scholarly journals Lead Discovery, Chemistry Optimization, and Biological Evaluation Studies of Novel Biamide Derivatives as CB2 Receptor Inverse Agonists and Osteoclast Inhibitors

2012 ◽  
Vol 55 (22) ◽  
pp. 9973-9987 ◽  
Author(s):  
Peng Yang ◽  
Kyaw-Zeyar Myint ◽  
Qin Tong ◽  
Rentian Feng ◽  
Haiping Cao ◽  
...  
Keyword(s):  
Evaluation Studies ◽  
Biological Evaluation ◽  
Cb2 Receptor ◽  
Lead Discovery ◽  
Inverse Agonists

scholarly journals Mechanisms of Osteoclastogenesis Inhibition by a Novel Class of Biphenyl-Type Cannabinoid CB2 Receptor Inverse Agonists

2011 ◽  
Vol 18 (8) ◽  
pp. 1053-1064 ◽  
Author(s):  
Wolfgang Schuehly ◽  
Juan Manuel Viveros Paredes ◽  
Jonas Kleyer ◽  
Antje Huefner ◽  
Sharon Anavi-Goffer ◽  
...  
Keyword(s):  
Cb2 Receptor ◽  
Inverse Agonists

Design, synthesis, and biological evaluation studies of novel quinazolinone derivatives as anticonvulsant agents

2013 ◽  
Vol 22 (12) ◽  
pp. 5823-5831 ◽  
Author(s):  
Mohamed F. Zayed ◽  
Hany E. A. Ahmed ◽  
Abdel-Sattar M. Omar ◽  
Adel S. Abdelrahim ◽  
Khaled El-Adl
Keyword(s):  
Evaluation Studies ◽  
Biological Evaluation ◽  
Design Synthesis ◽  
Anticonvulsant Agents ◽  
Quinazolinone Derivatives ◽  
Synthesis And Biological Evaluation

Identification of 2-arylquinazolines with alkyl-polyamine motifs as potent antileishmanial agents: Synthesis and biological evaluation studies

2022 ◽  
Author(s):  
Anjila Kumari ◽  
Tara Jaiswal ◽  
Vinay Kumar ◽  
Neha Hura ◽  
Gulshan Kumar ◽  
...  
Keyword(s):  
Evaluation Studies ◽  
Biological Evaluation ◽  
Side Chain ◽  
Chain Ring ◽  
Synthesis And Biological Evaluation

2-Arylquinazolines with a range of alkyl polyamines as side chain/ring functional motifs at 4th-position were considered for antileishmanial study with the rationale that related heterocyclic scaffolds and the polyamine functionalities...

scholarly journals Trisubstituted Sulfonamides: A New Chemotype for Development of Potent and Selective CB2 Receptor Inverse Agonists

2013 ◽  
Vol 4 (4) ◽  
pp. 387-392 ◽  
Author(s):  
Qin Ouyang ◽  
Qin Tong ◽  
Rentian Feng ◽  
Kyaw-Zeyar Myint ◽  
Peng Yang ◽  
...  
Keyword(s):  
Cb2 Receptor ◽  
Inverse Agonists

Identification and biological evaluation of thiazole-based inverse agonists of RORγt

2018 ◽  
Vol 28 (9) ◽  
pp. 1446-1455 ◽  
Author(s):  
Christian Gege ◽  
Maxwell D. Cummings ◽  
Michael Albers ◽  
Olaf Kinzel ◽  
Gerald Kleymann ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Inverse Agonists

Synthesis and SAR Studies of 2-Oxoquinoline Derivatives as CB2 Receptor Inverse Agonists

2006 ◽  
Vol 49 (6) ◽  
pp. 2022-2027 ◽  
Author(s):  
Katri H. Raitio ◽  
Juha R. Savinainen ◽  
Jouko Vepsäläinen ◽  
Jarmo T. Laitinen ◽  
Antti Poso ◽  
...  
Keyword(s):  
Cb2 Receptor ◽  
Inverse Agonists ◽  
Sar Studies
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