The Dopamine D2 Receptor Partial Agonist Antipsychotics, Aripiprazole, and Brexpiprazole

2021 ◽  
pp. 1-45
Author(s):  
Tetsuro Kikuchi ◽  
Kenji Maeda ◽  
Sakiko Yamada ◽  
Mikio Suzuki ◽  
Tsuyoshi Hirose ◽  
...  
Keyword(s):  
Dopamine D2 Receptor ◽  
Partial Agonist ◽  
D2 Receptor ◽  
Dopamine D2

scholarly journals Effects of 2-bromoterguride, a dopamine D2 receptor partial agonist, on cognitive dysfunction and social aversion in rats

2017 ◽  
Vol 235 (1) ◽  
pp. 99-108 ◽  
Author(s):  
Emilia Tarland ◽  
Robert T. Franke ◽  
Heidrun Fink ◽  
Heinz H. Pertz ◽  
Jan Brosda
Keyword(s):  
Cognitive Dysfunction ◽  
Dopamine D2 Receptor ◽  
Partial Agonist ◽  
D2 Receptor ◽  
Dopamine D2

Aplindore (DAB-452), a high affinity selective dopamine D2 receptor partial agonist

2006 ◽  
Vol 552 (1-3) ◽  
pp. 36-45 ◽  
Author(s):  
Julia N. Heinrich ◽  
Julie Brennan ◽  
Margaret H. Lai ◽  
Kelly Sullivan ◽  
Geoff Hornby ◽  
...  
Keyword(s):  
Dopamine D2 Receptor ◽  
Partial Agonist ◽  
D2 Receptor ◽  
High Affinity ◽  
Dopamine D2 ◽  
Selective Dopamine

The dopamine D2 receptor partial agonist aplindore improves motor deficits in MPTP-treated common marmosets alone and combined with l-dopa

2009 ◽  
Vol 117 (1) ◽  
pp. 55-67 ◽  
Author(s):  
Michael John Jackson ◽  
Terrance H. Andree ◽  
Matthew Hansard ◽  
Diane C. Hoffman ◽  
Mark R. Hurtt ◽  
...  
Keyword(s):  
Dopamine D2 Receptor ◽  
Partial Agonist ◽  
D2 Receptor ◽  
Motor Deficits ◽  
Common Marmosets ◽  
Dopamine D2

Pharmacology of aripiprazole, a novel antipsychotic: dopamine D2 receptor partial agonist

2004 ◽  
Vol 19 (3) ◽  
pp. 190
Author(s):  
Tetsuro Kikuchi ◽  
Stark Arlene ◽  
Frank Yocca ◽  
Yoshihiro Tadori ◽  
Tsuyoshi Hirose ◽  
...  
Keyword(s):  
Dopamine D2 Receptor ◽  
Partial Agonist ◽  
D2 Receptor ◽  
Dopamine D2 ◽  
Novel Antipsychotic

scholarly journals A Case of Hypersexuality in a Patient Receiving Aripiprazole for Schizophrenia

2021 ◽  
Vol 2021 ◽  
pp. 1-3
Author(s):  
Lakshmi Priya ◽  
Bini Moorthy
Keyword(s):  
Dopamine D2 Receptor ◽  
Partial Agonist ◽  
D2 Receptor ◽  
Agonist Activity ◽  
Partial Agonist Activity ◽  
Dopamine D2 ◽  
Compulsive Behaviors

Aripiprazole is an antipsychotic with partial agonist activity at the dopamine D2 receptor which may lead to compulsive behaviors including hypersexuality. The case presented is of a 24-year-old male with schizophrenia who developed hypersexuality symptoms after initiation of aripiprazole. Cessation of the aripiprazole led to a reduction in hypersexual behaviors. Clinicians should be aware of compulsive behaviors including hypersexuality with aripiprazole use and consider discontinuation of aripiprazole treatment in patients suffering from hypersexuality.

scholarly journals Effects of Dopamine D2 Receptor Partial Agonist Antipsychotic Aripiprazole on Dopamine Synthesis in Human Brain Measured by PET with L-[β-11C]DOPA

PLoS ONE ◽  
2012 ◽  
Vol 7 (9) ◽  
pp. e46488 ◽  
Author(s):  
Hiroshi Ito ◽  
Harumasa Takano ◽  
Ryosuke Arakawa ◽  
Hidehiko Takahashi ◽  
Fumitoshi Kodaka ◽  
...  
Keyword(s):  
Human Brain ◽  
Dopamine D2 Receptor ◽  
Partial Agonist ◽  
D2 Receptor ◽  
Dopamine Synthesis ◽  
Dopamine D2
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