cyclic lactam Recently Published Documents

Solid-phase peptide head-to-side chain cyclodimerization: Discovery of C2-symmetric cyclic lactam hybrid α-melanocyte-stimulating hormone (MSH)/agouti-signaling protein (ASIP) analogues with potent activities at the human melanocortin receptors

Peptides ◽

10.1016/j.peptides.2010.06.026 ◽

2010 ◽

Vol 31 (10) ◽

pp. 1894-1905 ◽

Cited By ~ 7

Author(s):

Alexander V. Mayorov ◽

Minying Cai ◽

Erin S. Palmer ◽

Zhihua Liu ◽

James P. Cain ◽

...

Keyword(s):

Solid Phase ◽

Side Chain ◽

Melanocortin Receptors ◽

Signaling Protein ◽

Cyclic Lactam ◽

ChemInform Abstract: Synthesis of Cyclic Lactam Containing Ecdysteroid Analogues.

ChemInform ◽

10.1002/chin.199131271 ◽

2010 ◽

Vol 22 (31) ◽

pp. no-no

Author(s):

N. V. KOVGANKO ◽

T. N. NETESOVA

Keyword(s):

Solid Phase Synthesis and Circular Dichroism Analysis of (i → i + 4) Cyclic Lactam Analogues of Kisspeptin

International Journal of Peptide Research and Therapeutics ◽

10.1007/s10989-008-9140-5 ◽

2008 ◽

Vol 14 (4) ◽

pp. 323-331 ◽

Cited By ~ 2

Author(s):

Michelle A. Camerino ◽

David C. M. Kong ◽

David K. Chalmers ◽

Philip E. Thompson

Keyword(s):

Circular Dichroism ◽

Solid Phase Synthesis ◽

Solid Phase ◽

Phase Synthesis ◽

Circular Dichroism Analysis ◽

Circular Dichroïsm ◽

Structure–Activity Relationships of Cyclic Lactam Analogues of α-Melanocyte-Stimulating Hormone (α-MSH) Targeting the Human Melanocortin-3 Receptor

Journal of Medicinal Chemistry ◽

10.1021/jm070461w ◽

2008 ◽

Vol 51 (2) ◽

pp. 187-195 ◽

Cited By ~ 8

Author(s):

Alexander V. Mayorov ◽

Minying Cai ◽

Erin S. Palmer ◽

Matthew M. Dedek ◽

James P. Cain ◽

...

Keyword(s):

Structure Activity Relationships ◽

Structure Activity ◽

Cyclic Lactam ◽

Effects of Macrocycle Size and Rigidity on Melanocortin Receptor-1 and -5 Selectivity in Cyclic Lactam alpha-Melanocyte-Stimulating Hormone Analogs

Chemical Biology & Drug Design ◽

10.1111/j.1747-0285.2006.00383.x ◽

2006 ◽

Vol 67 (5) ◽

pp. 329-335 ◽

Cited By ~ 13

Author(s):

Alexander V. Mayorov ◽

So-Yeop Han ◽

Minying Cai ◽

Matthew R. Hammer ◽

Dev Trivedi ◽

...

Keyword(s):

Melanocortin Receptor ◽

Hormone Analogs ◽

Cyclic Lactam ◽

The Glycine1Residue in Cyclic Lactam Analogues of Galanin(1−16)-NH2Is Important for Stabilizing an N-Terminal Helix

Biochemistry ◽

10.1021/bi991081i ◽

1999 ◽

Vol 38 (46) ◽

pp. 15295-15304 ◽

Cited By ~ 23

Author(s):

Katharine A. Carpenter ◽

Ralf Schmidt ◽

Shi Yi Yue ◽

Lejla Hodzic ◽

Chantevy Pou ◽

...

Keyword(s):

Synthesis and biological activities of cyclic lactam peptides as substrates for non-receptors PTKs

Letters in Peptide Science ◽

10.1007/bf02443625 ◽

1999 ◽

Vol 6 (2-3) ◽

pp. 117-121

Author(s):

Paolo Ruzza ◽

Arianna Donella-Deana ◽

Andrea Calderan ◽

Barbara Biondi ◽

Lorenzo A. Pinna ◽

...

Keyword(s):

Biological Activities ◽

Design, Synthesis, and Biological Activities of Cyclic Lactam Peptide Analogues of Dynorphin A(1−11)-NH21

Journal of Medicinal Chemistry ◽

10.1021/jm950369c ◽

1996 ◽

Vol 39 (5) ◽

pp. 1136-1141 ◽

Cited By ~ 17

Author(s):

Feng-Di T. Lung ◽

Nathan Collins ◽

Dagmar Stropova ◽

Peg Davis ◽

Henry I. Yamamura ◽

...

Keyword(s):

Biological Activities ◽

Dynorphin A ◽

Design Synthesis ◽

Peptide Analogues ◽

Cyclic lactam .alpha.-melanotropin analogs of Ac-Nle4-cyclo[Asp5,D-Phe7,Lys10]-.alpha.-melanocyte-stimulating hormone-(4-10)-NH2 with bulky aromatic amino acids at position 7 show high antagonist potency and selectivity at specific melanocortin receptors

Journal of Medicinal Chemistry ◽

10.1021/jm00018a005 ◽

1995 ◽

Vol 38 (18) ◽

pp. 3454-3461 ◽

Cited By ~ 256

Author(s):

Victor J. Hrubu ◽

Dongsi Lu ◽

Shubh D. Sharma ◽

Ana de L. Castrucci ◽

Robert A. Kesterson ◽

...

Keyword(s):

Amino Acids ◽

Aromatic Amino Acids ◽

Melanocortin Receptors ◽

Cyclic Lactam ◽