Asymmetric Synthesis of Dihydropyranones from Ynones by Sequential Copper(I)-Catalyzed Direct Aldol and Silver(I)-Catalyzed Oxy-Michael Reactions

2012 ◽  
Vol 124 (16) ◽  
pp. 3998-4001 ◽  
Author(s):  
Shi-Liang Shi ◽  
Motomu Kanai ◽  
Masakatsu Shibasaki
Keyword(s):  
Asymmetric Synthesis ◽  
Michael Reactions

Chiral Phase-Transfer-Catalyzed Intramolecular aza-Michael Reactions for the Asymmetric Synthesis of Isoindolinones

2015 ◽  
Vol 2015 (9) ◽  
pp. 1995-2004 ◽  
Author(s):  
Stéphane Lebrun ◽  
Romain Sallio ◽  
Mélanie Dubois ◽  
Francine Agbossou-Niedercorn ◽  
Eric Deniau ◽  
...  
Keyword(s):  
Asymmetric Synthesis ◽  
Phase Transfer ◽  
Chiral Phase ◽  
Michael Reactions

ChemInform Abstract: Chiral Phase-Transfer-Catalyzed Intramolecular Aza-Michael Reactions for the Asymmetric Synthesis of Isoindolinones.

ChemInform ◽  
2015 ◽  
Vol 46 (30) ◽  
pp. no-no
Author(s):  
Stephane Lebrun ◽  
Romain Sallio ◽  
Melanie Dubois ◽  
Francine Agbossou-Niedercorn ◽  
Eric Deniau ◽  
...  
Keyword(s):  
Asymmetric Synthesis ◽  
Phase Transfer ◽  
Chiral Phase ◽  
Michael Reactions

Recent advances in the asymmetric synthesis of pharmacology-relevant nitrogen heterocycles via stereoselective aza-Michael reactions

2019 ◽  
Vol 17 (15) ◽  
pp. 3670-3708 ◽  
Author(s):  
Maxim G. Vinogradov ◽  
Olga V. Turova ◽  
Sergei G. Zlotin
Keyword(s):  
Asymmetric Synthesis ◽  
Michael Reaction ◽  
Nitrogen Heterocycles ◽  
Michael Reactions ◽  
Naturally Occurring ◽  
Recent Advances

In this review, recent applications of a stereoselective aza-Michael reaction for asymmetric synthesis of naturally occurring N-containing heterocyclic scaffolds and their usefulness to pharmacology are summarized.

C 2-Symmetric pyrrolidine-derived squaramides as recyclable organocatalysts for asymmetric Michael reactions

2016 ◽  
Vol 14 (41) ◽  
pp. 9751-9759 ◽  
Author(s):  
A. S. Kucherenko ◽  
V. G. Lisnyak ◽  
A. A. Kostenko ◽  
S. V. Kochetkov ◽  
S. G. Zlotin
Keyword(s):  
Asymmetric Synthesis ◽  
Active Pharmaceutical Ingredients ◽  
Pharmaceutical Ingredients ◽  
Michael Reactions

Novel sustainable organocatalysts applicable to asymmetric synthesis of active pharmaceutical ingredients are developed.

Asymmetric synthesis of highly functionalized furanones via direct Michael reactions mediated by a bulky primary amine

2019 ◽  
Vol 6 (8) ◽  
pp. 1080-1083 ◽  
Author(s):  
Huicai Huang ◽  
Xue Lu ◽  
Yukang Mao ◽  
Jinxing Ye
Keyword(s):  
Asymmetric Synthesis ◽  
Primary Amine ◽  
Michael Reaction ◽  
Michael Reactions

A bulky chiral primary amine catalyzed Michael reaction of 3(2H)-furanones has been realized, leading to the construction of substituted furanone derivatives.

Sign in / Sign up

Export Citation Format

Share Document