Synthesis and pharmacological characterization of a new benzoxazole derivative as a potent 5-HT 3 receptor agonist

In Vitro Pharmacological Characterization of a Novel Selective α7 Neuronal Nicotinic Acetylcholine Receptor Agonist ABT-107

Journal of Pharmacology and Experimental Therapeutics ◽

10.1124/jpet.110.167072 ◽

2010 ◽

Vol 334 (3) ◽

pp. 863-874 ◽

Cited By ~ 40

Author(s):

John Malysz ◽

David J. Anderson ◽

Jens H. Grønlien ◽

Jianguo Ji ◽

William H. Bunnelle ◽

...

Keyword(s):

Acetylcholine Receptor ◽

Nicotinic Acetylcholine Receptor ◽

Receptor Agonist ◽

Neuronal Nicotinic Acetylcholine Receptor ◽

Nicotinic Acetylcholine

Pharmacological Characterization of PD151832, an M1 Muscarinic Receptor Agonist

Alzheimer Disease ◽

10.1007/978-1-4612-4116-4_46 ◽

1997 ◽

pp. 311-315

Author(s):

Roy D. Schwarz ◽

Michael J. Callahan ◽

Robert E. Davis ◽

Mark R. Emmerling ◽

Juan C. Jaen ◽

...

Keyword(s):

Muscarinic Receptor ◽

Receptor Agonist ◽

M1 Muscarinic

Pharmacological characterization of F-180: a selective human V1a vasopressin receptor agonist of high affinity

British Journal of Pharmacology ◽

10.1038/sj.bjp.0704634 ◽

2002 ◽

Vol 135 (7) ◽

pp. 1828-1836 ◽

Cited By ~ 21

Author(s):

Miriam Andrés ◽

Miguel Trueba ◽

Gilles Guillon

Keyword(s):

Receptor Agonist ◽

Vasopressin Receptor ◽

High Affinity

Pharmacological Characterization of a Novel 5-HT4 Receptor Agonist, TS-951, in vitro

Pharmacology ◽

10.1159/000056107 ◽

2001 ◽

Vol 63 (1) ◽

pp. 8-16 ◽

Cited By ~ 5

Author(s):

Sumiyo Kajita ◽

Chika Ito ◽

Reiko Kawamura ◽

Shoji Yasuda ◽

Yoshihiko Isobe ◽

...

Keyword(s):

Receptor Agonist ◽

Synthesis and pharmacological characterization of l-trans-4-tetrazolylproline (ly300020): A novel systemically-active ampa receptor agonist

Bioorganic & Medicinal Chemistry Letters ◽

10.1016/s0960-894x(00)80099-2 ◽

1993 ◽

Vol 3 (1) ◽

pp. 95-98 ◽

Cited By ~ 17

Author(s):

James A. Monn ◽

Matthew J. Valli ◽

Rebecca A. True ◽

Darryl D. Schoepp ◽

J.David Leander ◽

...

Keyword(s):

Ampa Receptor ◽

Receptor Agonist ◽

In vivo pharmacological characterization of the structurally novel, potent, selective mGlu2/3 receptor agonist LY404039 in animal models of psychiatric disorders

Psychopharmacology ◽

10.1007/s00213-007-0758-3 ◽

2007 ◽

Vol 193 (1) ◽

pp. 121-136 ◽

Cited By ~ 112

Author(s):

Linda M. Rorick-Kehn ◽

Bryan G. Johnson ◽

Karen M. Knitowski ◽

Craig R. Salhoff ◽

Jeffrey M. Witkin ◽

...

Keyword(s):

Animal Models ◽

Psychiatric Disorders ◽

Receptor Agonist ◽

ChemInform Abstract: Design, Synthesis, and Pharmacological Characterization of (+)-2- Aminobicyclo(3.1.0)hexane-2,6-dicarboxylic Acid (LY354740): A Potent, Selective, and Orally Active Group 2 Metabotropic Glutamate Receptor Agonist Possessing Anticonvul

ChemInform ◽

10.1002/chin.199722076 ◽

2010 ◽

Vol 28 (22) ◽

pp. no-no

Author(s):

J. A. MONN ◽

M. J. VALLI ◽

S. M. MASSEY ◽

R. A. WRIGHT ◽

C. R. SALHOFF ◽

...

Keyword(s):

Glutamate Receptor ◽

Receptor Agonist ◽

Metabotropic Glutamate Receptor ◽

Design Synthesis ◽

Metabotropic Glutamate ◽

Group 2 ◽

Glutamate Receptor Agonist ◽

Orally Active

Synthesis and Pharmacological Characterization of C4-Disubstituted Analogs of 1S,2S,5R,6S-2-Aminobicyclo[3.1.0]hexane-2,6-dicarboxylate: Identification of a Potent, Selective Metabotropic Glutamate Receptor Agonist and Determination of Agonist-Bound Human mGlu2 and mGlu3 Amino Terminal Domain Structures

Journal of Medicinal Chemistry ◽

10.1021/jm501612y ◽

2015 ◽

Vol 58 (4) ◽

pp. 1776-1794 ◽

Cited By ~ 42

Author(s):

James A. Monn ◽

Lourdes Prieto ◽

Lorena Taboada ◽

Concepcion Pedregal ◽

Junliang Hao ◽

...

Keyword(s):

Receptor Agonist ◽

Metabotropic Glutamate Receptor ◽

Metabotropic Glutamate ◽

Amino Terminal ◽

Domain Structures ◽

Glutamate Receptor Agonist ◽

Amino Terminal Domain

Synthesis and Pharmacological Characterization of Novel Analogues of the Nicotinic Acetylcholine Receptor Agonist (±)-UB-165

Journal of Medicinal Chemistry ◽

10.1021/jm020814l ◽

2002 ◽

Vol 45 (15) ◽

pp. 3235-3245 ◽

Cited By ~ 33

Author(s):

Christopher G. V. Sharples ◽

Gunter Karig ◽

Graham L. Simpson ◽

James A. Spencer ◽

Emma Wright ◽

...

Keyword(s):

Acetylcholine Receptor ◽

Nicotinic Acetylcholine Receptor ◽

Receptor Agonist ◽

Nicotinic Acetylcholine

Pharmacological characterization of a novel 5-HT4 receptor agonist, TS-951 in vitro.

The Japanese Journal of Pharmacology ◽

10.1016/s0021-5198(19)34836-x ◽

1999 ◽

Vol 79 ◽

pp. 206

Author(s):

Sumiyo Kajita ◽

Chika Ito ◽

Yoshihiko Isobe ◽

Kiyomi Fukushima

Keyword(s):

Receptor Agonist ◽