Pharmacology, toxicology, and radiation dosimetry evaluation of [123I]5-I-A-85380, a radioligand for in vivo imaging of cerebral neuronal nicotinic acetylcholine receptors in humans

In Vivo Imaging ◽

Acetylcholine Receptors ◽

Radiation Dosimetry ◽

Synthesis of 2-[18F]fluoro-3-[2(S)-2-azetidinylmethoxy]pyridine, a highly potent radioligand for in vivo imaging central nicotinic acetylcholine receptors

Journal of Labelled Compounds and Radiopharmaceuticals ◽

10.1002/(sici)1099-1344(199805)41:5<451::aid-jlcr111>3.0.co;2-r ◽

1998 ◽

Vol 41 (5) ◽

pp. 451-463 ◽

Cited By ~ 57

Author(s):

Frédéric Dolle ◽

Héric Valette ◽

Michel Bottlaender ◽

Françoise Hinnen ◽

Françoise Vaufrey ◽

...

Keyword(s):

In Vivo Imaging ◽

Acetylcholine Receptors ◽

In vivo labeling of neuronal nicotinic acetylcholine receptors with radiolabeled isomers of norchloroepibatidine

Neuroreport ◽

10.1097/00001756-199512150-00011 ◽

1995 ◽

Vol 6 (18) ◽

pp. 2483-2488 ◽

Cited By ~ 18

Author(s):

Ursula Scheffel ◽

George F. Taylor ◽

John A. Kepler ◽

F. Ivy Carroll ◽

Michael J. Kuhar

Keyword(s):

Acetylcholine Receptors ◽

Nicotinic Acetylcholine ◽

In Vivo Labeling

Synthesis of 3-[(1-[11C]methyl-2(S)-pyrrolidinyl) methoxy]pyridine and 3-[(1-[11C]methyl-2(R)-pyrrolidinyl) methoxy]pyridine: Radioligands for in vivo studies of neuronal nicotinic acetylcholine receptors

Journal of Labelled Compounds and Radiopharmaceuticals ◽

10.1002/(sici)1099-1344(199705)39:5<425::aid-jlcr984>3.0.co;2-r ◽

1997 ◽

Vol 39 (5) ◽

pp. 425-431 ◽

Cited By ~ 7

Author(s):

Michael Kassiou ◽

Hayden T. Ravert ◽

William B. Mathews ◽

John L. Musachio ◽

Edythe D. London ◽

...

Keyword(s):

Acetylcholine Receptors ◽

In Vivo Studies ◽

The Quest for Eldorado: Development of Radioligands for In Vivo Imaging of Nicotinic Acetylcholine Receptors in Human Brain

Current Pharmaceutical Design ◽

10.2174/138161206778559605 ◽

2006 ◽

Vol 12 (30) ◽

Cited By ~ 39

Author(s):

Andrew G. Horti ◽

Victor L. Villemagne

Keyword(s):

Human Brain ◽

In Vivo Imaging ◽

Acetylcholine Receptors ◽

In Vitro and in Vivo Neuronal Nicotinic Receptor Properties of (+)- and (−)-Pyrido[3,4]homotropane [(+)- and (−)-PHT]: (+)-PHT Is a Potent and Selective Full Agonist at α6β2 Containing Neuronal Nicotinic Acetylcholine Receptors

ACS Chemical Neuroscience ◽

10.1021/acschemneuro.5b00077 ◽

2015 ◽

Vol 6 (6) ◽

pp. 920-926 ◽

Cited By ~ 6

Author(s):

F. Ivy Carroll ◽

Hernán A. Navarro ◽

S. Wayne Mascarella ◽

Ana H. Castro ◽

Charles W. Luetje ◽

...

Keyword(s):

Nicotinic Receptor ◽

Acetylcholine Receptors ◽

Nicotinic Acetylcholine ◽

Full Agonist ◽

Neuronal Nicotinic Receptor

Methyllycaconitine: A non-radiolabeled ligand for mapping α7 neuronal nicotinic acetylcholine receptors — In vivo target localization and biodistribution in rat brain

Journal of Pharmacological and Toxicological Methods ◽

10.1016/j.vascn.2012.05.003 ◽

2012 ◽

Vol 66 (1) ◽

pp. 22-28 ◽

Cited By ~ 8

Author(s):

Ramakrishna Nirogi ◽

Vishwottam Kandikere ◽

Gopinadh Bhyrapuneni ◽

Ramanatha Saralaya ◽

Nageswararao Muddana ◽

...

Keyword(s):

Rat Brain ◽

Acetylcholine Receptors ◽

Target Localization ◽

Synthesis and biological evaluation of novel carbon-11 labeled pyridyl ethers: candidate ligands for in vivo imaging of α4β2 nicotinic acetylcholine receptors (α4β2-nAChRs) in the brain with positron emission tomography

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2009.05.021 ◽

2009 ◽

Vol 17 (13) ◽

pp. 4367-4377 ◽

Cited By ~ 6

Author(s):

Yongjun Gao ◽

Hayden T. Ravert ◽

Hiroto Kuwabara ◽

Yingxian Xiao ◽

Christopher J. Endres ◽

...

Keyword(s):

In Vivo Imaging ◽

Acetylcholine Receptors ◽

Biological Evaluation ◽

Emission Tomography ◽

Nicotinic Acetylcholine ◽

Positron Emission ◽

Synthesis And Biological Evaluation ◽

The Brain

Pharmacological evaluation of [11C]A-84543: An enantioselective ligand for in vivo studies of neuronal nicotinic acetylcholine receptors

Life Sciences ◽

10.1016/s0024-3205(98)00240-9 ◽

1998 ◽

Vol 63 (1) ◽

pp. PL13-PL18 ◽

Cited By ~ 23

Author(s):

Michael Kassiou ◽

Ursula A. Scheffel ◽

Hayden T. Ravert ◽

William B. Mathews ◽

John L. Musachio ◽

...

Keyword(s):

Acetylcholine Receptors ◽

In Vivo Studies ◽

Nicotinic Acetylcholine ◽

Pharmacological Evaluation

In Vivo Imaging of Nicotinic Acetylcholine Receptors in the Central Nervous System

Nicotinic Acetylcholine Receptor Signaling in Neuroprotection ◽

10.1007/978-981-10-8488-1_2 ◽

2018 ◽

pp. 17-44

Author(s):

Masashi Ueda ◽

Yuki Matsuura ◽

Ryosuke Hosoda ◽

Hideo Saji

Keyword(s):

Central Nervous System ◽

Nervous System ◽

In Vivo Imaging ◽

Acetylcholine Receptors ◽

Nicotinic Acetylcholine ◽

The Central Nervous System

6-[18F]fluoro-A-85380, a novel radioligand for in vivo imaging of central nicotinic acetylcholine receptors

Life Sciences ◽

10.1016/s0024-3205(00)00635-4 ◽

2000 ◽

Vol 67 (4) ◽

pp. 463-469 ◽

Cited By ~ 35

Author(s):

Andrew G. Horti ◽

Svetlana I. Chefer ◽

Alexey G. Mukhin ◽

Andrei O. Koren ◽

Daniela Gündisch ◽

...

Keyword(s):

In Vivo Imaging ◽

Acetylcholine Receptors ◽