The critical inclination problem: A simple treatment

1970 ◽  
Vol 2 (1) ◽  
pp. 121-122 ◽  
Author(s):  
R. R. Allan
Keyword(s):  
Critical Inclination ◽  
Simple Treatment ◽  
Inclination Problem

The critical inclination problem ? 30 years of progress

1987 ◽  
Vol 43 (1-4) ◽  
pp. 127-138 ◽  
Author(s):  
A. H. Jupp
Keyword(s):  
Critical Inclination ◽  
Inclination Problem

The critical inclination problem with small eccentricity

1980 ◽  
Vol 21 (4) ◽  
pp. 361-393 ◽  
Author(s):  
Alan H. Jupp
Keyword(s):  
Critical Inclination ◽  
Small Eccentricity ◽  
Inclination Problem

The critical inclination problem with small eccentricity

1983 ◽  
Vol 30 (3) ◽  
pp. 297-308 ◽  
Author(s):  
Alan H. Jupp ◽  
Ali Y. Abdulla
Keyword(s):  
Critical Inclination ◽  
Small Eccentricity ◽  
Inclination Problem

scholarly journals 2-Cyclopropyl-6-phenyl-2,3-dihydrothieno[3,2-d][1,3,2]diazaborinin-4(1H)-one

Molbank ◽  
10.3390/m1221 ◽  
2021 ◽  
Vol 2021 (2) ◽  
pp. M1221
Author(s):  
Romain Mustière ◽  
Patrice Vanelle ◽  
Nicolas Primas
Keyword(s):  
Scaffold Hopping ◽  
Simple Treatment ◽  
Biological Tests

As part of our ongoing scaffold hopping work on antimalarial 2-aminothieno[3,2-d]pyrimidin-4-one scaffold, we explored the dihydrothieno[3,2-d][1,3,2]diazaborinin-4(1H)-one as a potential new antimalarial series. Using conditions found in the literature, we obtained 2-cyclopropyl-6-phenyl-2,3-dihydrothieno[3,2-d][1,3,2]diazaborinin-4(1H)-one with 93% yield through a simple treatment. It was then characterized by NMR (1H and 13C) and HRMS. Given the structure of this molecule, its aqueous stability was assessed to determine its suitability for biological tests. To our knowledge, this is the first dihydrothieno[3,2-d][1,3,2]diazaborinin-4(1H)-one described.

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