Synthesis, radiosynthesis, in vitro and first in vivo evaluation of a new matrix metalloproteinase inhibitor based on γ-fluorinated α-sulfonylaminohydroxamic acid

In Vivo Evaluation ◽

Metalloproteinase Inhibitor

Characterisation of a novel matrix metalloproteinase inhibitor on pancreatic adenocarcinoma cells in vitro and in an orthotopic pancreatic cancer model in vivo

International Journal of Oncology ◽

10.3892/ijo.32.1.273 ◽

2008 ◽

Author(s):

Matthias Kapischke ◽

Tim Fischer ◽

Katrin Tiessen ◽

Harald Tschesche ◽

Hans-Peter Bruch ◽

...

Keyword(s):

Pancreatic Cancer ◽

Pancreatic Adenocarcinoma ◽

Cancer Model ◽

Adenocarcinoma Cells

In vitro pharmacological profiles and in vivo anti-angiogenesis activity of S-3304, a novel matrix metalloproteinase inhibitor

European Journal of Cancer ◽

10.1016/s0959-8049(02)80910-8 ◽

2002 ◽

Vol 38 ◽

pp. S81

Keyword(s):

Pharmacological Profiles

RGD peptide grafted polybutylene adipate-co-terephthalate/gelatin electrospun nanofibers loaded with a matrix metalloproteinase inhibitor drug for alleviating of wounds: an in vitro/in vivo study

Drug Development and Industrial Pharmacy ◽

10.1080/03639045.2020.1730397 ◽

2020 ◽

Vol 46 (3) ◽

pp. 484-497 ◽

Cited By ~ 2

Author(s):

Jaleh Varshosaz ◽

Khatereh Arabloo ◽

Nasim Sarrami ◽

Erfaneh Ghassami ◽

Emadeddin Yazdani Kachouei ◽

...

Keyword(s):

Electrospun Nanofibers ◽

Rgd Peptide ◽

In Vivo Study ◽

Inhibitor Drug

Design, (Radio)Synthesis, and in Vitro and in Vivo Evaluation of Highly Selective and Potent Matrix Metalloproteinase 12 (MMP-12) Inhibitors as Radiotracers for Positron Emission Tomography

Journal of Medicinal Chemistry ◽

10.1021/acs.jmedchem.8b00200 ◽

2018 ◽

Vol 61 (9) ◽

pp. 4115-4134 ◽

Cited By ~ 17

Author(s):

Viktoria Butsch ◽

Frederik Börgel ◽

Fabian Galla ◽

Katrin Schwegmann ◽

Sven Hermann ◽

...

Keyword(s):

Positron Emission Tomography ◽

Emission Tomography ◽

In Vivo Evaluation ◽

Positron Emission ◽

Matrix Metalloproteinase 12

Synthesis, radiosynthesis, in vitro and preliminary in vivo evaluation of biphenyl carboxylic and hydroxamic matrix metalloproteinase (MMP) inhibitors as potential tumor imaging agents

Applied Radiation and Isotopes ◽

10.1016/j.apradiso.2004.12.009 ◽

2005 ◽

Vol 62 (6) ◽

pp. 903-913 ◽

Cited By ~ 7

Author(s):

Ruth Oltenfreiter ◽

Ludovicus Staelens ◽

Ulrik Hillaert ◽

An Heremans ◽

Agnes Noël ◽

...

Keyword(s):

Tumor Imaging ◽

Imaging Agents ◽

In Vivo Evaluation ◽

Mmp Inhibitors

Expression of Matrix Metalloproteinases in Gastric Carcinoma and Possibility of Clinical Application of Matrix Metalloproteinase Inhibitor in Vivo

Annals of the New York Academy of Sciences ◽

10.1111/j.1749-6632.1999.tb07721.x ◽

1999 ◽

Vol 878 (1 INHIBITION OF) ◽

pp. 541-543 ◽

Cited By ~ 1

Author(s):

YOSHIHIDE OTANI ◽

TETSURO KUBOTA ◽

YOSHIHIKO SAKURAI ◽

NAOKI IGARASHI ◽

TAKEYOSHI YOKOYAMA ◽

...

Keyword(s):

Matrix Metalloproteinases ◽

Gastric Carcinoma ◽

Clinical Application ◽

Metalloproteinase Inhibitor

Effect of Matrix Metalloproteinase Inhibitor from Mulberry fruit extract on the Microtensile Bond Strength Stability: An in vitro Study

Egyptian Dental Journal ◽

10.21608/edj.2019.72811 ◽

2019 ◽

Vol 65 (1) ◽

pp. 541-550

Author(s):

Rania Mosallam ◽

Nermin Younis ◽

Hadeel Farouk ◽

Osama Mosallam

Keyword(s):

Bond Strength ◽

In Vitro Study ◽

Vitro Study ◽

Microtensile Bond Strength ◽

Fruit Extract ◽

Mulberry Fruit

Inverse 1,2,3-Triazole-1-yl-ethyl Substituted Hydroxamates as Highly Potent Matrix Metalloproteinase Inhibitors: (Radio)synthesis, in Vitro and First in Vivo Evaluation

Journal of Medicinal Chemistry ◽

10.1021/jm4006753 ◽

2013 ◽

Vol 56 (17) ◽

pp. 6858-6870 ◽

Cited By ~ 28

Author(s):

Verena Hugenberg ◽

Burkhard Riemann ◽

Sven Hermann ◽

Otmar Schober ◽

Michael Schäfers ◽

...

Keyword(s):

Matrix Metalloproteinase Inhibitors ◽

In Vivo Evaluation ◽

Metalloproteinase Inhibitors

Radiolabeled Selective Matrix Metalloproteinase 13 (MMP-13) Inhibitors: (Radio)Syntheses and in Vitro and First in Vivo Evaluation

Journal of Medicinal Chemistry ◽

10.1021/acs.jmedchem.6b01284 ◽

2016 ◽

Vol 60 (1) ◽

pp. 307-321 ◽

Cited By ~ 10

Author(s):

Verena Hugenberg ◽

Stefan Wagner ◽

Klaus Kopka ◽

Michael Schäfers ◽

Robert C. Schuit ◽

...

Keyword(s):

In Vivo Evaluation ◽

Matrix Metalloproteinase 13

Matrix Metalloproteinase Inhibitor CGS 27023A Protects COMP and Proteoglycan in the Bovine Articular Cartilage but not the Release of Their Fragments from Cartilage after Prolonged Stimulation in Vitro with IL-1alpha

Annals of the New York Academy of Sciences ◽

10.1111/j.1749-6632.1999.tb07740.x ◽

1999 ◽

Vol 878 (1 INHIBITION OF) ◽

pp. 607-611 ◽

Cited By ~ 6

Author(s):

VISHWAS GANU ◽

RICHARD MELTON ◽

WEIGWANG WANG ◽

DON ROBERTS

Keyword(s):

Articular Cartilage ◽

Bovine Articular Cartilage ◽

Prolonged Stimulation