Synthesis and biological evaluation of conformationally restricted 2-(1-pyrrolidinyl)-N-[2-(3,4-dichlorophenyl)ethyl]-N-methylethylenediamines as .sigma. receptor ligands. 1. Pyrrolidine, piperidine, homopiperidine, and tetrahydroisoquinoline classes

1992 ◽  
Vol 35 (23) ◽  
pp. 4334-4343 ◽  
Author(s):  
Brian R. De Costa ◽  
Celia Dominguez ◽  
Xiao Shu He ◽  
Wanda Williams ◽  
Lilian Radesca ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Sigma Receptor ◽  
Receptor Ligands ◽  
Conformationally Restricted ◽  
Sigma Receptor Ligands ◽  
Synthesis And Biological Evaluation

Novel conformationally restricted aromatic piperidines as selective sigma receptor ligands

1994 ◽  
Vol 4 (2) ◽  
pp. 329-334 ◽  
Author(s):  
Gary A. Cain ◽  
Thomas E. Christos ◽  
Charles J. Eyermann ◽  
Paul J. Gilligan ◽  
Dimitri E. Grigoriadis ◽  
...  
Keyword(s):  
Sigma Receptor ◽  
Receptor Ligands ◽  
Conformationally Restricted ◽  
Sigma Receptor Ligands

ChemInform Abstract: Novel Conformationally Restricted Aromatic Piperidines as Selective Sigma Receptor Ligands.

ChemInform ◽  
2010 ◽  
Vol 25 (27) ◽  
pp. no-no
Author(s):  
G. A. CAIN ◽  
T. E. CHRISTOS ◽  
C. J. EYERMANN ◽  
P. J. GILLIGAN ◽  
D. E. GRIGORIADIS ◽  
...  
Keyword(s):  
Sigma Receptor ◽  
Receptor Ligands ◽  
Conformationally Restricted ◽  
Sigma Receptor Ligands

Synthesis and biological evaluation of conformationally restricted σ1 receptor ligands with 7,9-diazabicyclo[4.2.2]decane scaffold

2010 ◽  
Vol 8 (24) ◽  
pp. 5525 ◽  
Author(s):  
Sunil K. Sunnam ◽  
Dirk Schepmann ◽  
Elisabeth Rack ◽  
Roland Fröhlich ◽  
Katharina Korpis ◽  
...  
Keyword(s):  
Biological Evaluation ◽  
Receptor Ligands ◽  
Conformationally Restricted ◽  
Σ1 Receptor ◽  
Synthesis And Biological Evaluation

scholarly journals Sigma Receptor Ligands Carrying a Nitric Oxide Donor Nitrate Moiety: Synthesis, In Silico, and Biological Evaluation

2020 ◽  
Vol 11 (5) ◽  
pp. 889-894
Author(s):  
Emanuele Amata ◽  
Maria Dichiara ◽  
Davide Gentile ◽  
Agostino Marrazzo ◽  
Rita Turnaturi ◽  
...  
Keyword(s):  
Nitric Oxide ◽  
In Silico ◽  
Biological Evaluation ◽  
Nitric Oxide Donor ◽  
Sigma Receptor ◽  
Receptor Ligands ◽  
Sigma Receptor Ligands

scholarly journals Recent Advances in the Development of Sigma Receptor Ligands as Cytotoxic Agents: A Medicinal Chemistry Perspective

2021 ◽  
Author(s):  
Antonino N. Fallica ◽  
Valeria Pittalà ◽  
Maria N. Modica ◽  
Loredana Salerno ◽  
Giuseppe Romeo ◽  
...  
Keyword(s):  
Medicinal Chemistry ◽  
Cytotoxic Agents ◽  
Sigma Receptor ◽  
Receptor Ligands ◽  
Sigma Receptor Ligands ◽  
Recent Advances

Design, synthesis and biological evaluation of piperazine analogues as CB1 cannabinoid receptor ligands

2008 ◽  
Vol 16 (7) ◽  
pp. 4035-4051 ◽  
Author(s):  
Kwang-Seop Song ◽  
Sung-Han Lee ◽  
Hyun Ji Chun ◽  
Jong Yup Kim ◽  
Myung Eun Jung ◽  
...  
Keyword(s):  
Cannabinoid Receptor ◽  
Biological Evaluation ◽  
Receptor Ligands ◽  
Design Synthesis ◽  
Cb1 Cannabinoid Receptor ◽  
Synthesis And Biological Evaluation

scholarly journals Effects of Acute Administration of Sigma Receptor Ligands on Mesolimbic Dopamine Neurotransmission in Rats

2009 ◽  
Vol 23 (S1) ◽  
Author(s):  
Gianluigi Tanda ◽  
Linda Garcés‐Ramírez ◽  
Jennifer L Green ◽  
Takato Hiranita ◽  
Jonathan L Katz
Keyword(s):  
Sigma Receptor ◽  
Acute Administration ◽  
Receptor Ligands ◽  
Mesolimbic Dopamine ◽  
Sigma Receptor Ligands
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