4-[(8-Alkyl-8-azabicyclo[3.2.1]octyl-3-yl)-3-arylanilino]- N , N -diethylbenzamides: high affinity, selective ligands for the delta opioid receptor illustrate factors important to antagonist activity

2000 ◽  
Vol 10 (11) ◽  
pp. 1281-1284 ◽  
Author(s):  
James B Thomas ◽  
Robert N Atkinson ◽  
Richard B Rothman ◽  
Jason P Burgess ◽  
S.Wayne Mascarella ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Delta Opioid Receptor ◽  
Antagonist Activity ◽  
High Affinity ◽  
Selective Ligands

scholarly journals A single residue, aspartic acid 95, in the delta opioid receptor specifies selective high affinity agonist binding.

1993 ◽  
Vol 268 (31) ◽  
pp. 23055-23058
Author(s):  
H Kong ◽  
K Raynor ◽  
K Yasuda ◽  
S.T. Moe ◽  
P.S. Portoghese ◽  
...  
Keyword(s):  
Aspartic Acid ◽  
Opioid Receptor ◽  
Delta Opioid Receptor ◽  
Agonist Binding ◽  
High Affinity

ChemInform Abstract: Novel Delta-Opioid-Receptor-Selective Ligands in the 14-Alkoxy-Substituted Indolo- and Benzofuromorphinan Series.

ChemInform ◽  
2010 ◽  
Vol 32 (46) ◽  
pp. no-no
Author(s):  
Dauren Biyashev ◽  
Krisztina Monory ◽  
Sandor Benyhe ◽  
Johannes Schuetz ◽  
Martin Koch ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Delta Opioid Receptor ◽  
Selective Ligands

Novel Delta-Opioid-Receptor-Selective Ligands in the 14-Alkoxy-Substituted Indolo- and Benzofuromorphinan Series

2001 ◽  
Vol 84 (7) ◽  
pp. 2015-2021 ◽  
Author(s):  
Dauren Biyashev ◽  
Krisztina Monory ◽  
Sandor Benyhe ◽  
Johannes Schütz ◽  
Martin Koch ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Delta Opioid Receptor ◽  
Selective Ligands

A high affinity, highly selective ligand for the delta opioid receptor: [3H]-[D-PEN2, pCl-PHE4, D-PEN5]enkephalin

Life Sciences ◽  
1989 ◽  
Vol 45 (11) ◽  
pp. 1001-1008 ◽  
Author(s):  
Linda K. Vaughn ◽  
Richard J. Knapp ◽  
Geza Toth ◽  
Y.-P. Wan ◽  
Victor J. Hruby ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Delta Opioid Receptor ◽  
High Affinity ◽  
Selective Ligand

Delta opioid receptor-selective ligands: [] enkephalin-dermenkephalin-dermenkephalin chimeric peptides

Life Sciences ◽  
1991 ◽  
Vol 49 (7) ◽  
pp. 495-503 ◽  
Author(s):  
Silvia Cavagnero ◽  
Aleksandra Misicka ◽  
Richard J. Knapp ◽  
Peg Davis ◽  
Lei Fang ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Delta Opioid Receptor ◽  
Selective Ligands ◽  
Chimeric Peptides

Delta opioid receptor selective ligands; DPLPE-deltorphin chimeric peptide analogues†

2009 ◽  
Vol 44 (1) ◽  
pp. 80-84 ◽  
Author(s):  
ALEKSANDRA MISICKA ◽  
ANDRZEJ W. LIPKOWSKI ◽  
ROBERT HORVATH ◽  
PEG DAVIS ◽  
FRANK PORRECA ◽  
...  
Keyword(s):  
Opioid Receptor ◽  
Delta Opioid Receptor ◽  
Chimeric Peptide ◽  
Selective Ligands ◽  
Peptide Analogues
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