Bone-targeted, nonpeptide inhibitors of the Src SH2 domain: Structure-based design and structure-activity relationships

2002 ◽  
pp. 558-560
Author(s):  
Regine Bohacek ◽  
Manfred Weigele ◽  
Virginia Jacobsen ◽  
Karina Macek ◽  
George Luke ◽  
...  
Keyword(s):  
Domain Structure ◽  
Sh2 Domain ◽  
Structure Activity Relationships ◽  
Structure Activity

Structure−Activity Relationships of Small Phosphopeptides, Inhibitors of Grb2 SH2 Domain, and Their Prodrugs

2004 ◽  
Vol 47 (5) ◽  
pp. 1223-1233 ◽  
Author(s):  
Wang-Qing Liu ◽  
Michel Vidal ◽  
Catherine Olszowy ◽  
Emmanuelle Million ◽  
Christine Lenoir ◽  
...  
Keyword(s):  
Sh2 Domain ◽  
Structure Activity Relationships ◽  
Structure Activity

Dissociation of I Domain and Global Conformational Changes in LFA-1:  Refinement of Small Molecule-I Domain Structure−Activity Relationships†

Biochemistry ◽  
2005 ◽  
Vol 44 (11) ◽  
pp. 4322-4331 ◽  
Author(s):  
Richard S. Larson ◽  
Terry Davis ◽  
Cristian Bologa ◽  
Gloria Semenuk ◽  
Sreejith Vijayan ◽  
...  
Keyword(s):  
Domain Structure ◽  
Small Molecule ◽  
Conformational Changes ◽  
Structure Activity Relationships ◽  
Structure Activity

Structure-activity relationships in the acronycine and benzo[b]acronycine series: Role of the pyran ring

Planta Medica ◽  
2008 ◽  
Vol 74 (09) ◽  
Author(s):  
Q Do ◽  
H Doan Thi Mai ◽  
T Gaslonde ◽  
B Pfeiffer ◽  
S Léonce ◽  
...  
Keyword(s):  
Pyran Ring ◽  
Structure Activity Relationships ◽  
Structure Activity

Structure activity-relationships of P-Glycoprotein modulation using a small library of macrocyclic lathyrane diterpenes

Planta Medica ◽  
2012 ◽  
Vol 78 (11) ◽  
Author(s):  
M Reis ◽  
RJ Ferreira ◽  
MMM Santos ◽  
DJVA dos Santos ◽  
J Molnár ◽  
...  
Keyword(s):  
Structure Activity Relationships ◽  
Structure Activity ◽  
P Glycoprotein
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