Identification of 2-arylquinazolines with alkyl-polyamine motifs as potent antileishmanial agents: Synthesis and biological evaluation studies

RSC Medicinal Chemistry ◽

10.1039/d1md00336d ◽

2022 ◽

Author(s):

Anjila Kumari ◽

Tara Jaiswal ◽

Vinay Kumar ◽

Neha Hura ◽

Gulshan Kumar ◽

...

Keyword(s):

Evaluation Studies ◽

Biological Evaluation ◽

Side Chain ◽

Chain Ring ◽

Synthesis And Biological Evaluation

2-Arylquinazolines with a range of alkyl polyamines as side chain/ring functional motifs at 4th-position were considered for antileishmanial study with the rationale that related heterocyclic scaffolds and the polyamine functionalities...

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Design, synthesis, and biological evaluation studies of novel quinazolinone derivatives as anticonvulsant agents

Medicinal Chemistry Research ◽

10.1007/s00044-013-0569-5 ◽

2013 ◽

Vol 22 (12) ◽

pp. 5823-5831 ◽

Cited By ~ 17

Author(s):

Mohamed F. Zayed ◽

Hany E. A. Ahmed ◽

Abdel-Sattar M. Omar ◽

Adel S. Abdelrahim ◽

Khaled El-Adl

Keyword(s):

Evaluation Studies ◽

Biological Evaluation ◽

Design Synthesis ◽

Anticonvulsant Agents ◽

Quinazolinone Derivatives ◽

Synthesis And Biological Evaluation

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Synthesis and biological evaluation of novel steroidal 5α,8α-endoperoxide derivatives with aliphatic side-chain as potential anticancer agents

Steroids ◽

10.1016/j.steroids.2017.05.013 ◽

2017 ◽

Vol 124 ◽

pp. 46-53 ◽

Cited By ~ 10

Author(s):

Ming Bu ◽

Tingting Cao ◽

Hongxia Li ◽

Mingzhou Guo ◽

Burton B. Yang ◽

...

Keyword(s):

Anticancer Agents ◽

Biological Evaluation ◽

Side Chain ◽

Aliphatic Side Chain ◽

Synthesis And Biological Evaluation

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Synthetic Epothilone Analogs with Modifications in the Northern Hemisphere and the Heterocyclic Side-Chain - Synthesis and Biological Evaluation

10.3390/ecsoc-4-01917 ◽

2000 ◽

Author(s):

Karl-Heinz Altmann ◽

Nicole End ◽

Guido Bold ◽

Giorgo Caravatti ◽

Markus Wartmann

Keyword(s):

Northern Hemisphere ◽

Biological Evaluation ◽

Side Chain ◽

Chain Synthesis ◽

Synthesis And Biological Evaluation

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Design, synthesis and biological evaluation of non-secosteriodal vitamin D receptor ligand bearing double side chain for the treatment of chronic pancreatitis

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2018.01.073 ◽

2018 ◽

Vol 146 ◽

pp. 541-553 ◽

Cited By ~ 3

Author(s):

Zi-Sheng Kang ◽

Cong Wang ◽

Xiao-Lin Han ◽

Jun-Jie Du ◽

Yan-Yi Li ◽

...

Keyword(s):

Vitamin D ◽

Chronic Pancreatitis ◽

Vitamin D Receptor ◽

Biological Evaluation ◽

Side Chain ◽

Receptor Ligand ◽

Design Synthesis ◽

Synthesis And Biological Evaluation

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Synthesis and Biological Evaluation of Novel Steroidal 5α,8α-Endoperoxide Derivatives with Aromatic Hydrazone Side Chain as Potential Anticancer Agents

Russian Journal of Bioorganic Chemistry ◽

10.1134/s1068162019060396 ◽

2019 ◽

Vol 45 (6) ◽

pp. 585-590 ◽

Cited By ~ 1

Author(s):

H. J. Wang ◽

M. Bu ◽

J. Wang ◽

L. Liu ◽

S. Zhang

Keyword(s):

Anticancer Agents ◽

Biological Evaluation ◽

Side Chain ◽

Synthesis And Biological Evaluation

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Synthesis and Biological Evaluation of Novel Epothilone B Side Chain Analogues

ChemMedChem ◽

10.1002/cmdc.201500401 ◽

2015 ◽

Vol 10 (12) ◽

pp. 1974-1979 ◽

Cited By ~ 7

Author(s):

K. C. Nicolaou ◽

Derek Rhoades ◽

Yanping Wang ◽

Sotirios Totokotsopoulos ◽

Ruoli Bai ◽

...

Keyword(s):

Biological Evaluation ◽

Side Chain ◽

Epothilone B ◽

Synthesis And Biological Evaluation

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Synthesis and Biological Evaluation of 1α,25-Dihydroxyvitamin D3Analogues with a Long Side Chain at C12 and Short C17 Side Chains

Journal of Medicinal Chemistry ◽

10.1021/jm3008272 ◽

2012 ◽

Vol 55 (20) ◽

pp. 8642-8656 ◽

Cited By ~ 11

Author(s):

Diego M. Carballa ◽

Samuel Seoane ◽

Flavia Zacconi ◽

Xenxo Pérez ◽

Antonio Rumbo ◽

...

Keyword(s):

Biological Evaluation ◽

Side Chain ◽

Side Chains ◽

Synthesis And Biological Evaluation

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Studies of vitamin D (calciferol) and its analogs. 39. Arocalciferols: synthesis and biological evaluation of aromatic side-chain analogs of 1.alpha.,25-dihydroxyvitamin D3

Journal of Medicinal Chemistry ◽

10.1021/jm00112a021 ◽

1991 ◽

Vol 34 (8) ◽

pp. 2452-2463 ◽

Cited By ~ 48

Author(s):

Bruno Figadere ◽

Anthony W. Norman ◽

Helen L. Henry ◽

H. Phillip Koeffler ◽

Jian Yuan Zhou ◽

...

Keyword(s):

Vitamin D ◽

Biological Evaluation ◽

Side Chain ◽

Aromatic Side Chain ◽

Dihydroxyvitamin D3 ◽

Synthesis And Biological Evaluation

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The Twisted Side Chain of Antillatoxin is Important for Potent Toxicity: Total Synthesis and Biological Evaluation of Antillatoxin and Analogues

Angewandte Chemie ◽

10.1002/ange.200905892 ◽

2009 ◽

Vol 122 (2) ◽

pp. 339-342 ◽

Cited By ~ 4

Author(s):

Ken Okura ◽

Shigeru Matsuoka ◽

Ryosuke Goto ◽

Masayuki Inoue

Keyword(s):

Total Synthesis ◽

Biological Evaluation ◽

Side Chain ◽

Synthesis And Biological Evaluation

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Design, synthesis and biological evaluation of cyclic angiotensin II analogues with 3,5 side-Chain bridges

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(02)00474-2 ◽

2002 ◽

Vol 12 (18) ◽

pp. 2627-2633 ◽

Cited By ~ 15

Author(s):

Panagiota Roumelioti ◽

Ludmila Polevaya ◽

Panagiotis Zoumpoulakis ◽

Nektarios Giatas ◽

Ilze Mutule ◽

...

Keyword(s):

Angiotensin Ii ◽

Biological Evaluation ◽

Side Chain ◽

Design Synthesis ◽

Angiotensin Ii Analogues ◽

Synthesis And Biological Evaluation

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