Synthesis and Biological Evaluation of the Pyrazole Class of Cyclooxygenase- 2-Inhibitors

Design, Synthesis, and Biological Evaluation of 1,5-Diaryl-1,2,4-triazole Derivatives as Selective Cyclooxygenase-2 Inhibitors

Archiv der Pharmazie ◽

10.1002/ardp.200900227 ◽

2010 ◽

Vol 343 (9) ◽

pp. 500-508 ◽

Cited By ~ 12

Author(s):

Bo Jiang ◽

Yi Zeng ◽

Meng-Jie Li ◽

Jin-Yi Xu ◽

Yong-Na Zhang ◽

...

Keyword(s):

Biological Evaluation ◽

Cyclooxygenase 2 ◽

Design Synthesis ◽

Triazole Derivatives ◽

Synthesis and biological evaluation of new benzo-thieno[3,2-d]pyrimidin-4-one sulphonamide thio-derivatives as potential selective cyclooxygenase-2 inhibitors

Molecular Diversity ◽

10.1007/s11030-013-9443-0 ◽

2013 ◽

Vol 17 (3) ◽

pp. 445-458 ◽

Cited By ~ 10

Author(s):

Mariarita Barone ◽

Adriana Carol Eleonora Graziano ◽

Agostino Marrazzo ◽

Pietro Gemmellaro ◽

Andrea Santagati ◽

...

Keyword(s):

Biological Evaluation ◽

Cyclooxygenase 2 ◽

ChemInform Abstract: Synthesis and Biological Evaluation of the 1,5-Diarylpyrazole Class of Cyclooxygenase-2 Inhibitors: Identification of 4-(5-(4-Methylphenyl)-3- (trifluoromethyl)-1H-pyrazol-1-yl)benzenesulfonamide (SC-58635, Celecoxib).

ChemInform ◽

10.1002/chin.199736141 ◽

2010 ◽

Vol 28 (36) ◽

pp. no-no

Author(s):

T. D. PENNING ◽

J. J. TALLAY ◽

S. R. BERTENSHAW ◽

J. S. CARTER ◽

P. W. COLLINS ◽

...

Keyword(s):

Biological Evaluation ◽

Cyclooxygenase 2 ◽

Synthesis and Biological Evaluation of the 1,5-Diarylpyrazole Class of Cyclooxygenase-2 Inhibitors: Identification of 4-[5-(4-Methylphenyl)-3- (trifluoromethyl)-1H-pyrazol-1-yl]benzenesulfonamide (SC-58635, Celecoxib)

Journal of Medicinal Chemistry ◽

10.1021/jm960803q ◽

1997 ◽

Vol 40 (9) ◽

pp. 1347-1365 ◽

Cited By ~ 1366

Author(s):

Thomas D. Penning ◽

John J. Talley ◽

Stephen R. Bertenshaw ◽

Jeffery S. Carter ◽

Paul W. Collins ◽

...

Keyword(s):

Biological Evaluation ◽

Cyclooxygenase 2 ◽

ChemInform Abstract: Design, Synthesis, and Biological Evaluation of 1,5-Diaryl-1,2,4-triazole Derivatives as Selective Cyclooxygenase-2 Inhibitors.

ChemInform ◽

10.1002/chin.201052210 ◽

2010 ◽

Vol 41 (52) ◽

pp. no-no

Author(s):

Bo Jiang ◽

Yi Zeng ◽

Meng-Jie Li ◽

Jin-Yi Xu ◽

Yong-Na Zhang ◽

...

Keyword(s):

Biological Evaluation ◽

Cyclooxygenase 2 ◽

Design Synthesis ◽

Triazole Derivatives ◽

Design, synthesis and biological evaluation of new 2,3-diarylquinoline derivatives as selective cyclooxygenase-2 inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2009.12.060 ◽

2010 ◽

Vol 18 (3) ◽

pp. 1029-1033 ◽

Cited By ~ 32

Author(s):

Razieh Ghodsi ◽

Afshin Zarghi ◽

Bahram Daraei ◽

Mehdi Hedayati

Keyword(s):

Biological Evaluation ◽

Cyclooxygenase 2 ◽

Design Synthesis ◽

Design, Synthesis and Biological Evaluation of New 5,5-Diarylhydantoin Derivatives as Selective Cyclooxygenase-2 Inhibitors

Scientia Pharmaceutica ◽

10.3797/scipharm.1104-20 ◽

2011 ◽

Vol 79 (3) ◽

pp. 449-460 ◽

Cited By ~ 7

Author(s):

Afshin ZARGHI

Keyword(s):

Biological Evaluation ◽

Cyclooxygenase 2 ◽

Design Synthesis ◽

Design, synthesis, and biological evaluation of (E)- and (Z)-styryl-2-acetoxyphenyl sulfides and sulfones as cyclooxygenase-2 inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2004.12.005 ◽

2005 ◽

Vol 13 (5) ◽

pp. 1715-1723 ◽

Cited By ~ 18

Author(s):

M.V. Ramana Reddy ◽

Muralidhar Reddy Mallireddigari ◽

Venkat R. Pallela ◽

Padmavathi Venkatapuram ◽

Rengasamy Boominathan ◽

...

Keyword(s):

Biological Evaluation ◽

Cyclooxygenase 2 ◽

Design Synthesis ◽

Synthesis and Biological Evaluation of 3,4-Diaryloxazolones: A New Class of Orally Active Cyclooxygenase-2 Inhibitors

Journal of Medicinal Chemistry ◽

10.1021/jm991106b ◽

2000 ◽

Vol 43 (2) ◽

pp. 214-223 ◽

Cited By ~ 60

Author(s):

Carles Puig ◽

María I. Crespo ◽

Núria Godessart ◽

Joan Feixas ◽

Javier Ibarzo ◽

...

Keyword(s):

Biological Evaluation ◽

Cyclooxygenase 2 ◽

New Class ◽

Orally Active ◽

ChemInform Abstract: Synthesis and Biological Evaluation of 3,4-Diaryloxazolones: A New Class of Orally Active Cyclooxygenase-2 Inhibitors.

ChemInform ◽

10.1002/chin.200016121 ◽

2010 ◽

Vol 31 (16) ◽

pp. no-no

Author(s):

Maria I. Crespo ◽

et al. et al.

Keyword(s):

Biological Evaluation ◽

Cyclooxygenase 2 ◽

New Class ◽

Orally Active ◽