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Age and circadian rhythm‐dependent effects of M 1 muscarinic acetylcholine receptor positive allosteric modulators and donepezil on sleep‐wake architecture and arousal
Alzheimer s & Dementia
◽
10.1002/alz.057851
◽
2021
◽
Vol 17
(S9)
◽
Author(s):
Jason K Russell
◽
Michael Bubser
◽
Paul A Newhouse
◽
Craig W Lindsley
◽
Carrie K Jones
Keyword(s):
Circadian Rhythm
◽
Acetylcholine Receptor
◽
Muscarinic Acetylcholine Receptor
◽
Allosteric Modulators
◽
Muscarinic Acetylcholine
◽
Positive Allosteric Modulators
Download Full-text
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P2-068: CIRCADIAN RHYTHM-DEPENDENT EFFECTS OF M1 MUSCARINIC ACETYLCHOLINE RECEPTOR POSITIVE ALLOSTERIC MODULATORS ON AROUSAL AND COGNITION
Alzheimer s & Dementia
◽
10.1016/j.jalz.2019.06.2475
◽
2019
◽
Vol 15
◽
pp. P596-P597
Author(s):
Jason K. Russell
◽
Robert W. Gould
◽
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Richard J. Fu
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Circadian Rhythm
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Acetylcholine Receptor
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Muscarinic Acetylcholine Receptor
◽
Allosteric Modulators
◽
Muscarinic Acetylcholine
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Positive Allosteric Modulators
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M1 Muscarinic Acetylcholine Receptor
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M1 Muscarinic
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Surface modified nano-lipid drug conjugates of positive allosteric modulators of M1 muscarinic acetylcholine receptor for the treatment of Alzheimer’s disease
Medical Hypotheses
◽
10.1016/j.mehy.2017.01.026
◽
2017
◽
Vol 101
◽
pp. 17-22
◽
Cited By ~ 3
Author(s):
Pavan Kumar Chintamaneni
◽
Praveen T. Krishnamurthy
◽
Pachava Vengal Rao
◽
SaiKiran S.S. Pindiprolu
Keyword(s):
Alzheimer’S Disease
◽
Acetylcholine Receptor
◽
Muscarinic Acetylcholine Receptor
◽
Allosteric Modulators
◽
Muscarinic Acetylcholine
◽
Drug Conjugates
◽
Positive Allosteric Modulators
◽
M1 Muscarinic Acetylcholine Receptor
◽
M1 Muscarinic
◽
Surface Modified
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Discovery of a Novel Class of Heteroaryl-Pyrrolidinones as Positive Allosteric Modulators of the Muscarinic Acetylcholine Receptor M1
Bioorganic & Medicinal Chemistry Letters
◽
10.1016/j.bmcl.2021.128193
◽
2021
◽
pp. 128193
Author(s):
Paul K. Spearing
◽
Hyekyung P. Cho
◽
Vincent B. Luscombe
◽
Anna L. Blobaum
◽
Olivier Boutaud
◽
...
Keyword(s):
Acetylcholine Receptor
◽
Muscarinic Acetylcholine Receptor
◽
Allosteric Modulators
◽
Muscarinic Acetylcholine
◽
Positive Allosteric Modulators
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Characterization of novel selective positive allosteric modulators (PAMS) of the M4 muscarinic acetylcholine receptor (mAChR)
The FASEB Journal
◽
10.1096/fasebj.22.1_supplement.714.2
◽
2008
◽
Vol 22
(S1)
◽
Author(s):
Ashley Elizabeth Brady
◽
Tom M Bridges
◽
Carrie K Jones
◽
Jana K Shirey
◽
Craig W Lindsley
◽
...
Keyword(s):
Acetylcholine Receptor
◽
Muscarinic Acetylcholine Receptor
◽
Allosteric Modulators
◽
Muscarinic Acetylcholine
◽
Positive Allosteric Modulators
Download Full-text
Faculty Opinions recommendation of Structure-based discovery of selective positive allosteric modulators of antagonists for the M2 muscarinic acetylcholine receptor.
Faculty Opinions – Post-Publication Peer Review of the Biomedical Literature
◽
10.3410/f.732691118.793543578
◽
2018
◽
Author(s):
Robert Copeland
Keyword(s):
Acetylcholine Receptor
◽
Muscarinic Acetylcholine Receptor
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Allosteric Modulators
◽
Muscarinic Acetylcholine
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Positive Allosteric Modulators
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Development of Novel 4‐Arylpyridin‐2‐one and 6‐Arylpyrimidin‐4‐one Positive Allosteric Modulators of the M 1 Muscarinic Acetylcholine Receptor
ChemMedChem
◽
10.1002/cmdc.202000540
◽
2020
◽
Author(s):
Manuela Jörg
◽
Elham Khajehali
◽
Emma T. Westhuizen
◽
K. H. C. Choy
◽
David M. Shackleford
◽
...
Keyword(s):
Acetylcholine Receptor
◽
Muscarinic Acetylcholine Receptor
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Allosteric Modulators
◽
Muscarinic Acetylcholine
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Positive Allosteric Modulators
Download Full-text
Structure–Activity Relationships of Pan-Gαq/11 Coupled Muscarinic Acetylcholine Receptor Positive Allosteric Modulators
ACS Chemical Neuroscience
◽
10.1021/acschemneuro.8b00136
◽
2018
◽
Vol 9
(7)
◽
pp. 1818-1828
◽
Cited By ~ 3
Author(s):
Alice E. Berizzi
◽
Aaron M. Bender
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Craig W. Lindsley
◽
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◽
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◽
...
Keyword(s):
Acetylcholine Receptor
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Muscarinic Acetylcholine Receptor
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Allosteric Modulators
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Muscarinic Acetylcholine
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Structure Activity Relationships
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Structure Activity
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Probing the binding site of novel selective positive allosteric modulators at the M1 muscarinic acetylcholine receptor
Biochemical Pharmacology
◽
10.1016/j.bcp.2018.05.009
◽
2018
◽
Vol 154
◽
pp. 243-254
◽
Cited By ~ 8
Author(s):
Elham Khajehali
◽
Celine Valant
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Manuela Jörg
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Andrew B. Tobin
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P. Jeffrey Conn
◽
...
Keyword(s):
Binding Site
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Acetylcholine Receptor
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Muscarinic Acetylcholine Receptor
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Allosteric Modulators
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Muscarinic Acetylcholine
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Positive Allosteric Modulators
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M1 Muscarinic Acetylcholine Receptor
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M1 Muscarinic
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Effects of M1 and M4 muscarinic acetylcholine receptor positive allosteric modulators on sleep and cognition in rodents
The FASEB Journal
◽
10.1096/fasebj.27.1_supplement.661.8
◽
2013
◽
Vol 27
(S1)
◽
Author(s):
Robert W Gould
◽
Michael T Nedelcovych
◽
Michael D Grannan
◽
Michael Bubser
◽
Michael R Wood
◽
...
Keyword(s):
Acetylcholine Receptor
◽
Muscarinic Acetylcholine Receptor
◽
Allosteric Modulators
◽
Muscarinic Acetylcholine
◽
Positive Allosteric Modulators
◽
Sleep And Cognition
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Discovery and structure-activity relationships study of positive allosteric modulators of the M3 muscarinic acetylcholine receptor
Bioorganic & Medicinal Chemistry
◽
10.1016/j.bmc.2020.115531
◽
2020
◽
Vol 28
(13)
◽
pp. 115531
Author(s):
Hiroaki Tanaka
◽
Kenji Negoro
◽
Takanori Koike
◽
Issei Tsukamoto
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Acetylcholine Receptor
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Muscarinic Acetylcholine Receptor
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Allosteric Modulators
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Muscarinic Acetylcholine
◽
Structure Activity Relationships
◽
M3 Muscarinic Acetylcholine Receptor
◽
Structure Activity
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Positive Allosteric Modulators
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