11C-NS14492 as a Novel PET Radioligand for Imaging Cerebral  7 Nicotinic Acetylcholine Receptors: In Vivo Evaluation and Drug Occupancy Measurements

Acetylcholine Receptors ◽

In Vivo Evaluation ◽

A Promising PET Tracer for Imaging of α7 Nicotinic Acetylcholine Receptors in the Brain: Design, Synthesis, and in Vivo Evaluation of a Dibenzothiophene-Based Radioligand

Molecules ◽

10.3390/molecules201018387 ◽

2015 ◽

Vol 20 (10) ◽

pp. 18387-18421 ◽

Cited By ~ 11

Author(s):

Rodrigo Teodoro ◽

Matthias Scheunemann ◽

Winnie Deuther-Conrad ◽

Barbara Wenzel ◽

Francesca Fasoli ◽

...

Keyword(s):

Acetylcholine Receptors ◽

In Vivo Evaluation ◽

Nicotinic Acetylcholine ◽

Design Synthesis ◽

Pet Tracer ◽

Α7 Nicotinic Acetylcholine Receptors ◽

The Brain

NIDA522131, a new radioligand for imaging extrathalamic nicotinic acetylcholine receptors: in vitro and in vivo evaluation

Journal of Neurochemistry ◽

10.1111/j.1471-4159.2007.05009.x ◽

2007 ◽

Vol 0 (0) ◽

pp. 071106220615006-???

Author(s):

Svetlana I. Chefer ◽

Olga A. Pavlova ◽

Yi Zhang ◽

D. Bruce Vaupel ◽

Alane S. Kimes ◽

...

Keyword(s):

Acetylcholine Receptors ◽

In Vivo Evaluation ◽

The Prototoxin lynx1 Acts on Nicotinic Acetylcholine Receptors to Balance Neuronal Activity and Survival In Vivo

Neuron ◽

10.1016/j.neuron.2006.07.025 ◽

2006 ◽

Vol 51 (5) ◽

pp. 587-600 ◽

Cited By ~ 89

Author(s):

Julie M. Miwa ◽

Tanya R. Stevens ◽

Sarah L. King ◽

Barbara J. Caldarone ◽

Ines Ibanez-Tallon ◽

...

Keyword(s):

Neuronal Activity ◽

Acetylcholine Receptors ◽

LC-MS Supported Studies on the in Vitro Metabolism of both Enantiomers of Flubatine and the in Vivo Metabolism of (+)-[18F]Flubatine—A Positron Emission Tomography Radioligand for Imaging α4β2 Nicotinic Acetylcholine Receptors

Molecules ◽

10.3390/molecules21091200 ◽

2016 ◽

Vol 21 (9) ◽

pp. 1200 ◽

Cited By ~ 7

Author(s):

Friedrich-Alexander Ludwig ◽

René Smits ◽

Steffen Fischer ◽

Cornelius Donat ◽

Alexander Hoepping ◽

...

Keyword(s):

Positron Emission Tomography ◽

Acetylcholine Receptors ◽

In Vitro Metabolism ◽

Emission Tomography ◽

In Vivo Metabolism ◽

Nicotinic Acetylcholine ◽

Positron Emission

Activation of nicotinic acetylcholine receptors induces long-term potentiation in vivo in the intact mouse dentate gyrus

European Journal of Neuroscience ◽

10.1046/j.1460-9568.2000.00259.x ◽

2000 ◽

Vol 12 (10) ◽

pp. 3741-3747 ◽

Cited By ~ 108

Author(s):

Shogo Matsuyama ◽

Akira Matsumoto ◽

Taira Enomoto ◽

Tomoyuki Nishizaki

Keyword(s):

Dentate Gyrus ◽

Acetylcholine Receptors ◽

Long Term Potentiation ◽

Intact Mouse ◽

Nicotinic Acetylcholine ◽

Term Potentiation

Methanandamide Allosterically Inhibits in Vivo the Function of Peripheral Nicotinic Acetylcholine Receptors Containing the α7-Subunit

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.108.140863 ◽

2008 ◽

Vol 326 (3) ◽

pp. 912-919 ◽

Cited By ~ 14

Author(s):

Urszula Baranowska ◽

Manfred Göthert ◽

Radosław Rudź ◽

Barbara Malinowska

Keyword(s):

Acetylcholine Receptors ◽

Nicotinic Acetylcholine ◽

Α7 Subunit

In vivo quantification of the greater densities of alpha4beta2* nicotinic acetylcholine receptors in smokers compared to non-smokers

NeuroImage ◽

10.1016/j.neuroimage.2006.04.136 ◽

2006 ◽

Vol 31 ◽

pp. T153 ◽

Cited By ~ 2

Author(s):

Alane S. Kimes ◽

S. Chefer ◽

C.S. Contoreggi ◽

A. Hall ◽

A. Horti ◽

...

Keyword(s):

Acetylcholine Receptors ◽

Pharmacology, toxicology, and radiation dosimetry evaluation of [123I]5-I-A-85380, a radioligand for in vivo imaging of cerebral neuronal nicotinic acetylcholine receptors in humans

Drug Development Research ◽

10.1002/ddr.10152 ◽

2003 ◽

Vol 58 (2) ◽

pp. 149-168 ◽

Cited By ~ 11

Author(s):

D. Bruce Vaupel ◽

Srihari R. Tella ◽

David L. Huso ◽

Alexey G. Mukhin ◽

Ira Baum ◽

...

Keyword(s):

In Vivo Imaging ◽

Acetylcholine Receptors ◽

Radiation Dosimetry ◽

Neuronal Nicotinic Acetylcholine Receptors ◽

In Vivo Activation of Midbrain Dopamine Neurons via Sensitized, High-Affinity α6∗ Nicotinic Acetylcholine Receptors

Neuron ◽

10.1016/j.neuron.2008.09.009 ◽

2008 ◽

Vol 60 (1) ◽

pp. 123-136 ◽

Cited By ~ 144

Author(s):

Ryan M. Drenan ◽

Sharon R. Grady ◽

Paul Whiteaker ◽

Tristan McClure-Begley ◽

Sheri McKinney ◽

...

Keyword(s):

Acetylcholine Receptors ◽

Dopamine Neurons ◽

Nicotinic Acetylcholine ◽

High Affinity ◽

Midbrain Dopamine ◽

Midbrain Dopamine Neurons

In vivo measurement of nicotinic acetylcholine receptors with [18F]norchloro-fluoro-homoepibatidine

Synapse ◽

10.1002/syn.20480 ◽

2008 ◽

Vol 62 (3) ◽

pp. 205-218 ◽

Cited By ~ 35

Author(s):

Peter Brust ◽

Jörg Thomas Patt ◽

Winnie Deuther-Conrad ◽

Georg Becker ◽

Marianne Patt ◽

...

Keyword(s):

Acetylcholine Receptors ◽

Nicotinic Acetylcholine ◽

In Vivo Measurement