Stereoselective Solid-Phase Synthesis of Cyclopentane and Cyclohexane Derivatives by Two-Component Domino Reactions: Generation of Combinatorial Libraries

Lutz F. Tietze; Adrian Steinmetz

doi:10.1002/anie.199606511

Stereoselective Solid-Phase Synthesis of Cyclopentane and Cyclohexane Derivatives by Two-Component Domino Reactions: Generation of Combinatorial Libraries

Angewandte Chemie International Edition in English ◽

10.1002/anie.199606511 ◽

1996 ◽

Vol 35 (6) ◽

pp. 651-652 ◽

Cited By ~ 43

Author(s):

Lutz F. Tietze ◽

Adrian Steinmetz

Keyword(s):

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Domino Reactions ◽

Phase Synthesis ◽

Two Component

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Combinatorial Libraries on Rigid Scaffolds: Solid Phase Synthesis of Variably Substituted Pyrazoles and Isoxazoles

Molecules ◽

10.3390/jan97p5 ◽

1997 ◽

Vol 2 (12) ◽

pp. 17-30 ◽

Cited By ~ 14

Author(s):

Andreas Marzinzik ◽

Eduard Felder

Keyword(s):

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis ◽

Substituted Pyrazoles

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How to Optimize Reactions for Solid-Phase Synthesis of Combinatorial Libraries Using RF-Tagged Microreactors

Optimization of Solid-Phase Combinatorial Synthesis ◽

10.1201/9781482271058-5 ◽

2001 ◽

pp. 69-82

Keyword(s):

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis

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Elimination Chemistry in the Solution- and Solid-Phase Synthesis of Combinatorial Libraries

ChemInform ◽

10.1002/chin.200411244 ◽

2004 ◽

Vol 35 (11) ◽

Author(s):

Demosthenes Fokas ◽

Carmen Baldino

Keyword(s):

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis

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Solid phase synthesis of mixture-based acyclic and heterocyclic small molecule combinatorial libraries from resin-bound polyamides

Biopolymers ◽

10.1002/1097-0282(2001)60:3<212::aid-bip10033>3.0.co;2-d ◽

2001 ◽

Vol 60 (3) ◽

pp. 212-219 ◽

Cited By ~ 8

Author(s):

Adel Nefzi ◽

John M. Ostresh ◽

Richard A. Houghten

Keyword(s):

Small Molecule ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis

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ChemInform Abstract: Solid-Phase Synthesis of Mixture-Based Acyclic and Heterocyclic Small Molecule Combinatorial Libraries from Resin-Bound Polyamides.

ChemInform ◽

10.1002/chin.200225266 ◽

2010 ◽

Vol 33 (25) ◽

pp. no-no

Author(s):

Adel Nefzi ◽

John M. Ostresh ◽

Richard A. Houghten

Keyword(s):

Small Molecule ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis

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ChemInform Abstract: A Novel Concept in Combinatorial Chemistry in Solution with the Advantages of Solid-Phase Synthesis: Formation of N-Betaines by Multicomponent Domino Reactions.

ChemInform ◽

10.1002/chin.200124047 ◽

2010 ◽

Vol 32 (24) ◽

pp. no-no

Author(s):

Lutz F. Tietze ◽

Holger Evers ◽

Enno Toepken

Keyword(s):

Combinatorial Chemistry ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Domino Reactions ◽

Phase Synthesis ◽

Novel Concept

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Faculty Opinions recommendation of Solid phase synthesis of mixture-based acyclic and heterocyclic small molecule combinatorial libraries from resin-bound polyamides.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.1003350.35604 ◽

2002 ◽

Author(s):

Morten Meldal

Keyword(s):

Small Molecule ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis

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Solid-phase synthesis and screening of N-acylated polyamine (NAPA) combinatorial libraries for protein binding

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2010.09.054 ◽

2010 ◽

Vol 20 (22) ◽

pp. 6500-6503 ◽

Cited By ~ 11

Author(s):

Jaclyn A. Iera ◽

Lisa M. Miller Jenkins ◽

Hiroshi Kajiyama ◽

Jeffrey B. Kopp ◽

Daniel H. Appella

Keyword(s):

Protein Binding ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis

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Determination of isokinetic ratios necessary for equimolar incorporation of carboxylic acids in the solid-phase synthesis of mixture-based combinatorial libraries

Biopolymers ◽

10.1002/bip.10206 ◽

2002 ◽

Vol 65 (1) ◽

pp. 32-39 ◽

Cited By ~ 9

Author(s):

Achyuta N. Acharya ◽

John M. Ostresh ◽

Richard A. Houghten

Keyword(s):

Carboxylic Acids ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis

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Solid-phase synthesis of combinatorial libraries based on enatiomerically pure (1S,2S,4R,5S)-4,5-dihydroxycyclohexan-1,2-dicarboxylic acid scaffolds

Il Farmaco ◽

10.1016/s0014-827x(02)01306-x ◽

2002 ◽

Vol 57 (10) ◽

pp. 861-864

Author(s):

Daniela Arosio ◽

Anna Bernardi ◽

Donatella Dellavecchia ◽

Fabrizio Micheli ◽

Alessandra Pasquarello

Keyword(s):

Dicarboxylic Acid ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Combinatorial Libraries ◽

Phase Synthesis

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