Site-specific conjugation of a lanthanide chelator and its effects on the chemical synthesis and receptor binding affinity of human relaxin-2 hormone

Relaxin 2

Improved Chemical Synthesis and Demonstration of the Relaxin Receptor Binding Affinity and Biological Activity of Mouse Relaxin†

Biochemistry ◽

10.1021/bi700238h ◽

2007 ◽

Vol 46 (18) ◽

pp. 5374-5381 ◽

Cited By ~ 32

Author(s):

Chrishan S. Samuel ◽

Feng Lin ◽

Mohammed Akhter Hossain ◽

Chongxin Zhao ◽

Tania Ferraro ◽

...

Keyword(s):

Biological Activity ◽

Chemical Synthesis ◽

Binding Affinity ◽

Receptor Binding ◽

Relaxin Receptor

Antiproliferative and antiviral effects of mutated IFN-alpha with increased IFN receptor binding affinity

Zeitschrift für Gastroenterologie ◽

10.1055/s-0030-1269699 ◽

2011 ◽

Vol 49 (01) ◽

Author(s):

MF Sprinzl ◽

L Bührer ◽

D Strand ◽

G Schreiber ◽

PR Galle ◽

...

Keyword(s):

Binding Affinity ◽

Receptor Binding ◽

Ifn Alpha ◽

Antiviral Effects

Ring-substituted 1,1,2,2-tetraalkylated 1,2-bis(hydroxyphenyl)ethanes. 4. Synthesis, estrogen receptor binding affinity, and evaluation of antiestrogenic and mammary tumor inhibiting activity of symmetrically disubstituted 1,1,2,2-tetramethyl-1,2-bis(hydroxyphenyl)ethanes

10.1021/jm00147a031 ◽

1985 ◽

Vol 28 (9) ◽

pp. 1295-1301 ◽

Cited By ~ 16

Author(s):

Rolf W. Hartmann ◽

Walter Schwarz ◽

Alexander Heindl ◽

Helmut Schoenenberger

Keyword(s):

Estrogen Receptor ◽

Binding Affinity ◽

Receptor Binding ◽

Mammary Tumor ◽

Inhibiting Activity ◽

Estrogen Receptor Binding

Correction: Mouse IgG2c Fc loop residues promote greater receptor-binding affinity than mouse IgG2b or human IgG1

PLoS ONE ◽

10.1371/journal.pone.0196609 ◽

2018 ◽

Vol 13 (4) ◽

pp. e0196609

Author(s):

Keyword(s):

Binding Affinity ◽

Receptor Binding ◽

Human Igg1

Ring-substituted 1,2-dialkylated 1,2-bis(hydroxyphenyl)ethanes. 1. Synthesis and estrogen receptor binding affinity of 2,2'- and 3,3'-disubstituted hexestrols

10.1021/jm00362a010 ◽

1983 ◽

Vol 26 (8) ◽

pp. 1137-1144 ◽

Cited By ~ 14

Author(s):

Rolf W. Hartmann ◽

Walter Schwarz ◽

Helmut Schoenenberger

Keyword(s):

Estrogen Receptor ◽

Binding Affinity ◽

Receptor Binding ◽

Estrogen Receptor Binding

Bromine- and Iodine-Substituted 16α,17α-Dioxolane Progestins for Breast Tumor Imaging and Radiotherapy: Synthesis and Receptor Binding Affinity

10.1021/jm060348q ◽

2006 ◽

Vol 49 (15) ◽

pp. 4737-4744 ◽

Cited By ~ 14

Author(s):

Dong Zhou ◽

Kathryn E. Carlson ◽

John A. Katzenellenbogen ◽

Michael J. Welch

Keyword(s):

Binding Affinity ◽

Receptor Binding ◽

Breast Tumor ◽

Tumor Imaging ◽

[Aladan3]TIPP: A fluorescent ?-opioid antagonist with high ?-receptor binding affinity and ? selectivity

Biopolymers ◽

10.1002/bip.20200 ◽

2005 ◽

Vol 80 (2-3) ◽

pp. 325-331 ◽

Cited By ~ 17

Author(s):

Heru Chen ◽

Nga N. Chung ◽

Carole Lemieux ◽

Bogumil Zelent ◽

Jane M. Vanderkooi ◽

...

Keyword(s):

Binding Affinity ◽

Receptor Binding ◽

Opioid Antagonist ◽

Additional disulfide bonds in insulin: Prediction, recombinant expression, receptor binding affinity, and stability

Protein Science ◽

10.1002/pro.2649 ◽

2015 ◽

Vol 24 (5) ◽

pp. 779-788 ◽

Cited By ~ 9

Author(s):

Tine N. Vinther ◽

Ingrid Pettersson ◽

Kasper Huus ◽

Morten Schlein ◽

Dorte B. Steensgaard ◽

...

Keyword(s):

Binding Affinity ◽

Receptor Binding ◽

Disulfide Bonds ◽

Recombinant Expression ◽

Arginine-vasopressin analogs with high antidiuretic/vasopressor selectivity. Synthesis, biological activity and receptor binding affinity of arginine-vasopressin analogs with substitutions in positions 1, 2, 4, 7, and 8

10.1021/jm00151a016 ◽

1986 ◽

Vol 29 (1) ◽

pp. 96-99 ◽

Cited By ~ 8

Author(s):

Zbigniew Grzonka ◽

Franciszek Kasprzykowski ◽

Elzbieta Kojro ◽

Krzysztof Darlak ◽

Per Melin ◽

...

Keyword(s):

Biological Activity ◽

Binding Affinity ◽

Receptor Binding ◽

Arginine Vasopressin ◽

ChemInform Abstract: Synthesis and Receptor-Binding Affinity of Fluorotamoxifen, a Possible Estrogen-Receptor Imaging Agent.

Chemischer Informationsdienst ◽

10.1002/chin.198606130 ◽

1986 ◽

Vol 17 (6) ◽

Author(s):

J. SHANI ◽

A. GAZIT ◽

T. LIVSHITZ ◽

S. BIRAN

Keyword(s):

Estrogen Receptor ◽

Binding Affinity ◽

Receptor Binding ◽

Imaging Agent ◽

Receptor Imaging ◽