scholarly journals Discovery and Pharmacological Characterization of JNJ-42756493 (Erdafitinib), a Functionally Selective Small-Molecule FGFR Family Inhibitor

2017 ◽  
Vol 16 (6) ◽  
pp. 1010-1020 ◽  
Author(s):  
Timothy P.S. Perera ◽  
Eleonora Jovcheva ◽  
Laurence Mevellec ◽  
Jorge Vialard ◽  
Desiree De Lange ◽  
...  
Keyword(s):  
Small Molecule ◽  
Pharmacological Characterization

Pharmacological Characterization of [3H]VUF11211, a Novel Radiolabeled Small-Molecule Inverse Agonist for the Chemokine Receptor CXCR3

2015 ◽  
Vol 87 (4) ◽  
pp. 639-648 ◽  
Author(s):  
Danny J. Scholten ◽  
Maikel Wijtmans ◽  
Jeffrey R. van Senten ◽  
Hans Custers ◽  
Ailas Stunnenberg ◽  
...  
Keyword(s):  
Small Molecule ◽  
Chemokine Receptor ◽  
Inverse Agonist ◽  
Pharmacological Characterization

scholarly journals Pharmacological characterization of GLPG1972/S201086, a potent and selective small molecule inhibitor of ADAMTS5

2021 ◽  
Author(s):  
Philippe Clement-Lacroix ◽  
Christopher B. Little ◽  
Margaret M. Smith ◽  
Céline Cottereaux ◽  
Didier Merciris ◽  
...  
Keyword(s):  
Small Molecule ◽  
Small Molecule Inhibitor ◽  
Pharmacological Characterization ◽  
Molecule Inhibitor

Discovery and Pharmacological Characterization of a Small-Molecule Antagonist at Neuromedin U Receptor NMUR2

2009 ◽  
Vol 330 (1) ◽  
pp. 268-275 ◽  
Author(s):  
Jay J. Liu ◽  
Kemal Payza ◽  
Jian Huang ◽  
Ruifeng Liu ◽  
Tongming Chen ◽  
...  
Keyword(s):  
Small Molecule ◽  
Pharmacological Characterization ◽  
Small Molecule Antagonist

Pharmacological Characterization of CXC Chemokine Receptor 3 Ligands and a Small Molecule Antagonist

2005 ◽  
Vol 313 (3) ◽  
pp. 1263-1271 ◽  
Author(s):  
Christopher E. Heise ◽  
Anil Pahuja ◽  
Sarah C. Hudson ◽  
Monica S. Mistry ◽  
Amy L. Putnam ◽  
...  
Keyword(s):  
Small Molecule ◽  
Chemokine Receptor ◽  
Pharmacological Characterization ◽  
Small Molecule Antagonist ◽  
Cxc Chemokine

Pharmacological characterization of INCB3344, a small molecule antagonist of human CCR2

2009 ◽  
Vol 387 (2) ◽  
pp. 251-255 ◽  
Author(s):  
Niu Shin ◽  
Frédéric Baribaud ◽  
Kathy Wang ◽  
Genjie Yang ◽  
Rich Wynn ◽  
...  
Keyword(s):  
Small Molecule ◽  
Pharmacological Characterization ◽  
Small Molecule Antagonist

scholarly journals Pharmacological characterization of a small-molecule agonist for the chemokine receptor CXCR3

2012 ◽  
Vol 166 (3) ◽  
pp. 898-911 ◽  
Author(s):  
DJ Scholten ◽  
M Canals ◽  
M Wijtmans ◽  
S de Munnik ◽  
P Nguyen ◽  
...  
Keyword(s):  
Small Molecule ◽  
Chemokine Receptor ◽  
Pharmacological Characterization
Sign in / Sign up

Export Citation Format

Share Document