutamate Receptor, mGluR4b

Neuropharmacology ◽

10.1016/s0028-3908(96)00153-0 ◽

1997 ◽

Vol 36 (1) ◽

pp. 21-30 ◽

Cited By ~ 34

Author(s):

C. THOMSEN ◽

R. PEKHLETSKI ◽

B. HALDEMAN ◽

T.A. GILBERT ◽

P. O'HARA ◽

...

Keyword(s):

Glutamate Receptor ◽

Molecular mechanism of positive allosteric modulation of the metabotropic glutamate receptor 2 by JNJ-46281222

British Journal of Pharmacology ◽

10.1111/bph.13390 ◽

2016 ◽

Vol 173 (3) ◽

pp. 588-600 ◽

Cited By ~ 24

Author(s):

Maarten L J Doornbos ◽

Laura Pérez-Benito ◽

Gary Tresadern ◽

Thea Mulder-Krieger ◽

Ilse Biesmans ◽

...

Keyword(s):

Molecular Mechanism ◽

Glutamate Receptor ◽

Allosteric Modulation ◽

Expression and functional characterization of Metabotropic Glutamate Receptor Type 6 (mGluR6) in detergent micelles

Biophysical Journal ◽

10.1016/j.bpj.2008.12.3167 ◽

2009 ◽

Vol 96 (3) ◽

pp. 593a

Author(s):

Kalyan C. Tirupula ◽

Harpreet K. Dhiman ◽

Naveena Yanamala ◽

Judith Klein-Seetharaman

Keyword(s):

Glutamate Receptor ◽

Functional Characterization ◽

Receptor Type ◽

Metabotropic Glutamate ◽

Detergent Micelles

Selective metabotropic glutamate receptor 2 positive allosteric modulation alleviates L-DOPA-induced psychosis-like behaviours and dyskinesia in the MPTP-lesioned marmoset

European Journal of Pharmacology ◽

10.1016/j.ejphar.2020.172957 ◽

2020 ◽

Vol 873 ◽

pp. 172957 ◽

Cited By ~ 6

Author(s):

Lamia Sid-Otmane ◽

Adjia Hamadjida ◽

Stephen G. Nuara ◽

Dominique Bédard ◽

Fleur Gaudette ◽

...

Keyword(s):

Glutamate Receptor ◽

Allosteric Modulation ◽

In Vitro Pharmacological Characterization of Novel Isoxazolopyridone Derivatives as Allosteric Metabotropic Glutamate Receptor 7 Antagonists

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.107.124701 ◽

2007 ◽

Vol 323 (1) ◽

pp. 147-156 ◽

Cited By ~ 96

Author(s):

Gentaroh Suzuki ◽

Naohiro Tsukamoto ◽

Hiroshi Fushiki ◽

Aki Kawagishi ◽

Masayuki Nakamura ◽

...

Keyword(s):

Glutamate Receptor ◽

Pharmacological Characterization ◽

Molecular Cloning, Functional Expression and Pharmacological Characterization of the Human Metabotropic Glutamate Receptor Type 2

European Journal of Neuroscience ◽

10.1111/j.1460-9568.1995.tb00666.x ◽

1995 ◽

Vol 7 (4) ◽

pp. 622-629 ◽

Cited By ~ 49

Author(s):

P. J. Flor ◽

K. Lindauer ◽

I. Püttner ◽

D. Rüegg ◽

S. Lukic ◽

...

Keyword(s):

Molecular Cloning ◽

Glutamate Receptor ◽

Functional Expression ◽

Receptor Type ◽

Pharmacological Characterization ◽

Characterization of a Truncated Metabotropic Glutamate Receptor in a Primitive Metazoan, the Parasitic Flatworm Schistosoma mansoni

PLoS ONE ◽

10.1371/journal.pone.0027119 ◽

2011 ◽

Vol 6 (11) ◽

pp. e27119 ◽

Cited By ~ 12

Author(s):

Amira Taman ◽

Paula Ribeiro

Keyword(s):

Schistosoma Mansoni ◽

Glutamate Receptor ◽

Metabotropic Glutamate ◽

Parasitic Flatworm

Synthesis and Pharmacological Characterization of Aminocyclopentanetricarboxylic Acids: New Tools to Discriminate between Metabotropic Glutamate Receptor Subtypes

Journal of Medicinal Chemistry ◽

10.1021/jm970207b ◽

1997 ◽

Vol 40 (19) ◽

pp. 3119-3129 ◽

Cited By ~ 106

Author(s):

Francine C. Acher ◽

Frédérique J. Tellier ◽

Robert Azerad ◽

Isabelle N. Brabet ◽

Laurent Fagni ◽

...

Keyword(s):

Glutamate Receptor ◽

Receptor Subtypes ◽

Pharmacological Characterization ◽

Characterization of a metabotropic glutamate receptor: direct negative coupling to adenylyl cyclase and involvement of a pertussis toxin-sensitive G protein.

Proceedings of the National Academy of Sciences ◽

10.1073/pnas.89.17.8040 ◽

1992 ◽

Vol 89 (17) ◽

pp. 8040-8044 ◽

Cited By ~ 23

Author(s):

L. Prezeau ◽

O. Manzoni ◽

V. Homburger ◽

F. Sladeczek ◽

K. Curry ◽

...

Keyword(s):

Adenylyl Cyclase ◽

G Protein ◽

Glutamate Receptor ◽

Pertussis Toxin ◽

Metabotropic Glutamate ◽

Negative Coupling