Solid-Phase Synthesis of 4-Arylazetidin-2-ones via Suzuki and Heck Cross-Coupling Reactions

1997 ◽  
Vol 62 (22) ◽  
pp. 7820-7826 ◽  
Author(s):  
Beatrice Ruhland ◽  
Agnes Bombrun ◽  
Mark A. Gallop
Keyword(s):  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Cross Coupling ◽  
Coupling Reactions ◽  
Phase Synthesis ◽  
Cross Coupling Reactions

Solid-Phase Synthesis of Oligo(triacetylene)s and Oligo(phenylenetriacetylene)s EmployingSonogashira andCadiotChodkiewicz-Type Cross-Coupling Reactions

2004 ◽  
Vol 87 (3) ◽  
pp. 698-718 ◽  
Author(s):  
Nils F. Utesch ◽  
François Diederich ◽  
Corinne Boudon ◽  
Jean-Paul Gisselbrecht ◽  
Maurice Gross
Keyword(s):  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Cross Coupling ◽  
Coupling Reactions ◽  
Phase Synthesis ◽  
Cross Coupling Reactions

A general solid phase synthesis of 4-substituted quinolinones via Pd-catalyzed cross coupling

2006 ◽  
Vol 47 (28) ◽  
pp. 4885-4888 ◽  
Author(s):  
Caiding Xu ◽  
Lydie Yang ◽  
Ashok Bhandari ◽  
Christopher P. Holmes
Keyword(s):  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Cross Coupling ◽  
Phase Synthesis

Solid-phase synthesis of 5-arylhistidines via a microwave-assisted Suzuki–Miyaura cross-coupling

Tetrahedron ◽  
2008 ◽  
Vol 64 (46) ◽  
pp. 10538-10545 ◽  
Author(s):  
Vanessa Cerezo ◽  
Muriel Amblard ◽  
Jean Martinez ◽  
Pascal Verdié ◽  
Marta Planas ◽  
...  
Keyword(s):  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Cross Coupling ◽  
Phase Synthesis ◽  
Microwave Assisted

Solid-phase Suzuki cross-coupling reactions using a phosphine ligand based on a phospha-adamantane framework

2004 ◽  
Vol 45 (29) ◽  
pp. 5661-5663 ◽  
Author(s):  
Stephan A. Ohnmacht ◽  
Tim Brenstrum ◽  
Konrad H. Bleicher ◽  
James McNulty ◽  
Alfredo Capretta
Keyword(s):  
Solid Phase ◽  
Cross Coupling ◽  
Phosphine Ligand ◽  
Coupling Reactions ◽  
Cross Coupling Reactions

Solid-Phase Synthesis of 5-Arylhistidine-Containing Peptides with Antimicrobial Activity Through a Microwave-Assisted Suzuki-Miyaura Cross-Coupling

2012 ◽  
Vol 2012 (23) ◽  
pp. 4321-4332 ◽  
Author(s):  
Iteng Ng-Choi ◽  
Marta Soler ◽  
Vanessa Cerezo ◽  
Esther Badosa ◽  
Emilio Montesinos ◽  
...  
Keyword(s):  
Antimicrobial Activity ◽  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Cross Coupling ◽  
Phase Synthesis ◽  
Microwave Assisted

Combinatorial Solid-Phase Synthesis of 6-Aryl-1,3,5-triazines via Suzuki Coupling

2011 ◽  
Vol 64 (5) ◽  
pp. 540 ◽  
Author(s):  
Jae Wook Lee ◽  
Hyung-Ho Ha ◽  
Marc Vendrell ◽  
Jacqueline T. Bork ◽  
Young-Tae Chang
Keyword(s):  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Cross Coupling ◽  
Structural Diversity ◽  
Suzuki Coupling ◽  
Purification Step ◽  
Solid Supports ◽  
Phase Synthesis ◽  
Triazine Derivatives ◽  
Polymer Supported

A synthetic methodology to prepare collections of trisubstituted aryl 1,3,5-triazines with broad structural diversity via Suzuki coupling has been developed. We first optimized the combinatorial derivatization of the triazine core using Suzuki cross-coupling. Second, in order to further expand the methodology for the preparation of negatively charged triazines, we adapted this approach to polymer-supported amino acids and prepared aryl triazines with different charge distribution. With a collection of 160 aryl triazine derivatives in good purities and without any purification step, we proved the viability of this orthogonal scheme for the preparation of triazine libraries using amine/amino acid-captured solid supports and Suzuki cross-coupling.

Solid Phase Synthesis of 2-substituted Melatonin Derivativesvia Palladium-mediated Coupling Reactions using Microwave Irradiation

2004 ◽  
Vol 23 (10) ◽  
pp. 850-853 ◽  
Author(s):  
Aur�lie Berthault ◽  
Sabine Berteina-Raboin ◽  
Adriana Finaru ◽  
G�rald Guillaumet
Keyword(s):  
Microwave Irradiation ◽  
Solid Phase Synthesis ◽  
Solid Phase ◽  
Coupling Reactions ◽  
Phase Synthesis
Sign in / Sign up

Export Citation Format

Share Document