Design, synthesis, in silico ADMET, docking, and antiproliferative evaluations of [1,2,4]triazolo[4,3‐ c ]quinazolines as classical DNA intercalators

2022 ◽  
Author(s):  
Mohamed S. Alesawy ◽  
Mohamed‐Kamal Ibrahim ◽  
Ibrahim H. Eissa ◽  
Khaled El‐Adl
2021 ◽  
Author(s):  
Khaled El-Adl ◽  
Abdel-Ghany A. El-Helby ◽  
Helmy Sakr ◽  
Alaa Elwan

In view of their DNA intercalation activities as anticancer agents, 17 novel [1,2,4]triazolo[4,3-a]quinoxaline derivatives have been designed, synthesized and evaluated against HepG2, HCT-116 and MCF-7 cells.


2021 ◽  
Vol 108 ◽  
pp. 104669
Author(s):  
Asmaa M Sayed ◽  
Fatma A. Taher ◽  
Mohammad R.K. Abdel-Samad ◽  
Mohamed S.A. El-Gaby ◽  
Khaled El‐Adl ◽  
...  

2019 ◽  
Vol 352 (5) ◽  
pp. 1800387 ◽  
Author(s):  
Abdel‐Ghany A. El‐Helby ◽  
Rezk R. A. Ayyad ◽  
Mohamed F. Zayed ◽  
Hamada S. Abulkhair ◽  
Hazem Elkady ◽  
...  

2018 ◽  
Vol 264 ◽  
pp. 367-374 ◽  
Author(s):  
Nadjet Rezki ◽  
Salsabeel A. Al-Sodies ◽  
Mouslim Messali ◽  
Sanaa K. Bardaweel ◽  
Pramod K. Sahu ◽  
...  

2021 ◽  
Author(s):  
Fathalla Khedr ◽  
Mohamed‐Kamal Ibrahim ◽  
Ibrahim H. Eissa ◽  
Hamada S. Abulkhair ◽  
Khaled El‐Adl

2020 ◽  
Vol 1222 ◽  
pp. 128881 ◽  
Author(s):  
Mayuri A. Borad ◽  
Divya J. Jethava ◽  
Manoj N. Bhoi ◽  
Chirag N. Patel ◽  
Himanshu A. Pandya ◽  
...  

2021 ◽  
Author(s):  
Nashwa M. Saleh ◽  
Adel A.‐H. Abdel‐Rahman ◽  
Asmaa M. Omar ◽  
Mohamed M. Khalifa ◽  
Khaled El‐Adl

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