Navigating CYP1A Induction and Arylhydrocarbon Receptor Agonism in Drug Discovery. A Case History with S1P1Agonists

Journal of Medicinal Chemistry ◽

10.1021/acs.jmedchem.5b01102 ◽

2015 ◽

Vol 58 (20) ◽

pp. 8236-8256 ◽

Author(s):

Simon J. Taylor ◽

Emmanuel H. Demont ◽

James Gray ◽

Nigel Deeks ◽

Aarti Patel ◽

...

Keyword(s):

Drug Discovery ◽

Case History ◽

Arylhydrocarbon Receptor ◽

Cyp1a Induction

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Faculty Opinions recommendation of Navigating CYP1A Induction and Arylhydrocarbon Receptor Agonism in Drug Discovery. A Case History with S1P1 Agonists.

Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature ◽

10.3410/f.725803874.793510021 ◽

2015 ◽

Author(s):

John Lowe

Keyword(s):

Drug Discovery ◽

Case History ◽

Arylhydrocarbon Receptor ◽

Cyp1a Induction

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Complex Target-Oriented Synthesis in the Drug Discovery Process: A Case History in the dEpoB Series

The Journal of Organic Chemistry ◽

10.1021/jo991006d ◽

1999 ◽

Vol 64 (23) ◽

pp. 8434-8456 ◽

Author(s):

Samuel J. Danishefsky

Keyword(s):

Drug Discovery ◽

Case History ◽

Discovery Process ◽

Drug Discovery Process ◽

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Chapter 12. A Case History on the Challenges of Central Nervous System and Dual Pharmacology Drug Discovery

Accounts in Drug Discovery ◽

10.1039/9781849731980-00267 ◽

2010 ◽

pp. 267-286

Author(s):

Paul V. Fish ◽

Anthony Harrison ◽

Florian Wakenhut ◽

Gavin A. Whitlock

Keyword(s):

Central Nervous System ◽

Nervous System ◽

Drug Discovery ◽

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ChemInform Abstract: Complex Target-Oriented Synthesis in the Drug Discovery Process: A Case History in the dEpoB Series

10.1002/chin.200011263 ◽

2010 ◽

Vol 31 (11) ◽

pp. no-no ◽

Author(s):

Christina R. Harris ◽

Samuel J. Danishefsky

Keyword(s):

Drug Discovery ◽

Case History ◽

Discovery Process ◽

Drug Discovery Process ◽

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A drug discovery case history of ‘delta-9-tetrahydrocannabinol, cannabidiol’

Expert Opinion on Drug Discovery ◽

10.1517/17460441.2011.560935 ◽

2011 ◽

Vol 6 (4) ◽

pp. 437-452 ◽

Author(s):

Radu Tanasescu ◽

David Rog ◽

Cris S Constantinescu

Keyword(s):

Drug Discovery ◽

Case History ◽

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Sobetirome: a case history of bench-to-clinic drug discovery and development

Heart Failure Reviews ◽

10.1007/s10741-008-9122-x ◽

2008 ◽

Vol 15 (2) ◽

pp. 177-182 ◽

Author(s):

Thomas S. Scanlan

Keyword(s):

Drug Discovery ◽

Case History ◽

Drug Discovery And Development ◽

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Epigenetics for Drug Discovery

10.1039/9781782628484 ◽

2015 ◽

Keyword(s):

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Drug Discovery for Leishmaniasis

10.1039/9781788010177 ◽

2017 ◽

Keyword(s):

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Artificial Intelligence in Drug Discovery

10.1039/9781788016841 ◽

2020 ◽

Keyword(s):

Artificial Intelligence ◽

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Phenotypic Drug Discovery

10.1039/9781839160721 ◽

2020 ◽

Keyword(s):

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