Characterization of a non-approved selective androgen receptor modulator drug candidate sold via the Internet and identification ofin vitrogenerated phase-I metabolites for human sports drug testing

2015 ◽  
Vol 29 (11) ◽  
pp. 991-999 ◽  
Author(s):  
Mario Thevis ◽  
Andreas Lagojda ◽  
Dirk Kuehne ◽  
Andreas Thomas ◽  
Josef Dib ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Phase I ◽  
Drug Testing ◽  
Drug Candidate ◽  
The Internet ◽  
Selective Androgen Receptor Modulator ◽  
Receptor Modulator ◽  
Sports Drug Testing

Expanding sports drug testing assays: Mass spectrometric characterization of the selective androgen receptor modulator drug candidates RAD140 and ACP-105

2013 ◽  
Vol 27 (11) ◽  
pp. 1173-1182 ◽  
Author(s):  
Mario Thevis ◽  
Thomas Piper ◽  
Simon Beuck ◽  
Hans Geyer ◽  
Wilhelm Schänzer
Keyword(s):  
Androgen Receptor ◽  
Drug Testing ◽  
Mass Spectrometric ◽  
Selective Androgen Receptor Modulator ◽  
Drug Candidates ◽  
Receptor Modulator ◽  
Sports Drug Testing

Use of an Electrochemically Synthesised Metabolite of a Selective Androgen Receptor Modulator for Mass Spectrometry-Based Sports Drug Testing

2008 ◽  
Vol 14 (3) ◽  
pp. 163-170 ◽  
Author(s):  
Mario Thevis ◽  
Wiebke Lohmann ◽  
Yvonne Schrader ◽  
Maxie Kohler ◽  
Wolfgang Bornatsch ◽  
...  
Keyword(s):  
Mass Spectrometry ◽  
Androgen Receptor ◽  
Drug Testing ◽  
Selective Androgen Receptor Modulator ◽  
Receptor Modulator ◽  
Sports Drug Testing

Identification of Selected in vitro-Generated Phase-I Metabolites of the Steroidal Selective Androgen Receptor Modulator MK-0773 for Doping Control Purposes

2016 ◽  
Vol 22 (2) ◽  
pp. 49-59 ◽  
Author(s):  
Andreas Lagojda ◽  
Dirk Kuehne ◽  
Oliver Krug ◽  
Andreas Thomas ◽  
Tina Wigger ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Phase I ◽  
Doping Control ◽  
Selective Androgen Receptor Modulator ◽  
Receptor Modulator

Pharmacological characterization of an imidazolopyrazole as novel selective androgen receptor modulator

2013 ◽  
Vol 134 ◽  
pp. 51-58 ◽  
Author(s):  
Xuqing Zhang ◽  
George F. Allan ◽  
Pamela Tannenbaum ◽  
Tifanie Sbriscia ◽  
Olivia Linton ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Selective Androgen Receptor Modulator ◽  
Pharmacological Characterization ◽  
Receptor Modulator

Mass spectrometric characterization of the selective androgen receptor modulator (SARM) YK-11 for doping control purposes

2017 ◽  
Vol 31 (14) ◽  
pp. 1175-1183 ◽  
Author(s):  
Mario Thevis ◽  
Thomas Piper ◽  
Josef Dib ◽  
Andreas Lagojda ◽  
Dirk Kühne ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Mass Spectrometric ◽  
Doping Control ◽  
Selective Androgen Receptor Modulator ◽  
Receptor Modulator

scholarly journals Design, Synthesis, and Preclinical Characterization of the Selective Androgen Receptor Modulator (SARM) RAD140

2010 ◽  
Vol 2 (2) ◽  
pp. 124-129 ◽  
Author(s):  
Chris P. Miller ◽  
Maysoun Shomali ◽  
C. Richard Lyttle ◽  
Louis St. L. O’Dea ◽  
Hillary Herendeen ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Selective Androgen Receptor Modulator ◽  
Design Synthesis ◽  
Receptor Modulator

scholarly journals Characterization of GLPG0492, a selective androgen receptor modulator, in a mouse model of hindlimb immobilization

2014 ◽  
Vol 15 (1) ◽  
Author(s):  
Roland Blanqué ◽  
Liên Lepescheux ◽  
Marielle Auberval ◽  
Dominique Minet ◽  
Didier Merciris ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Mouse Model ◽  
Selective Androgen Receptor Modulator ◽  
Receptor Modulator

Mass spectrometric characterization of urinary metabolites of the selective androgen receptor modulator andarine (S-4) for routine doping control purposes

2010 ◽  
Vol 24 (15) ◽  
pp. 2245-2254 ◽  
Author(s):  
Mario Thevis ◽  
Andreas Thomas ◽  
Gregor Fußhöller ◽  
Simon Beuck ◽  
Hans Geyer ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Urinary Metabolites ◽  
Mass Spectrometric ◽  
Doping Control ◽  
Selective Androgen Receptor Modulator ◽  
Receptor Modulator

Pharmacological characterization of AC-262536, a novel selective androgen receptor modulator

2008 ◽  
Vol 109 (1-2) ◽  
pp. 129-137 ◽  
Author(s):  
Fabrice Piu ◽  
Luis R. Gardell ◽  
Thomas Son ◽  
Nathalie Schlienger ◽  
Birgitte W. Lund ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Selective Androgen Receptor Modulator ◽  
Pharmacological Characterization ◽  
Receptor Modulator

Mass spectrometric characterization of urinary metabolites of the selective androgen receptor modulator S-22 to identify potential targets for routine doping controls

2011 ◽  
Vol 25 (15) ◽  
pp. 2187-2195 ◽  
Author(s):  
Mario Thevis ◽  
Andreas Thomas ◽  
Ines Möller ◽  
Hans Geyer ◽  
James T. Dalton ◽  
...  
Keyword(s):  
Androgen Receptor ◽  
Urinary Metabolites ◽  
Mass Spectrometric ◽  
Selective Androgen Receptor Modulator ◽  
Receptor Modulator
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