Synthesis and Biological Evaluation of Isophthalamide Derivatives as T-type Calcium Channel Blockers

Biological Evaluation ◽

Channel Blockers ◽

Synthesis and biological evaluation of novel N3- substituted dihydropyrimidine derivatives as T-type calcium channel blockers and their efficacy as analgesics in mouse models of inflammatory pain

Bioorganic & Medicinal Chemistry ◽

10.1016/j.bmc.2017.02.015 ◽

2017 ◽

Vol 25 (6) ◽

pp. 1926-1938 ◽

Cited By ~ 16

Author(s):

Mohamed Teleb ◽

Fang-Xiong Zhang ◽

Junting Huang ◽

Vinicius M. Gadotti ◽

Ahmed M. Farghaly ◽

...

Keyword(s):

Calcium Channel ◽

Mouse Models ◽

Inflammatory Pain ◽

Biological Evaluation ◽

Channel Blockers ◽

ChemInform Abstract: Facile Synthesis and Biological Evaluation of 3,3-Diphenylpropanoyl Piperazines as T-Type Calcium Channel Blockers.

ChemInform ◽

10.1002/chin.201120168 ◽

2011 ◽

Vol 42 (20) ◽

pp. no-no

Author(s):

Yeon-hee Choi ◽

Du Jong Baek ◽

Seon Hee Seo ◽

Jae Kyun Lee ◽

Ae Nim Pae ◽

...

Keyword(s):

Calcium Channel ◽

Biological Evaluation ◽

Channel Blockers ◽

Facile Synthesis ◽

Synthesis and biological evaluation of substituted 4-(OBz)phenylalanine derivatives as novel N-type calcium channel blockers

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(99)00160-2 ◽

1999 ◽

Vol 9 (8) ◽

pp. 1121-1126 ◽

Cited By ~ 21

Author(s):

Lain-Yen Hu ◽

Todd R. Ryder ◽

Sham S. Nikam ◽

Elizabeth Millerman ◽

Balazs G. Szoke ◽

...

Keyword(s):

Calcium Channel ◽

Biological Evaluation ◽

Channel Blockers ◽

ChemInform Abstract: Synthesis and Biological Evaluation of Substituted 4-(OBz)Phenylalanine Derivatives as Novel N-Type Calcium Channel Blockers.

ChemInform ◽

10.1002/chin.199933216 ◽

2010 ◽

Vol 30 (33) ◽

pp. no-no

Author(s):

Lain-Yen Hu ◽

Todd R. Ryder ◽

Sham S. Nikam ◽

Elizabeth Millerman ◽

Balazs G. Szoke ◽

...

Keyword(s):

Calcium Channel ◽

Biological Evaluation ◽

Channel Blockers ◽

Synthesis and Biological Evaluation of Pentacycloundecylamines and Triquinylamines as Voltage-Gated Calcium Channel Blockers

Archiv der Pharmazie ◽

10.1002/ardp.201500293 ◽

2016 ◽

Vol 349 (4) ◽

pp. 252-267 ◽

Cited By ~ 7

Author(s):

Lois-May Young ◽

Werner J. Geldenhuys ◽

Olwen C. Domingo ◽

Sarel F. Malan ◽

Cornelis J. Van der Schyf

Keyword(s):

Calcium Channel ◽

Biological Evaluation ◽

Channel Blockers ◽

Voltage Gated ◽

Voltage Gated Calcium Channel ◽

Synthesis and Biological Evaluation of 1-Heteroarylmethyl 1,4-Diazepanes Derivatives as Potential T-type Calcium Channel Blockers

Bulletin of the Korean Chemical Society ◽

10.5012/bkcs.2011.32.8.3063 ◽

2011 ◽

Vol 32 (spc8) ◽

pp. 3063-3073 ◽

Cited By ~ 5

Author(s):

Punna Reddy Ullapu ◽

Su-Jin Ku ◽

Yeon-Hee Choi ◽

Ji-Yeon Park ◽

So-Yeop Han ◽

...

Keyword(s):

Calcium Channel ◽

Biological Evaluation ◽

Channel Blockers ◽

Synthesis and biological evaluation of 1-(isoxazol-5-ylmethylaminoethyl)-4-phenyl tetrahydropyridine and piperidine derivatives as potent T-type calcium channel blockers with antinociceptive effect in a neuropathic pain model

European Journal of Medicinal Chemistry ◽

10.1016/j.ejmech.2013.12.056 ◽

2014 ◽

Vol 74 ◽

pp. 246-257 ◽

Cited By ~ 12

Author(s):

Ju-Hyeon Lee ◽

Seon Hee Seo ◽

Eun Jeong Lim ◽

Nam-Chul Cho ◽

Ghilsoo Nam ◽

...

Keyword(s):

Neuropathic Pain ◽

Calcium Channel ◽

Antinociceptive Effect ◽

Biological Evaluation ◽

Channel Blockers ◽

Pain Model ◽

Neuropathic Pain Model ◽

Synthesis and biological evaluation of 4-piperidinecarboxylate and 4-piperidinecyanide derivatives for T-type calcium channel blockers

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2011.07.087 ◽

2011 ◽

Vol 21 (19) ◽

pp. 5910-5915 ◽

Cited By ~ 8

Author(s):

Hyun Min Woo ◽

Yun Suk Lee ◽

Eun Joo Roh ◽

Seon Hee Seo ◽

Chi Man Song ◽

...

Keyword(s):

Calcium Channel ◽

Biological Evaluation ◽

Channel Blockers ◽

Synthesis and biological evaluation of 1,4-diazepane derivatives as T-type calcium channel blockers

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/j.bmcl.2010.03.084 ◽

2010 ◽

Vol 20 (9) ◽

pp. 2705-2708 ◽

Cited By ~ 18

Author(s):

Su Jin Gu ◽

Jae Kyun Lee ◽

Ae Nim Pae ◽

Hye Jin Chung ◽

Hyewon Rhim ◽

...

Keyword(s):

Calcium Channel ◽

Biological Evaluation ◽

Channel Blockers ◽

Synthesis and Biological Evaluation of Falcarinol-Type Analogues as Potential Calcium Channel Blockers

Journal of Natural Products ◽

10.1021/acs.jnatprod.1c00136 ◽

2021 ◽

Author(s):

Yang Li ◽

Wan-Li Tan ◽

Kai Guo ◽

Xiao-Wei Gao ◽

Jun Wei ◽

...

Keyword(s):

Calcium Channel ◽

Biological Evaluation ◽

Channel Blockers ◽