Mechanism-Based Discovery of Small Molecules that Prevent Noncompetitive Inhibition by Cocaine and MK-801 Mediated by Two Different Sites on the Nicotinic Acetylcholine Receptor†

Biochemistry ◽  
2004 ◽  
Vol 43 (31) ◽  
pp. 10149-10156 ◽  
Author(s):  
Yongli Chen ◽  
Anamitro Banerjee ◽  
George P. Hess
Keyword(s):  
Small Molecules ◽  
Acetylcholine Receptor ◽  
Nicotinic Acetylcholine Receptor ◽  
Nicotinic Acetylcholine ◽  
Mk 801 ◽  
Noncompetitive Inhibition

Interaction of MK-801 with the nicotinic acetylcholine receptor-associated ion channel from electroplax

1989 ◽  
Vol 164 (2) ◽  
pp. 397-398 ◽  
Author(s):  
M.P. Kavanaugh ◽  
B.A.C. Tester ◽  
E. Weber
Keyword(s):  
Ion Channel ◽  
Acetylcholine Receptor ◽  
Nicotinic Acetylcholine Receptor ◽  
Nicotinic Acetylcholine ◽  
Mk 801

Reversing the Action of Noncompetitive Inhibitors (MK-801 and Cocaine) on a Protein (Nicotinic Acetylcholine Receptor)-Mediated Reaction†

Biochemistry ◽  
2003 ◽  
Vol 42 (20) ◽  
pp. 6106-6114 ◽  
Author(s):  
George P. Hess ◽  
Armanda M. Gameiro ◽  
Ryan C. Schoenfeld ◽  
Yongli Chen ◽  
Henning Ulrich ◽  
...  
Keyword(s):  
Acetylcholine Receptor ◽  
Nicotinic Acetylcholine Receptor ◽  
Nicotinic Acetylcholine ◽  
Mk 801 ◽  
Noncompetitive Inhibitors

Effect of MK-801 at the human α7 nicotinic acetylcholine receptor

1996 ◽  
Vol 35 (4) ◽  
pp. 407-414 ◽  
Author(s):  
Clark A. Briggs ◽  
David G. McKenna
Keyword(s):  
Acetylcholine Receptor ◽  
Nicotinic Acetylcholine Receptor ◽  
Α7 Nicotinic Acetylcholine Receptor ◽  
Nicotinic Acetylcholine ◽  
Mk 801

scholarly journals Mechanism-based discovery of ligands that counteract inhibition of the nicotinic acetylcholine receptor by cocaine and MK-801

2000 ◽  
Vol 97 (25) ◽  
pp. 13895-13900 ◽  
Author(s):  
G. P. Hess ◽  
H. Ulrich ◽  
H.-G. Breitinger ◽  
L. Niu ◽  
A. M. Gameiro ◽  
...  
Keyword(s):  
Acetylcholine Receptor ◽  
Nicotinic Acetylcholine Receptor ◽  
Nicotinic Acetylcholine ◽  
Mk 801

MK-801 inhibition of nicotinic acetylcholine receptor channels

Synapse ◽  
1991 ◽  
Vol 7 (3) ◽  
pp. 207-215 ◽  
Author(s):  
Mariano Amador ◽  
John A. Dani
Keyword(s):  
Acetylcholine Receptor ◽  
Nicotinic Acetylcholine Receptor ◽  
Nicotinic Acetylcholine ◽  
Mk 801
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