Synthesis and Biological Evaluation of Certain Alkenyldiarylmethanes as Anti-HIV-1 Agents Which Act as Non-Nucleoside Reverse Transcriptase Inhibitors

Anti Hiv ◽

Hiv 1

ChemInform Abstract: Synthesis and Biological Evaluation of Certain Alkenyldiarylmethanes as Anti-HIV-1 Agents Which Act as Non-Nucleoside Reverse Transcriptase Inhibitors.

ChemInform ◽

10.1002/chin.199648103 ◽

2010 ◽

Vol 27 (48) ◽

pp. no-no

Author(s):

M. CUSHMAN ◽

W. M. GOLEBIEWSKI ◽

L. GRAHAM ◽

J. A. TURPIN ◽

W. G. RICE ◽

...

Keyword(s):

Reverse Transcriptase ◽

Biological Evaluation ◽

Anti Hiv ◽

Hiv 1

Design, synthesis, and biological evaluation of novel 5-Alkyl-6-Adamantylmethylpyrimidin-4(3H)-ones as HIV-1 non-nucleoside reverse-transcriptase inhibitors

Chemical Biology & Drug Design ◽

10.1111/cbdd.12765 ◽

2016 ◽

Vol 88 (3) ◽

pp. 380-385 ◽

Cited By ~ 2

Author(s):

Wenxin Li ◽

Boshi Huang ◽

Dongwei Kang ◽

Erik De Clercq ◽

Dirk Daelemans ◽

...

Keyword(s):

Reverse Transcriptase ◽

Biological Evaluation ◽

Design Synthesis ◽

Hiv 1

Synthesis and Biological Evaluation of Alkenyldiarylmethane HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors That Possess Increased Hydrolytic Stability

Journal of Medicinal Chemistry ◽

10.1021/jm070382k ◽

2007 ◽

Vol 50 (20) ◽

pp. 4854-4867 ◽

Cited By ~ 17

Author(s):

Matthew D. Cullen ◽

Bo-Liang Deng ◽

Tracy L. Hartman ◽

Karen M. Watson ◽

Robert W. Buckheit, ◽

...

Keyword(s):

Reverse Transcriptase ◽

Hydrolytic Stability ◽

Biological Evaluation ◽

Hiv 1

Design, discovery, modelling, synthesis, and biological evaluation of novel and small, low toxicity s-triazine derivatives as HIV-1 non-nucleoside reverse transcriptase inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2016.04.018 ◽

2016 ◽

Vol 24 (11) ◽

pp. 2519-2529 ◽

Cited By ~ 13

Author(s):

Birgit Viira ◽

Anastasia Selyutina ◽

Alfonso T. García-Sosa ◽

Maarit Karonen ◽

Jari Sinkkonen ◽

...

Keyword(s):

Reverse Transcriptase ◽

Biological Evaluation ◽

Triazine Derivatives ◽

Low Toxicity ◽

Hiv 1

Design, Synthesis, and Biological Evaluation of 1-[(2-Benzyloxyl/alkoxyl)methyl]-5-halo-6-aryluracils as Potent HIV-1 Non-nucleoside Reverse Transcriptase Inhibitors with an Improved Drug Resistance Profile

Journal of Medicinal Chemistry ◽

10.1021/jm201506e ◽

2012 ◽

Vol 55 (5) ◽

pp. 2242-2250 ◽

Cited By ~ 26

Author(s):

Xiaowei Wang ◽

Jianfang Zhang ◽

Yang Huang ◽

Ruiping Wang ◽

Liang Zhang ◽

...

Keyword(s):

Drug Resistance ◽

Reverse Transcriptase ◽

Biological Evaluation ◽

Design Synthesis ◽

Resistance Profile ◽

Drug Resistance Profile ◽

Hiv 1

Synthesis and biological evaluation of novel 1-aryl-5-iodo-6-benzyluracils as potent HIV-1 non-nucleoside reverse transcriptase inhibitors

Journal of Chinese Pharmaceutical Sciences ◽

10.5246/jcps.2010.04.044 ◽

2010 ◽

Vol 19 (4) ◽

Author(s):

Wei Wang ◽

Jun-Yi Liu

Keyword(s):

Reverse Transcriptase ◽

Biological Evaluation ◽

Hiv 1

ChemInform Abstract: Structure-Based Design, Synthesis, and Biological Evaluation of Novel Pyrrolyl Aryl Sulfones (I): HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors Active at Nanomolar Concentrations.

ChemInform ◽

10.1002/chin.200030099 ◽

2010 ◽

Vol 31 (30) ◽

pp. no-no

Author(s):

Marino Artico ◽

et al. et al.

Keyword(s):

Reverse Transcriptase ◽

Biological Evaluation ◽

Design Synthesis ◽

Abstract Structure ◽

Hiv 1

Synthesis and biological evaluation of novel quinoxalinone-based HIV-1 reverse transcriptase inhibitors

MedChemComm ◽

10.1039/c3md00337j ◽

2014 ◽

Vol 5 (4) ◽

pp. 441-444 ◽

Cited By ~ 6

Author(s):

Jie Zhou ◽

Mingyu Ba ◽

Bo Wang ◽

Haibo Zhou ◽

Jianbo Bie ◽

...

Keyword(s):

Reverse Transcriptase ◽

Biological Evaluation ◽

Quinoxalinone Derivatives ◽

Anti Hiv ◽

Hiv 1

A series of novel quinoxalinone derivatives were identified as potent anti-HIV-1 agents with IC50 values at 10−8 μmol L−1 level.

Synthesis and biological evaluation of CHX-DAPYs as HIV-1 non-nucleoside reverse transcriptase inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2014.03.020 ◽

2014 ◽

Vol 22 (12) ◽

pp. 3220-3226 ◽

Cited By ~ 12

Author(s):

Zi-Hong Yan ◽

Hai-Qiu Wu ◽

Wen-Xue Chen ◽

Yan Wu ◽

Hu-Ri Piao ◽

...

Keyword(s):

Reverse Transcriptase ◽

Biological Evaluation ◽

Hiv 1

Synthesis and biological evaluation of 5′-O-dicarboxylic fatty acyl monoester derivatives of anti-HIV nucleoside reverse transcriptase inhibitors

Tetrahedron Letters ◽

10.1016/j.tetlet.2014.02.001 ◽

2014 ◽

Vol 55 (12) ◽

pp. 1983-1986 ◽

Cited By ~ 2

Author(s):

Bhanu Pemmaraju ◽

Hitesh K. Agarwal ◽

Donghoon Oh ◽

Karen W. Buckheit ◽

Robert W. Buckheit ◽

...

Keyword(s):

Reverse Transcriptase ◽

Biological Evaluation ◽

Fatty Acyl ◽

Derivatives Of ◽

Anti Hiv