In vitro and in vivo pharmacokinetic characteristics of clazosentan, an intravenous endothelin receptor antagonist, in humans

In vivo and in vitro disposition profile of tezosentan, an intravenous dual endothelin receptor antagonist, in humans

Xenobiotica ◽

10.1080/0049825021000061624 ◽

2003 ◽

Vol 33 (4) ◽

pp. 399-414 ◽

Cited By ~ 8

Author(s):

A. Treiber ◽

P. L. M. Van Giersbergen ◽

J. Dingemanse

Keyword(s):

Receptor Antagonist ◽

The endothelin system in Morris hepatoma-7777: an endothelin receptor antagonist inhibits growth in vitro and in vivo

British Journal of Pharmacology ◽

10.1038/sj.bjp.0705601 ◽

2004 ◽

Vol 141 (2) ◽

pp. 215-222 ◽

Cited By ~ 7

Author(s):

Thiemo Pfab ◽

Gisela Stoltenburg-Didinger ◽

Christoph Trautner ◽

Michael Godes ◽

Christian Bauer ◽

...

Keyword(s):

Receptor Antagonist ◽

Endothelin Receptor ◽

Endothelin System ◽

Morris Hepatoma

Bosentan, a new endothelin receptor antagonist: prediction of the systemic plasma clearance in man from combined in vivo and in vitro data

Xenobiotica ◽

10.3109/00498259509061925 ◽

1995 ◽

Vol 25 (12) ◽

pp. 1381-1390 ◽

Cited By ~ 36

Author(s):

G. Ubeaud ◽

C. Schmitt ◽

D. Jaeck ◽

T. Lave ◽

Ph. Coassolo

Keyword(s):

Receptor Antagonist ◽

Plasma Clearance ◽

Endothelin Receptor ◽

Vitro Data ◽

In Vitro Data

In vivo and in vitro studies exploring the pharmacokinetic interaction between bosentan, a dual endothelin receptor antagonist, and glyburide

Clinical Pharmacology & Therapeutics ◽

10.1067/mcp.2002.122473 ◽

2002 ◽

Vol 71 (4) ◽

pp. 253-262 ◽

Cited By ~ 41

Author(s):

P VANGIERSBERGEN ◽

A TREIBER ◽

M CLOZEL ◽

F BODIN ◽

J DINGEMANSE

Keyword(s):

Receptor Antagonist ◽

Pharmacokinetic Interaction ◽

In Vitro Studies ◽

Cpu0507, An Endothelin Receptor Antagonist, Improves Rat Hypoxic Pulmonary Artery Hypertension And Constriction In Vivo And In Vitro

Clinical and Experimental Pharmacology and Physiology ◽

10.1111/j.1440-1681.2006.04488.x ◽

2006 ◽

Vol 33 (11) ◽

pp. 1066-1072 ◽

Cited By ~ 8

Author(s):

Sheng-hua Yuan ◽

De-zai Dai ◽

Li Guan ◽

Yin Dai ◽

Min Ji

Keyword(s):

Pulmonary Artery ◽

Receptor Antagonist ◽

Pulmonary Artery Hypertension ◽

Coronary vasoconstriction in vitro in the hearts of polyarthritic rats: effectiveness of in vivo treatment with the endothelin receptor antagonist SB 209670

British Journal of Pharmacology ◽

10.1111/j.1476-5381.1995.tb13351.x ◽

1995 ◽

Vol 114 (7) ◽

pp. 1327-1328 ◽

Cited By ~ 3

Author(s):

Timothy D. Warner ◽

Dean Willis ◽

Adrian R. Moore ◽

John R. Vane ◽

Peter Klemm

Keyword(s):

Receptor Antagonist ◽

Endothelin Receptor ◽

Coronary Vasoconstriction ◽

In Vivo Treatment

In vivo subcellular elemental dynamics in liver graft: With special reference to effect of non-selective endothelin receptor antagonist, TAK-044, on the graft injury

Hepatology Research ◽

10.1016/s1386-6346(99)00099-6 ◽

2000 ◽

Vol 18 (3) ◽

pp. 171-183

Author(s):

Y Takaya

Keyword(s):

Special Reference ◽

Receptor Antagonist ◽

Liver Graft ◽

Application of Serial In Vivo Magnetic Resonance Imaging to Evaluate the Efficacy of Endothelin Receptor Antagonist SB 217242 in the Rat Carotid Artery Model of Neointima Formation

Circulation ◽

10.1161/01.cir.97.22.2252 ◽

1998 ◽

Vol 97 (22) ◽

pp. 2252-2258 ◽

Cited By ~ 5

Author(s):

Sudeep Chandra ◽

Lynne V. Clark ◽

Robert W. Coatney ◽

Le Phan ◽

Susanta K. Sarkar ◽

...

Keyword(s):

Magnetic Resonance Imaging ◽

Magnetic Resonance ◽

Carotid Artery ◽

Receptor Antagonist ◽

Neointima Formation ◽

Endothelin Receptor ◽

Resonance Imaging

Pharmacological Profile in vitro of A New Endothelin Receptor Antagonist, TAK-044.

The Japanese Journal of Pharmacology ◽

10.1016/s0021-5198(19)50309-2 ◽

1994 ◽

Vol 64 ◽

pp. 167

Author(s):

Yumiko Awane ◽

Keiji Kusumoto ◽

Kazuki Kubo ◽

Akira Kawata ◽

Takashi Kikuchi ◽

...

Keyword(s):

Receptor Antagonist ◽

Endothelin Receptor ◽

Pharmacological Profile

In Vivo Pharmacology of Ro 46-2005, The First Synthetic Nonpeptide Endothelin Receptor Antagonist: Implications for Endothelin Physiology

Journal of Cardiovascular Pharmacology ◽

10.1097/00005344-199322008-00099 ◽

1993 ◽

Vol 22 (Supplement 8) ◽

pp. S377-S379 ◽

Cited By ~ 34

Author(s):

Martine Clozel ◽

Volker Breu ◽

Gillian A. Gray ◽

Bernd-Michael Löffler

Keyword(s):

Receptor Antagonist ◽