Binding characterization of
            N
            ‐(2‐chloro‐5‐thiomethylphenyl)‐
            N
            ′‐(3‐[
            3
            H]
            3
            methoxy phenyl)‐
            N
            ′‐methylguanidine ([
            3
            H]
            GMOM
            ), a non‐competitive
            N
            ‐methyl‐D‐aspartate (
            NMDA
            ) receptor antagonist

Athanasios Metaxas; Bart N. M. van Berckel; Pieter J. Klein; Joost Verbeek; Emily C. Nash; Esther J. M. Kooijman; Véronique A. Renjaän; Sandeep S. V. Golla; Ronald Boellaard; Johannes A. M. Christiaans; Albert D. Windhorst; Josée E. Leysen

doi:10.1002/prp2.458

Binding characterization of N ‐(2‐chloro‐5‐thiomethylphenyl)‐ N ′‐(3‐[ 3 H] 3 methoxy phenyl)‐ N ′‐methylguanidine ([ 3 H] GMOM ), a non‐competitive N ‐methyl‐D‐aspartate ( NMDA ) receptor antagonist

Pharmacology Research & Perspectives ◽

10.1002/prp2.458 ◽

2019 ◽

Vol 7 (1) ◽

pp. e00458 ◽

Cited By ~ 1

Author(s):

Athanasios Metaxas ◽

Bart N. M. van Berckel ◽

Pieter J. Klein ◽

Joost Verbeek ◽

Emily C. Nash ◽

...

Keyword(s):

Nmda Receptor ◽

Receptor Antagonist ◽

Nmda Receptor Antagonist

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Quantitative physiological characterization of a quinoxalinedione non- NMDA receptor antagonist

Journal of Neuroscience ◽

10.1523/jneurosci.09-09-03230.1989 ◽

1989 ◽

Vol 9 (9) ◽

pp. 3230-3236 ◽

Cited By ~ 60

Author(s):

KA Yamada ◽

JM Dubinsky ◽

SM Rothman

Keyword(s):

Nmda Receptor ◽

Receptor Antagonist ◽

Nmda Receptor Antagonist ◽

Physiological Characterization

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Crystal Structure and Pharmacological Characterization of a NovelN-Methyl-d-aspartate (NMDA) Receptor Antagonist at the GluN1 Glycine Binding Site

Journal of Biological Chemistry ◽

10.1074/jbc.m113.480210 ◽

2013 ◽

Vol 288 (46) ◽

pp. 33124-33135 ◽

Cited By ~ 14

Author(s):

Trine Kvist ◽

Thomas Bielefeldt Steffensen ◽

Jeremy R. Greenwood ◽

Fatemeh Mehrzad Tabrizi ◽

Kasper B. Hansen ◽

...

Keyword(s):

Crystal Structure ◽

Nmda Receptor ◽

Receptor Antagonist ◽

Binding Site ◽

Nmda Receptor Antagonist ◽

Pharmacological Characterization

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Characterization of 3-carboxy-5-phosphono-1,2,3,4-tetrahydroisoquinoline (SC-48981), a potent competitive (NMDA) receptor antagonist, in vitro and in vivo

Neuroscience Letters ◽

10.1016/0304-3940(92)90424-6 ◽

1992 ◽

Vol 135 (2) ◽

pp. 149-152 ◽

Cited By ~ 3

Author(s):

Michael L. Vazquez ◽

Danny J. Garland ◽

Eric T. Sun ◽

Julie A. Cler ◽

Steve J. Mick ◽

...

Keyword(s):

Nmda Receptor ◽

Receptor Antagonist ◽

Nmda Receptor Antagonist

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Isolation and characterization of histogranin, a natural peptide with NMDA receptor antagonist activity

European Journal of Pharmacology Molecular Pharmacology ◽

10.1016/0922-4106(93)90104-h ◽

1993 ◽

Vol 245 (3) ◽

pp. 247-256 ◽

Cited By ~ 37

Author(s):

Simon Lemaire ◽

Vijay Kumar Shukla ◽

Cheryl Rogers ◽

Ibrahim H. Ibrahim ◽

Chantal Lapierre ◽

...

Keyword(s):

Nmda Receptor ◽

Receptor Antagonist ◽

Nmda Receptor Antagonist ◽

Antagonist Activity ◽

Isolation And Characterization ◽

Natural Peptide

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Functional in vitro characterization of CR 3394: A novel voltage dependent N-methyl-d-aspartate (NMDA) receptor antagonist

Neuropharmacology ◽

10.1016/j.neuropharm.2005.09.002 ◽

2006 ◽

Vol 50 (3) ◽

pp. 277-285 ◽

Cited By ~ 8

Author(s):

Gabriele Losi ◽

Marco Lanza ◽

Francesco Makovec ◽

Roberto Artusi ◽

Gianfranco Caselli ◽

...

Keyword(s):

Nmda Receptor ◽

Receptor Antagonist ◽

Nmda Receptor Antagonist ◽

In Vitro Characterization ◽

Voltage Dependent

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Electrophysiological characterization of a novel potent and orally active NMDA receptor antagonist: CGP 37849 and its ethylester CGP 39551

European Journal of Pharmacology ◽

10.1016/0014-2999(90)90496-s ◽

1990 ◽

Vol 182 (1) ◽

pp. 91-100 ◽

Cited By ~ 26

Author(s):

Mario F. Pozza ◽

Hans-Rudolf Olpe ◽

Felix Brugger ◽

Graham E. Fagg

Keyword(s):

Nmda Receptor ◽

Receptor Antagonist ◽

Nmda Receptor Antagonist ◽

Cgp 37849 ◽

Cgp 39551 ◽

Electrophysiological Characterization ◽

Orally Active

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Continuous brachial plexus blockade in combination with the NMDA receptor antagonist memantine prevents phantom pain in acute traumatic upper limb amputees

Yearbook of Anesthesiology and Pain Management ◽

10.1016/s1073-5437(08)70995-1 ◽

2008 ◽

Vol 2008 ◽

pp. 265-266

Author(s):

S.E. Abram

Keyword(s):

Nmda Receptor ◽

Brachial Plexus ◽

Receptor Antagonist ◽

Upper Limb ◽

Nmda Receptor Antagonist ◽

Phantom Pain ◽

Brachial Plexus Blockade

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Microinjection of NMDA Receptor Antagonist AP5 to the Telencephalon

PsycEXTRA Dataset ◽

10.1037/e413802005-463 ◽

2001 ◽

Author(s):

Jennifer Bazner ◽

Min Qi ◽

Xiaojuan Xu

Keyword(s):

Nmda Receptor ◽

Receptor Antagonist ◽

Nmda Receptor Antagonist

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Regionally different responses of GABAergic interneuron populations to a NMDA receptor antagonist challenge with MK-801 and an antipsychotic “rescue therapy“ in an animal model of psychosis

Pharmacopsychiatry ◽

10.1055/s-2007-991763 ◽

2007 ◽

Vol 40 (05) ◽

Author(s):

J Genius ◽

I Braun ◽

H Grunze ◽

J Benninghoff ◽

HJ Möller ◽

...

Keyword(s):

Animal Model ◽

Nmda Receptor ◽

Receptor Antagonist ◽

Rescue Therapy ◽

Nmda Receptor Antagonist ◽

Gabaergic Interneuron ◽

Mk 801

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Disturbed alpha and gamma oscillations ex vivo after single application of the NMDA receptor antagonist MK-801

10.26226/morressier.5785edccd462b80296c98efe ◽

2016 ◽

Author(s):

Zoltan Gerevich

Keyword(s):

Nmda Receptor ◽

Receptor Antagonist ◽

Ex Vivo ◽

Gamma Oscillations ◽

Nmda Receptor Antagonist ◽

Single Application ◽

Mk 801

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