Design and efficient synthesis of novel vitamin D analogues bearing an aniline moiety in their side chains

Antonio Obelleiro; Uxía Gómez-Bouzó; Generosa Gómez; Yagamare Fall; Hugo Santalla

doi:10.1016/j.tetlet.2020.152493

Design and efficient synthesis of novel vitamin D analogues bearing an aniline moiety in their side chains

Tetrahedron Letters ◽

10.1016/j.tetlet.2020.152493 ◽

2020 ◽

Vol 61 (45) ◽

pp. 152493

Author(s):

Antonio Obelleiro ◽

Uxía Gómez-Bouzó ◽

Generosa Gómez ◽

Yagamare Fall ◽

Hugo Santalla

Keyword(s):

Vitamin D ◽

Side Chains ◽

Efficient Synthesis ◽

Vitamin D Analogues

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Efficient Synthesis of 1α-Fluoro A-Ring Phosphine Oxide, a Useful Building Block for Vitamin D Analogues, from (S)-Carvone via a Highly Selective Palladium-Catalyzed Isomerization of Dieneoxide to Dieneol

The Journal of Organic Chemistry ◽

10.1021/jo015788y ◽

2001 ◽

Vol 66 (18) ◽

pp. 6141-6150 ◽

Cited By ~ 22

Author(s):

Marek M. Kabat ◽

Lisa M. Garofalo ◽

Andrzej R. Daniewski ◽

Stanley D. Hutchings ◽

Wen Liu ◽

...

Keyword(s):

Vitamin D ◽

Phosphine Oxide ◽

Building Block ◽

Efficient Synthesis ◽

Vitamin D Analogues ◽

Palladium Catalyzed

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ChemInform Abstract: Efficient Synthesis of 1α-Fluoro A-Ring Phosphine Oxide, a Useful Building Block for Vitamin D Analogues, from (S)-Carvone via a Highly Selective Palladium-Catalyzed Isomerization of Dienoxide to Dienol.

ChemInform ◽

10.1002/chin.200202246 ◽

2010 ◽

Vol 33 (2) ◽

pp. no-no

Author(s):

Marek M. Kabat ◽

Lisa M. Garofalo ◽

Andrzej R. Daniewski ◽

Stanley D. Hutchings ◽

Wen Liu ◽

...

Keyword(s):

Vitamin D ◽

Phosphine Oxide ◽

Building Block ◽

Efficient Synthesis ◽

Vitamin D Analogues ◽

Palladium Catalyzed

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Vitamin D and Click Chemistry. Part 1. A Stereoselective Route to Vitamin D Analogues (VI) with Triazole Rings in Their Side Chains.

ChemInform ◽

10.1002/chin.200438208 ◽

2004 ◽

Vol 35 (38) ◽

Author(s):

Pedro Lois Suarez ◽

Zoila Gandara ◽

Generosa Gomez ◽

Yagamare Fall

Keyword(s):

Vitamin D ◽

Click Chemistry ◽

Side Chains ◽

Vitamin D Analogues

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Vitamin D and click chemistry. Part 1: A stereoselective route to vitamin D analogues with triazole rings in their side chains

Tetrahedron Letters ◽

10.1016/j.tetlet.2004.04.117 ◽

2004 ◽

Vol 45 (24) ◽

pp. 4619-4621 ◽

Cited By ~ 19

Author(s):

Pedro Lois Suarez ◽

Zoila Gándara ◽

Generosa Gómez ◽

Yagamare Fall

Keyword(s):

Vitamin D ◽

Click Chemistry ◽

Side Chains ◽

Vitamin D Analogues

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Design, Synthesis, Evaluation, and Structure of Vitamin D Analogues with Furan Side Chains

Chemistry - A European Journal ◽

10.1002/chem.201102695 ◽

2011 ◽

Vol 18 (2) ◽

pp. 603-612 ◽

Cited By ~ 12

Author(s):

Ramón Fraga ◽

Flavia Zacconi ◽

Fredy Sussman ◽

Paloma Ordóñez-Morán ◽

Alberto Muñoz ◽

...

Keyword(s):

Vitamin D ◽

Side Chains ◽

Design Synthesis ◽

Vitamin D Analogues

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SYNTHESIS AND BIOLOGICAL ACTIVITY OF 1a-HYDROXYLATED VITAMIN D ANALOGUES WITH POLY-UNSATURATED SIDE CHAINS

Vitamin D ◽

10.1515/9783110850345-054 ◽

1991 ◽

pp. 192-193 ◽

Cited By ~ 6

Keyword(s):

Vitamin D ◽

Biological Activity ◽

Side Chains ◽

Vitamin D Analogues

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Synthesis and immunoregulating activity of vitamin D analogues bearing pregnane side chains

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(00)80232-2 ◽

1992 ◽

Vol 2 (10) ◽

pp. 1289-1292 ◽

Cited By ~ 3

Author(s):

Eigoro Murayama ◽

Katsuhito Miyamoto ◽

Kiyoshige Ochi ◽

Noboru Kubodera

Keyword(s):

Vitamin D ◽

Side Chains ◽

Vitamin D Analogues

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Active vitamin D analogues and oral phosphate for the treatment of X-linked hypophosphataemia in paediatric patients: A systematic literature review and survey of expert opinion on current needs

Bone Abstracts ◽

10.1530/boneabs.7.p75 ◽

2019 ◽

Author(s):

Gema Ariceta ◽

Carmen de Lucas Collantes ◽

Ravi Jandhyala ◽

Zulf Mughal

Keyword(s):

Vitamin D ◽

Literature Review ◽

Expert Opinion ◽

Systematic Literature Review ◽

Active Vitamin ◽

Active Vitamin D ◽

Vitamin D Analogues ◽

Paediatric Patients

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Faculty Opinions recommendation of Vitamin D and vitamin D analogues for preventing fractures associated with involutional and post-menopausal osteoporosis.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.4120.461604 ◽

2005 ◽

Author(s):

Olof Johnell

Keyword(s):

Vitamin D ◽

Vitamin D Analogues ◽

Post Menopausal Osteoporosis ◽

Post Menopausal ◽

Menopausal Osteoporosis

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Highly efficient synthesis of polymer brushes with PEO and PCL as side chains via click chemistry

Polymer ◽

10.1016/j.polymer.2012.02.055 ◽

2012 ◽

Vol 53 (10) ◽

pp. 1992-2000 ◽

Cited By ~ 48

Author(s):

Peng Zhao ◽

Yechao Yan ◽

Xiaoqin Feng ◽

Lixin Liu ◽

Chun Wang ◽

...

Keyword(s):

Click Chemistry ◽

Polymer Brushes ◽

Side Chains ◽

Efficient Synthesis ◽

Highly Efficient

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