Quantitative Structure-Activity Relationship Studies on Matrix Metalloproteinase Inhibitors: Bicyclic Heteroaryl Hydroxamic Acid Analogs

Letters in Drug Design & Discovery ◽

10.2174/157018005774479096 ◽

2005 ◽

Vol 2 (7) ◽

pp. 522-528 ◽

Author(s):

S. Gupta ◽

S. Kumaran

Keyword(s):

Matrix Metalloproteinase ◽

Hydroxamic Acid ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Matrix Metalloproteinase Inhibitors ◽

Structure Activity ◽

Metalloproteinase Inhibitors

Download Full-text

Quantitative Structure-Activity Relationship Studies on Matrix Metalloproteinase Inhibitors: Piperazine, Piperidine and Diazepine Hydroxamic Acid Analogs

Asian Journal of Biochemistry ◽

10.3923/ajb.2006.211.223 ◽

2006 ◽

Vol 1 (3) ◽

pp. 211-223 ◽

Author(s):

S.P. Gupta ◽

S. Kumaran

Keyword(s):

Matrix Metalloproteinase ◽

Hydroxamic Acid ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Matrix Metalloproteinase Inhibitors ◽

Structure Activity ◽

Metalloproteinase Inhibitors

Download Full-text

A Quantitative Structure-Activity Relationship Study on a Novel Series of Hydroxamic Acid Analogs Acting as Matrix Metalloproteinase Inhibitors

Letters in Drug Design & Discovery ◽

10.2174/157018008784619852 ◽

2008 ◽

Vol 5 (4) ◽

pp. 281-285 ◽

Author(s):

S. Gupta ◽

Priyanka Bagaria ◽

V. Kumar Satuluri

Keyword(s):

Matrix Metalloproteinase ◽

Hydroxamic Acid ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Matrix Metalloproteinase Inhibitors ◽

Structure Activity ◽

Metalloproteinase Inhibitors ◽

Relationship Study

Download Full-text

Quantitative Structure-Activity Relationship Studies on Matrix Metalloproteinase Inhibitors: Hydroxamic Acid Analogs

Medicinal Chemistry ◽

10.2174/157340606776930790 ◽

2006 ◽

Vol 2 (3) ◽

pp. 243-250 ◽

Author(s):

S. Gupta ◽

S. Kumaran

Keyword(s):

Matrix Metalloproteinase ◽

Hydroxamic Acid ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Matrix Metalloproteinase Inhibitors ◽

Structure Activity ◽

Metalloproteinase Inhibitors

Download Full-text

A Quantitative Structure-Activity Relationship Study on Some Novel Series of Hydroxamic Acid Analogs Acting as Matrix Metalloproteinase Inhibitors

Medicinal Chemistry ◽

10.2174/157340607780059477 ◽

2007 ◽

Vol 3 (2) ◽

pp. 167-173 ◽

Author(s):

S. Kumaran ◽

S. Gupta

Keyword(s):

Matrix Metalloproteinase ◽

Hydroxamic Acid ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Matrix Metalloproteinase Inhibitors ◽

Structure Activity ◽

Metalloproteinase Inhibitors ◽

Relationship Study

Download Full-text

A quantitative structure-activity relationship study on matrix metalloproteinase inhibitors: Piperidine sulfonamide aryl hydroxamic acid analogs

Journal of Enzyme Inhibition and Medicinal Chemistry ◽

10.1080/14756360600956655 ◽

2007 ◽

Vol 22 (1) ◽

pp. 23-27 ◽

Author(s):

S. Kumaran ◽

S. P. Gupta

Keyword(s):

Matrix Metalloproteinase ◽

Hydroxamic Acid ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Matrix Metalloproteinase Inhibitors ◽

Structure Activity ◽

Metalloproteinase Inhibitors ◽

Relationship Study

Download Full-text

A quantitative structure–activity relationship study on some series of anthranilic acid-based matrix metalloproteinase inhibitors

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2005.05.055 ◽

2005 ◽

Vol 13 (18) ◽

pp. 5454-5462 ◽

Author(s):

S.P. Gupta ◽

S. Kumaran

Keyword(s):

Matrix Metalloproteinase ◽

Anthranilic Acid ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Matrix Metalloproteinase Inhibitors ◽

Structure Activity ◽

Metalloproteinase Inhibitors ◽

Relationship Study

Download Full-text

A quantitative structure–activity relationship study of hydroxamate matrix metalloproteinase inhibitors derived from funtionalized 4-aminoprolines

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(03)00069-5 ◽

2003 ◽

Vol 11 (9) ◽

pp. 1975-1981 ◽

Author(s):

S.P. Gupta ◽

Dalip Kumar ◽

S. Kumaran

Keyword(s):

Matrix Metalloproteinase ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Quantitative Structure ◽

Matrix Metalloproteinase Inhibitors ◽

Structure Activity ◽

Metalloproteinase Inhibitors ◽

Relationship Study

Download Full-text

Three-dimensional quantitative structure-activity relationship (CoMFA and CoMSIA) studies on galardin derivatives as gelatinase A (matrix metalloproteinase 2) inhibitors

Journal of Enzyme Inhibition and Medicinal Chemistry ◽

10.1080/14756360701632221 ◽

2008 ◽

Vol 23 (4) ◽

pp. 445-453 ◽

Author(s):

Jianbin Zheng ◽

Ren Wen ◽

Dominique Guillaume

Keyword(s):

Matrix Metalloproteinase ◽

Three Dimensional ◽

Quantitative Structure Activity Relationship ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Matrix Metalloproteinase 2 ◽

Gelatinase A ◽

Quantitative Structure ◽

Structure Activity

Download Full-text

Synthesis and Structure−Activity Relationship of α-Sulfonylhydroxamic Acids as Novel, Orally Active Matrix Metalloproteinase Inhibitors for the Treatment of Osteoarthritis

Journal of Medicinal Chemistry ◽

10.1021/jm0205548 ◽

2003 ◽

Vol 46 (12) ◽

pp. 2361-2375 ◽

Author(s):

Venkatesan Aranapakam ◽

George T. Grosu ◽

Jamie M. Davis ◽

Baihua Hu ◽

John Ellingboe ◽

...

Keyword(s):

Matrix Metalloproteinase ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Matrix Metalloproteinase Inhibitors ◽

Active Matrix ◽

Structure Activity ◽

Metalloproteinase Inhibitors ◽

Relationship Of ◽

Download Full-text

Tetrahydroisoquinoline-3-carboxylate based matrix-metalloproteinase inhibitors: design, synthesis and structure–activity relationship

Bioorganic & Medicinal Chemistry ◽

10.1016/s0968-0896(02)00215-8 ◽

2002 ◽

Vol 10 (11) ◽

pp. 3529-3544 ◽

Author(s):

Hans Matter ◽

Manfred Schudok ◽

Wilfried Schwab ◽

Werner Thorwart ◽

Denis Barbier ◽

...

Keyword(s):

Matrix Metalloproteinase ◽

Structure Activity Relationship ◽

Activity Relationship ◽

Matrix Metalloproteinase Inhibitors ◽

Design Synthesis ◽

Structure Activity ◽

Metalloproteinase Inhibitors

Download Full-text