Synthesis and Biological Evaluation of the 1,5-Diarylpyrazole Class of Cyclooxygenase-2 Inhibitors:  Identification of 4-[5-(4-Methylphenyl)-3- (trifluoromethyl)-1H-pyrazol-1-yl]benzenesulfonamide (SC-58635, Celecoxib)

1997 ◽  
Vol 40 (9) ◽  
pp. 1347-1365 ◽  
Author(s):  
Thomas D. Penning ◽  
John J. Talley ◽  
Stephen R. Bertenshaw ◽  
Jeffery S. Carter ◽  
Paul W. Collins ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Cyclooxygenase 2 ◽  
Synthesis And Biological Evaluation ◽  
Cyclooxygenase 2 Inhibitors

Synthesis and biological evaluation of new benzo-thieno[3,2-d]pyrimidin-4-one sulphonamide thio-derivatives as potential selective cyclooxygenase-2 inhibitors

2013 ◽  
Vol 17 (3) ◽  
pp. 445-458 ◽  
Author(s):  
Mariarita Barone ◽  
Adriana Carol Eleonora Graziano ◽  
Agostino Marrazzo ◽  
Pietro Gemmellaro ◽  
Andrea Santagati ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Cyclooxygenase 2 ◽  
Synthesis And Biological Evaluation ◽  
Cyclooxygenase 2 Inhibitors

Design, synthesis, and biological evaluation of (E)- and (Z)-styryl-2-acetoxyphenyl sulfides and sulfones as cyclooxygenase-2 inhibitors

2005 ◽  
Vol 13 (5) ◽  
pp. 1715-1723 ◽  
Author(s):  
M.V. Ramana Reddy ◽  
Muralidhar Reddy Mallireddigari ◽  
Venkat R. Pallela ◽  
Padmavathi Venkatapuram ◽  
Rengasamy Boominathan ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Cyclooxygenase 2 ◽  
Design Synthesis ◽  
Synthesis And Biological Evaluation ◽  
Cyclooxygenase 2 Inhibitors

Synthesis and Biological Evaluation of 3,4-Diaryloxazolones:  A New Class of Orally Active Cyclooxygenase-2 Inhibitors

2000 ◽  
Vol 43 (2) ◽  
pp. 214-223 ◽  
Author(s):  
Carles Puig ◽  
María I. Crespo ◽  
Núria Godessart ◽  
Joan Feixas ◽  
Javier Ibarzo ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Cyclooxygenase 2 ◽  
New Class ◽  
Orally Active ◽  
Synthesis And Biological Evaluation ◽  
Cyclooxygenase 2 Inhibitors
Sign in / Sign up

Export Citation Format

Share Document