scholarly journals COMBINED METHOD OF OBTAINING PHOSPHORYLATED MONO- AND DIIMIDATES

2021 ◽  
pp. 49-52
Author(s):  
V. E. Shishkin ◽  
E. V. Shishkin ◽  
O. V. Anishchenko ◽  
M. A. Shevchenko ◽  
I. D. Kravchenko
Keyword(s):  
Biological Activity ◽  
Combined Method ◽  
Potential Biological Activity ◽  
Derivatives Of

The interaction of mono- and diimidate hydrochlorides with dialkyl chlorophosphates in the presence of triethylamine without the release of free imidates was studied. A combined method for obtaining N-phosphorylated derivatives of imidic acids with potential biological activity has been developed.

Synthesis and Reactions of Some New Quinoline Thiosemicarbazide Derivatives of Potential Biological Activity

2008 ◽  
Vol 183 (6) ◽  
pp. 1323-1343 ◽  
Author(s):  
E. M. Keshk ◽  
S. I. El-Desoky ◽  
M. A. A. Hammouda ◽  
A. H. Abdel-Rahman ◽  
A. G. Hegazi
Keyword(s):  
Biological Activity ◽  
Potential Biological Activity ◽  
Thiosemicarbazide Derivatives ◽  
Derivatives Of

Lactamomethyl derivatives of diphenols: synthesis, structure, and potential biological activity

2018 ◽  
Vol 67 (8) ◽  
pp. 1518-1529 ◽  
Author(s):  
Vad. V. Negrebetsky ◽  
S. V. Vorobyev ◽  
E. P. Kramarova ◽  
A. G. Shipov ◽  
T. A. Shmigol ◽  
...  
Keyword(s):  
Biological Activity ◽  
Potential Biological Activity ◽  
Derivatives Of

The Synthesis of Some New Quinazolone Derivatives of Potential Biological Activity

2006 ◽  
Vol 181 (8) ◽  
pp. 1895-1912 ◽  
Author(s):  
A. A. El-Barbary ◽  
A. Z. Abou El-Ezz ◽  
A. M. Sharaf ◽  
C. Nielsen
Keyword(s):  
Biological Activity ◽  
Potential Biological Activity ◽  
Derivatives Of

scholarly journals Synthesis and characterization of 2-arylidene derivatives of thiazolopyrimidines with potential biological activity

2016 ◽  
Author(s):  
M. Matilde Marques ◽  
Mohamed Mahgoub ◽  
Awatef Elmaghraby ◽  
Abd-Elfttah Harb ◽  
Filipa Galego ◽  
...  
Keyword(s):  
Biological Activity ◽  
Synthesis And Characterization ◽  
Potential Biological Activity ◽  
Derivatives Of

scholarly journals New pyrazole derivatives of potential biological activity

ARKIVOC ◽  
2012 ◽  
Vol 2012 (7) ◽  
pp. 228-241 ◽  
Author(s):  
Abdel-Rahman Farghaly ◽  
Sabah Esmail ◽  
Ali Abdel-Hafez ◽  
Patrice Vanelle ◽  
Hussein El-Kashef
Keyword(s):  
Biological Activity ◽  
Pyrazole Derivatives ◽  
Potential Biological Activity ◽  
Derivatives Of

Synthesis and structure investigation of novel pyrimidine-2,4,6-trione derivatives of highly potential biological activity as anti-diabetic agent

2015 ◽  
Vol 1098 ◽  
pp. 365-376 ◽  
Author(s):  
Assem Barakat ◽  
Saied M. Soliman ◽  
Abdullah Mohammed Al-Majid ◽  
Gehad Lotfy ◽  
Hazem A. Ghabbour ◽  
...  
Keyword(s):  
Biological Activity ◽  
Structure Investigation ◽  
Potential Biological Activity ◽  
Derivatives Of

scholarly journals Derivatives of 1,2,4-Triazole-3,4-Disubstituted Based on Aminoacids with Potential Biological Activity

2020 ◽  
Vol 71 (5) ◽  
pp. 211-221
Author(s):  
Corina Cheptea ◽  
Valeriu Sunel ◽  
Cezarina Morosanu ◽  
Dana Ortansa Dorohoi
Keyword(s):  
Biological Activity ◽  
Chemical Structure ◽  
Malignant Tumors ◽  
Potential Biological Activity ◽  
New Compounds ◽  
Derivatives Of

In order to obtain new substances with potential biological activity dipeptide derivatives from p-aminobenzoyl-phenylglycine and p-aminobenzoyl-phenylalanine were grafted on 1,2,4-triazolic heterocycle. The new synthesized compounds belong to the group of antimetabolites, group used in medicine for treating malignant tumors. Also, it is possible to study the correlation between chemical structure and biological activity of the new compounds.

scholarly journals A New Type of Synthesis of 1,2,3-Thiadiazole and 1,2,3-Diazaphosphole Derivatives Via-Hurd-Mori Cyclization

2012 ◽  
Vol 9 (3) ◽  
pp. 1276-1287 ◽  
Author(s):  
Mona A. Hosny ◽  
Taghreed H. El-Sayed ◽  
Emtithal El-Sawi
Keyword(s):  
Biological Activity ◽  
Large Scale ◽  
High Potential ◽  
Efficient Synthesis ◽  
Anticancer Effect ◽  
Potential Biological Activity ◽  
Large Scale Preparation ◽  
New Type ◽  
Scale Preparation ◽  
Derivatives Of

We present a short and efficient synthesis of the title compounds starting with cheap and readily available camphor and derivatives of acetophenone. The optimized sequence allows the large-scale preparation of this new type of synthesis in a few steps. New 1,2,3-thiadiazole and 1,2,3-diazaphosphole derivatives 11-20, were prepared from the ketones 1-5 via the corresponding semicarbazones 6-10. The Hurd-Mori and Lalezari methods were used, respectively, for the preparation of these 1,2,3-thiadiazole and 1,2,3-diazaphospholene derivatives. These derivatives exhibit anticancer effect due to their high potential biological activity.

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