Synthesis of 16β-derivatives of 3-(2-bromoethyl)-estra-1,3,5(10)-trien-17β-ol as inhibitors of 17β-HSD1 and/or steroid sulfatase for the treatment of estrogen-dependent diseases

Steroids ◽  
2021 ◽  
pp. 108856
Author(s):  
Maxime Lespérance ◽  
Jenny Roy ◽  
Adrien Djiemeny Ngueta ◽  
René Maltais ◽  
Donald Poirier
Keyword(s):  
Steroid Sulfatase ◽  
Derivatives Of

Structure−Activity Relationships of 17α-Derivatives of Estradiol as Inhibitors of Steroid Sulfatase

2000 ◽  
Vol 43 (23) ◽  
pp. 4465-4478 ◽  
Author(s):  
Roch P. Boivin ◽  
Van Luu-The ◽  
Roger Lachance ◽  
Fernand Labrie ◽  
Donald Poirier
Keyword(s):  
Steroid Sulfatase ◽  
Structure Activity Relationships ◽  
Structure Activity ◽  
Derivatives Of

Synthesis and steroid sulfatase inhibitory activities of N-phosphorylated 3-(4-aminophenyl)-coumarin-7-O-sulfamates

MedChemComm ◽  
2016 ◽  
Vol 7 (6) ◽  
pp. 1146-1150 ◽  
Author(s):  
Mateusz Daśko ◽  
Maciej Masłyk ◽  
Konrad Kubiński ◽  
Justyna Aszyk ◽  
Janusz Rachon ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Steroid Sulfatase ◽  
Coumarin 7 ◽  
Inhibitory Activities ◽  
Synthesis And Biological Evaluation ◽  
Derivatives Of

In the present work, we report convenient methods for the synthesis and biological evaluation of N-phosphorylated derivatives of 3-(4-aminophenyl)-coumarin-7-O-sulfamate as potential steroid sulfatase (STS) inhibitors.

17α-Alkan (or alkyn) amide derivatives of estradiol as inhibitors of steroid-sulfatase activity

Steroids ◽  
1999 ◽  
Vol 64 (12) ◽  
pp. 825-833 ◽  
Author(s):  
Roch P Boivin ◽  
Fernand Labrie ◽  
Donald Poirier
Keyword(s):  
Steroid Sulfatase ◽  
Amide Derivatives ◽  
Sulfatase Activity ◽  
Derivatives Of

Sulfate derivatives of 2-phenylindols as novel steroid sulfatase inhibitors

1990 ◽  
Vol 39 (11) ◽  
pp. 1709-1713 ◽  
Author(s):  
Herbert Birnböck ◽  
Erwin von Angerer
Keyword(s):  
Steroid Sulfatase ◽  
Derivatives Of
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