Synthesis and receptor binding properties of fluoro- and iodo-substituted high-affinity .sigma.-receptor ligands: identification of potential PET and SPECT .sigma.-receptor imaging agents

1992 ◽  
Vol 35 (12) ◽  
pp. 2221-2230 ◽  
Author(s):  
Brian De Costa ◽  
Lilian Radesca ◽  
Celia Dominguez ◽  
Lisa Di Paolo ◽  
Wayne D. Bowen
Keyword(s):  
Receptor Binding ◽  
Sigma Receptor ◽  
Imaging Agents ◽  
Receptor Imaging ◽  
Receptor Ligands ◽  
Binding Properties ◽  
High Affinity ◽  
Sigma Receptor Ligands

Examination of four 123I-labeled piperidine-based sigma receptor ligands as potential melanoma imaging agents: Initial studies in mouse tumor models

1997 ◽  
Vol 24 (6) ◽  
pp. 587-593 ◽  
Author(s):  
Rikki N. Waterhouse ◽  
Janette Chapman ◽  
Beverley Izard ◽  
Angela Donald ◽  
Kerynne Belbin ◽  
...  
Keyword(s):  
Sigma Receptor ◽  
Imaging Agents ◽  
Mouse Tumor ◽  
Receptor Ligands ◽  
Tumor Models ◽  
Sigma Receptor Ligands ◽  
Mouse Tumor Models

N,N′-disubstituted acetamidines as high affinity sigma receptor ligands

1993 ◽  
Vol 3 (10) ◽  
pp. 2113-2116 ◽  
Author(s):  
N.Laxma Reddy ◽  
James B. Fischer ◽  
Kathleen J. Burke-Howie ◽  
Peter Barmettler ◽  
Michael R. Rhodes ◽  
...  
Keyword(s):  
Sigma Receptor ◽  
Receptor Ligands ◽  
High Affinity ◽  
Sigma Receptor Ligands

Effects of sigma receptor ligands on schedule-controlled behavior of rats: relation to sigma and PCP receptor binding affinity

1991 ◽  
Vol 104 (2) ◽  
pp. 157-163 ◽  
Author(s):  
Joseph G. Wettstein ◽  
François J. Roman ◽  
Marie-Noëlle Rocher ◽  
Jean-Louis Junien
Keyword(s):  
Binding Affinity ◽  
Receptor Binding ◽  
Sigma Receptor ◽  
Receptor Ligands ◽  
Receptor Binding Affinity ◽  
Sigma Receptor Ligands ◽  
Behavior Of Rats

Synthesis and evaluation of [18F] labeled benzamides: High affinity sigma receptor ligands for PET imaging

1997 ◽  
Vol 24 (4) ◽  
pp. 333-340 ◽  
Author(s):  
Carmen S. Dence ◽  
Christy S. John ◽  
Wayne D. Bowen ◽  
Michael J. Welch
Keyword(s):  
Pet Imaging ◽  
Sigma Receptor ◽  
Receptor Ligands ◽  
High Affinity ◽  
Sigma Receptor Ligands

N-(1-Arylpropionyl)-4-aryltetrahydropyridines, a new class of high-affinity selective .sigma. receptor ligands

1993 ◽  
Vol 36 (24) ◽  
pp. 3923-3928 ◽  
Author(s):  
David I. Schuster ◽  
Yan Ping Pan ◽  
Guyanand Singh ◽  
George Stoupakis ◽  
Bing Cai ◽  
...  
Keyword(s):  
Sigma Receptor ◽  
Receptor Ligands ◽  
New Class ◽  
High Affinity ◽  
Sigma Receptor Ligands

ChemInform Abstract: N,N′-Disubstituted Acetamidines as High Affinity Sigma Receptor Ligands.

ChemInform ◽  
2010 ◽  
Vol 25 (23) ◽  
pp. no-no
Author(s):  
N. L. REDDY ◽  
J. B. FISCHER ◽  
K. J. BURKE-HOWIE ◽  
P. BARMETTLER ◽  
M. R. RHODES ◽  
...  
Keyword(s):  
Sigma Receptor ◽  
Receptor Ligands ◽  
High Affinity ◽  
Sigma Receptor Ligands

scholarly journals Recent Advances in the Development of Sigma Receptor Ligands as Cytotoxic Agents: A Medicinal Chemistry Perspective

2021 ◽  
Author(s):  
Antonino N. Fallica ◽  
Valeria Pittalà ◽  
Maria N. Modica ◽  
Loredana Salerno ◽  
Giuseppe Romeo ◽  
...  
Keyword(s):  
Medicinal Chemistry ◽  
Cytotoxic Agents ◽  
Sigma Receptor ◽  
Receptor Ligands ◽  
Sigma Receptor Ligands ◽  
Recent Advances
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