Synthesis and Structure−Activity Relationships of 2-Substitutedd-Tryptophan-Containing Peptidic Endothelin Receptor Antagonists:  Importance of the C-2 Substituent of thed-Tryptophan Residue for Endothelin A and B Receptor Subtype Selectivity

1996 ◽  
Vol 39 (12) ◽  
pp. 2313-2330 ◽  
Author(s):  
Takehiro Fukami ◽  
Takeru Yamakawa ◽  
Kenji Niiyama ◽  
Hisaki Kojima ◽  
Yuuka Amano ◽  
...  
Keyword(s):  
Tryptophan Residue ◽  
Receptor Subtype ◽  
Endothelin Receptor Antagonists ◽  
Endothelin Receptor ◽  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Subtype Selectivity ◽  
Structure Activity ◽  
Endothelin A

Structure–Activity relationships of 2-substituted 5,7-Diarylcyclopenteno[1,2-b]pyridine-6-carboxylic acids as a novel class of endothelin receptor antagonists

2002 ◽  
Vol 12 (21) ◽  
pp. 3041-3045 ◽  
Author(s):  
Kenji Niiyama ◽  
Hirobumi Takahashi ◽  
Toshio Nagase ◽  
Hisaki Kojima ◽  
Yuka Amano ◽  
...  
Keyword(s):  
Carboxylic Acids ◽  
Endothelin Receptor Antagonists ◽  
Endothelin Receptor ◽  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Structure Activity

scholarly journals Synthesis and Structure-Activity Relationships in a Series of Ethenesulfonamide Derivatives, a Novel Class of Endothelin Receptor Antagonists.

2001 ◽  
Vol 49 (12) ◽  
pp. 1593-1603 ◽  
Author(s):  
Hironori HARADA ◽  
Jun-ichi KAZAMI ◽  
Susumu WATANUKI ◽  
Ryuji TSUZUKI ◽  
Katsumi SUDOH ◽  
...  
Keyword(s):  
Endothelin Receptor Antagonists ◽  
Endothelin Receptor ◽  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Structure Activity

Endothelin receptor antagonists: synthesis and structure–activity relationships of substituted benzothiazine-1,1-dioxides

1998 ◽  
Vol 6 (9) ◽  
pp. 1447-1456 ◽  
Author(s):  
K.A. Berryman ◽  
J.J. Edmunds ◽  
A.M. Bunker ◽  
S. Haleen ◽  
J. Bryant ◽  
...  
Keyword(s):  
Endothelin Receptor Antagonists ◽  
Endothelin Receptor ◽  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Structure Activity

ChemInform Abstract: Synthesis and Structure-Activity Relationships in a Series of Ethenesulfonamide Derivatives, a Novel Class of Endothelin Receptor Antagonists.

ChemInform ◽  
2010 ◽  
Vol 33 (17) ◽  
pp. no-no
Author(s):  
Hironori Harada ◽  
Jun-ichi Kazami ◽  
Susumu Watanuki ◽  
Ryuji Tsuzuki ◽  
Katsumi Sudoh ◽  
...  
Keyword(s):  
Endothelin Receptor Antagonists ◽  
Endothelin Receptor ◽  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Structure Activity

Selective endothelin A receptor antagonists. 2. Discovery and structure-activity relationships of 5-ketopentanoic acid derivatives

1997 ◽  
Vol 32 (6) ◽  
pp. 515-522 ◽  
Author(s):  
P.C. Astles ◽  
T.J. Brown ◽  
N.V. Harris ◽  
M.F. Harper ◽  
C McCarthy ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Endothelin A Receptor ◽  
Endothelin A

Synthesis and structure-activity relationships of 9-substituted acridines as endothelin-A receptor antagonists

1996 ◽  
Vol 6 (24) ◽  
pp. 2999-3002 ◽  
Author(s):  
X.-M. Cheng ◽  
C. Lee ◽  
S. Klutchko ◽  
T. Winters ◽  
E.E. Reynolds ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Endothelin A Receptor ◽  
Endothelin A

Selective Endothelin A Receptor Antagonists. 4. Discovery and Structure−Activity Relationships of Stilbene Acid and Alcohol Derivatives1-3

1998 ◽  
Vol 41 (15) ◽  
pp. 2745-2753 ◽  
Author(s):  
Peter C. Astles ◽  
Thomas J. Brown ◽  
Frank Halley ◽  
Caroline M. Handscombe ◽  
Neil V. Harris ◽  
...  
Keyword(s):  
Receptor Antagonists ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Endothelin A Receptor ◽  
Endothelin A
Sign in / Sign up

Export Citation Format

Share Document